Loading
PDBj
English日本語简体中文繁體中文한국어
✖
ﾒﾆｭｰPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help
PDB: 7 件
6CMJ
DownloadVisualize
BU of 6cmj by Molmil
Human CAMKK2 with GSK650393
分子名称: 1,2-ETHANEDIOL, 2-(2-methylpropyl)-4-(5-phenyl-1H-pyrrolo[2,3-b]pyridin-3-yl)benzoic acid, Calcium/calmodulin-dependent protein kinase kinase 2, ...
著者Williams, S.P, Reid, R.A, Price, D.J, Drewry, D.H.
登録日2018-03-05
公開日2018-04-04
最終更新日2018-05-16
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献An orally available, brain-penetrant CAMKK2 inhibitor reduces food intake in rodent model.
Bioorg. Med. Chem. Lett., 28, 2018
5WAV
DownloadVisualize
BU of 5wav by Molmil
Fc AbVance: Increasing our knowledge of antibody structural space to enable faster and better decision-making in antibody drug discovery.
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-3)-[2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-6)]alpha-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, GLYCEROL, Immunoglobulin gamma-1 heavy chain,Immunoglobulin gamma-1 heavy chain
著者Williams, S.P, Reid, R.A, Convery, M.A.
登録日2017-06-27
公開日2017-11-08
最終更新日2024-10-23
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献AbVance: Increasing our knowledge of antibody structural space to enable faster and better decision-making in antibody drug discovery.
To Be Published
3DDU
DownloadVisualize
BU of 3ddu by Molmil
Prolyl Oligopeptidase with GSK552
分子名称: (6S)-1-chloro-3-[(4-fluorobenzyl)oxy]-6-(pyrrolidin-1-ylcarbonyl)pyrrolo[1,2-a]pyrazin-4(6H)-one, ACETATE ION, GLYCEROL, ...
著者Madauss, K.P, Reid, R.A, Haffner, C.D, Miller, A.B.
登録日2008-06-06
公開日2008-08-19
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.56 Å)
主引用文献Pyrrolidinyl pyridone and pyrazinone analogues as potent inhibitors of prolyl oligopeptidase (POP)
Bioorg.Med.Chem.Lett., 18, 2008
7SZQ
DownloadVisualize
BU of 7szq by Molmil
Human P300 complexed with an azaindazole inhibitor
分子名称: 1-[1-(4-chlorophenyl)cyclopentane-1-carbonyl]-N-1H-pyrazolo[4,3-b]pyridin-5-yl-D-prolinamide, Histone acetyltransferase p300
著者Shewchuk, L.M, Reid, R.A.
登録日2021-11-29
公開日2022-11-09
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Discovery of Proline-Based p300/CBP Inhibitors Using DNA-Encoded Library Technology in Combination with High-Throughput Screening.
J.Med.Chem., 65, 2022
7SSK
DownloadVisualize
BU of 7ssk by Molmil
Human P300 complexed with a glycine-based inhibitor
分子名称: 1,2-ETHANEDIOL, ACETATE ION, Histone acetyltransferase p300, ...
著者Shewchuk, L.M, Reid, R.A.
登録日2021-11-11
公開日2022-11-09
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.36 Å)
主引用文献Discovery of Proline-Based p300/CBP Inhibitors Using DNA-Encoded Library Technology in Combination with High-Throughput Screening.
J.Med.Chem., 65, 2022
7SS8
DownloadVisualize
BU of 7ss8 by Molmil
Human P300 complexed with a proline-based inhibitor
分子名称: 1,2-ETHANEDIOL, 1-[1-(4-chlorophenyl)cyclopentane-1-carbonyl]-N-{[3-(methylcarbamoyl)phenyl]methyl}-D-prolinamide, Histone acetyltransferase p300, ...
著者Shewchuk, L.M, Reid, R.A.
登録日2021-11-10
公開日2022-11-09
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献Discovery of Proline-Based p300/CBP Inhibitors Using DNA-Encoded Library Technology in Combination with High-Throughput Screening.
J.Med.Chem., 65, 2022
5WAW
DownloadVisualize
BU of 5waw by Molmil
FcAbVance: Increasing our knowledge of antibody structural space to enable faster and better decision-making in antibody drug discovery
分子名称: GLYCEROL, ZINC ION, fAb Heavy Chain, ...
著者Williams, S.P, Reid, R.A, Convery, M.
登録日2017-06-27
公開日2017-11-08
最終更新日2019-05-22
実験手法X-RAY DIFFRACTION (2.25 Å)
主引用文献AbVance: Increasing our knowledge of antibody structural space to enable faster and better decision-making in antibody drug discovery.
Not Published

226707

件を2024-10-30に公開中

PDB statisticsPDBj update infoContact PDBjnumon