4MQM
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![BU of 4mqm by Molmil](/molmil-images/mine/4mqm) | Crystal structure of Antigen 85C in presence of Ebselen | 分子名称: | Diacylglycerol acyltransferase/mycolyltransferase Ag85C | 著者 | Favrot, L, Grzegorzewicz, A.E, Lajiness, D.H, Marvin, R.K, Boucau, J, Isailovic, D, Jackson, M, Ronning, D.R. | 登録日 | 2013-09-16 | 公開日 | 2013-11-13 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.346 Å) | 主引用文献 | Mechanism of inhibition of Mycobacterium tuberculosis antigen 85 by ebselen. Nat Commun, 4, 2013
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5VNS
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![BU of 5vns by Molmil](/molmil-images/mine/5vns) | M.tb Antigen 85C Acyl-Enzyme Intermediate with Tetrahydrolipstatin | 分子名称: | (2S,3S,5S)-5-[(N-FORMYL-L-LEUCYL)OXY]-2-HEXYL-3-HYDROXYHEXADECANOIC ACID, (4S)-2-METHYL-2,4-PENTANEDIOL, Diacylglycerol acyltransferase/mycolyltransferase Ag85C, ... | 著者 | Goins, C.M, Ronning, D.R. | 登録日 | 2017-05-01 | 公開日 | 2018-01-24 | 最終更新日 | 2019-12-11 | 実験手法 | X-RAY DIFFRACTION (1.45 Å) | 主引用文献 | Mycolyltransferase fromMycobacterium tuberculosisin covalent complex with tetrahydrolipstatin provides insights into antigen 85 catalysis. J. Biol. Chem., 293, 2018
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5WAS
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5W95
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![BU of 5w95 by Molmil](/molmil-images/mine/5w95) | Mtb Rv3802c with PEG bound | 分子名称: | Conserved membrane protein of uncharacterised function, PENTAETHYLENE GLYCOL | 著者 | Goins, C.M, Schreidah, C.M, Ronning, D.R. | 登録日 | 2017-06-22 | 公開日 | 2017-12-27 | 最終更新日 | 2019-12-11 | 実験手法 | X-RAY DIFFRACTION (1.723 Å) | 主引用文献 | Structural basis for lipid binding and mechanism of the Mycobacterium tuberculosis Rv3802 phospholipase. J. Biol. Chem., 293, 2018
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4QDT
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4OJT
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4QDO
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4QDU
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4QE3
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![BU of 4qe3 by Molmil](/molmil-images/mine/4qe3) | Crystal structure of Antigen 85C-H260Q mutant | 分子名称: | ACETIC ACID, CHAPSO, Diacylglycerol acyltransferase/mycolyltransferase Ag85C | 著者 | Favrot, L, Lajiness, D.H, Ronning, D.R. | 登録日 | 2014-05-15 | 公開日 | 2014-07-09 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.351 Å) | 主引用文献 | Inactivation of the Mycobacterium tuberculosis Antigen 85 Complex by Covalent, Allosteric Inhibitors. J.Biol.Chem., 289, 2014
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4QDX
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4QDZ
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![BU of 4qdz by Molmil](/molmil-images/mine/4qdz) | Crystal structure of Antigen 85C-E228Q mutant | 分子名称: | ACETATE ION, Diacylglycerol acyltransferase/mycolyltransferase Ag85C, HEXAETHYLENE GLYCOL | 著者 | Favrot, L, Lajiness, D.H, Ronning, D.R. | 登録日 | 2014-05-14 | 公開日 | 2014-07-09 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.885 Å) | 主引用文献 | Inactivation of the Mycobacterium tuberculosis Antigen 85 Complex by Covalent, Allosteric Inhibitors. J.Biol.Chem., 289, 2014
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7S3E
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9FQ2
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![BU of 9fq2 by Molmil](/molmil-images/mine/9fq2) | Poliovirus 3C protease in H32 spacegroup | 分子名称: | Protease 3C | 著者 | Fairhead, M, Lithgo, R.M, MacLean, E.M, Bowesman-Jones, H, Aschenbrenner, J.C, Balcomb, B.H, Capkin, E, Chandran, A.V, Godoy, A.S, Marples, P.G, Fearon, D, von Delft, F, Koekemoer, L. | 登録日 | 2024-06-14 | 公開日 | 2024-06-26 | 実験手法 | X-RAY DIFFRACTION (2.37 Å) | 主引用文献 | Poliovirus 3C protease in H32 spacegroup To Be Published
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1RZ9
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![BU of 1rz9 by Molmil](/molmil-images/mine/1rz9) | Crystal Structure of AAV Rep complexed with the Rep-binding sequence | 分子名称: | 26-MER, Rep protein | 著者 | Hickman, A.B, Ronning, D.R, Perez, Z.N, Kotin, R.M, Dyda, F. | 登録日 | 2003-12-24 | 公開日 | 2004-02-17 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | The nuclease domain of adeno-associated virus rep coordinates replication initiation using two distinct DNA recognition interfaces. Mol.Cell, 13, 2004
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9FWC
