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PDB: 4 件
3LOK
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BU of 3lok by Molmil
Drug resistant cSrc kinase domain in complex with covalent inhibitor PD168393
分子名称: N-[4-(3-BROMO-PHENYLAMINO)-QUINAZOLIN-6-YL]-ACRYLAMIDE, Proto-oncogene tyrosine-protein kinase Src
著者Gruetter, C, Rode, H.B, Rauh, D.
登録日2010-02-04
公開日2010-12-22
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (2.48 Å)
主引用文献Characterization of irreversible kinase inhibitors by directly detecting covalent bond formation: a tool for dissecting kinase drug resistance
Chembiochem, 11, 2010
2QLQ
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BU of 2qlq by Molmil
Crystal structure of SRC kinase domain with covalent inhibitor RL3
分子名称: (2E)-N-{4-[(3-bromophenyl)amino]quinazolin-6-yl}-4-(dimethylamino)but-2-enamide, Proto-oncogene tyrosine-protein kinase Src
著者Michalczyk, A, Rode, H.B, Gruetter, C, Rauh, D.
登録日2007-07-13
公開日2008-03-11
最終更新日2021-10-20
実験手法X-RAY DIFFRACTION (2.33 Å)
主引用文献Structural insights into how irreversible inhibitors can overcome drug resistance in EGFR.
Bioorg.Med.Chem., 16, 2008
2QI8
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BU of 2qi8 by Molmil
Crystal structure of drug resistant SRC kinase domain
分子名称: GLYCEROL, Proto-oncogene tyrosine-protein kinase Src
著者Michalczyk, A, Rode, H.B, Gruetter, C, Rauh, D.
登録日2007-07-03
公開日2008-03-18
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.32 Å)
主引用文献Structural insights into how irreversible inhibitors can overcome drug resistance in EGFR.
Bioorg.Med.Chem., 16, 2008
2QQ7
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BU of 2qq7 by Molmil
Crystal structure of drug resistant SRC kinase domain with irreversible inhibitor
分子名称: (2E)-N-{4-[(3-bromophenyl)amino]quinazolin-6-yl}-4-(dimethylamino)but-2-enamide, Proto-oncogene tyrosine-protein kinase Src
著者Michalczyk, A, Rode, H.B, Gruetter, C, Rauh, D.
登録日2007-07-26
公開日2008-03-11
最終更新日2021-10-20
実験手法X-RAY DIFFRACTION (2.38 Å)
主引用文献Structural insights into how irreversible inhibitors can overcome drug resistance in EGFR.
Bioorg.Med.Chem., 16, 2008

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件を2024-09-11に公開中

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