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![BU of 9fwc by Molmil](/molmil-images/mine/9fwc) | Coxsackievirus B3 3C protease in C121 spacegroup | 分子名称: | Genome polyprotein | 著者 | Fairhead, M, Lithgo, R.M, MacLean, E.M, Bowesman-Jones, H, Aschenbrenner, J.C, Balcomb, B.H, Capkin, E, Chandran, A.V, Godoy, A.S, Marples, P.G, Fearon, D, von Delft, F, Koekemoer, L. | 登録日 | 2024-06-28 | 公開日 | 2024-07-10 | 実験手法 | X-RAY DIFFRACTION (1.34 Å) | 主引用文献 | Coxsackievirus B3 3C protease in C121 spacegroup To Be Published
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9FS7
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![BU of 9fs7 by Molmil](/molmil-images/mine/9fs7) | Coxsackievirus A16 3C protease in C2 2 21 spacegroup | 分子名称: | Genome polyprotein | 著者 | Fairhead, M, Lithgo, R, MacLean, M, Bowesman-Jones, H, Aschenbrenner, J.C, Balcomb, B.H, Capkin, E, Chandran, A.V, Godoy, A.S, Marples, P.G, Fearon, D, von Delft, F, Koekemoer, L. | 登録日 | 2024-06-20 | 公開日 | 2024-07-10 | 実験手法 | X-RAY DIFFRACTION (1.37 Å) | 主引用文献 | Coxsackievirus A16 3C protease in C2 2 21 spacegroup To Be Published
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5CCE
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![BU of 5cce by Molmil](/molmil-images/mine/5cce) | Joint X-ray/neutron structure of wild type MTAN complexed with SRH and adenine | 分子名称: | 5'-Methylthioadenosine Nucleosidase, ADENINE, S-ribosylhomocysteine, ... | 著者 | Banco, M.T, Kovalevsky, A.Y, Ronning, D.R. | 登録日 | 2015-07-02 | 公開日 | 2016-11-16 | 最終更新日 | 2023-09-27 | 実験手法 | NEUTRON DIFFRACTION (2.5 Å), X-RAY DIFFRACTION | 主引用文献 | Neutron structures of the Helicobacter pylori 5'-methylthioadenosine nucleosidase highlight proton sharing and protonation states. Proc. Natl. Acad. Sci. U.S.A., 113, 2016
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5CCD
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7MEL
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![BU of 7mel by Molmil](/molmil-images/mine/7mel) | Sco GlgEI-V279S in complex with 4-alpha-glucoside of validamine | 分子名称: | (1R,2R,3S,4S,6R)-4-amino-2,3-dihydroxy-6-(hydroxymethyl)cyclohexyl alpha-D-glucopyranoside, 1,2-ETHANEDIOL, Alpha-1,4-glucan:maltose-1-phosphate maltosyltransferase 1, ... | 著者 | Jayasinghe, T.D, Ronning, D.R. | 登録日 | 2021-04-06 | 公開日 | 2021-07-14 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | Stereoselective synthesis of a 4-alpha-glucoside of valienamine and its X-ray structure in complex with Streptomyces coelicolor GlgE1-V279S. Sci Rep, 11, 2021
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7MYG
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![BU of 7myg by Molmil](/molmil-images/mine/7myg) | M. tb Ag85C modified by THL-10d | 分子名称: | Diacylglycerol acyltransferase, GLYCEROL | 著者 | Sudasinghe, T.D, Ronning, D.R. | 登録日 | 2021-05-21 | 公開日 | 2021-09-15 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.51 Å) | 主引用文献 | Total Synthesis of Tetrahydrolipstatin, Its Derivatives, and Evaluation of Their Ability to Potentiate Multiple Antibiotic Classes against Mycobacterium Species. Acs Infect Dis., 7, 2021
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8F5V
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7MGY
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![BU of 7mgy by Molmil](/molmil-images/mine/7mgy) | Sco GlgEI-V279S in complex with 4-alpha-glucoside of valienamine | 分子名称: | (1R,4S,5S,6R)-4-amino-5,6-dihydroxy-2-(hydroxymethyl)cyclohex-2-en-1-yl alpha-D-glucopyranoside, Alpha-1,4-glucan:maltose-1-phosphate maltosyltransferase 1, DI(HYDROXYETHYL)ETHER, ... | 著者 | Jayasinghe, T.D, Ronning, D.R. | 登録日 | 2021-04-13 | 公開日 | 2021-07-14 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.83 Å) | 主引用文献 | Stereoselective synthesis of a 4-⍺-glucoside of valienamine and its X-ray structure in complex with Streptomyces coelicolor GlgE1-V279S. Sci Rep, 11, 2021
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8D6K
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![BU of 8d6k by Molmil](/molmil-images/mine/8d6k) | Sco GlgEI-V279S in complex with cyclohexyl carbasugar | 分子名称: | (1R,4S,5S,6R)-4-(cyclohexylamino)-5,6-dihydroxy-2-(hydroxymethyl)cyclohex-2-en-1-yl alpha-D-glucopyranoside, Alpha-1,4-glucan:maltose-1-phosphate maltosyltransferase 1, DI(HYDROXYETHYL)ETHER | 著者 | Jayasinghe, T.J, Ronning, D.R. | 登録日 | 2022-06-06 | 公開日 | 2022-10-19 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.73 Å) | 主引用文献 | Synthesis of C 7 /C 8 -cyclitols and C 7 N-aminocyclitols from maltose and X-ray crystal structure of Streptomyces coelicolor GlgEI V279S in a complex with an amylostatin GXG-like derivative. Front Chem, 10, 2022
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8FFF
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8F2L
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