6NCJ
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![BU of 6ncj by Molmil](/molmil-images/mine/6ncj) | Structure of HIV-1 Integrase with potent 5,6,7,8-Tetrahydro-1,6-naphthyridine Derivatives Allosteric Site Inhibitors | 分子名称: | (2~{S})-2-[4-(8-fluoranyl-5-methyl-3,4-dihydro-2~{H}-chromen-6-yl)-2-methyl-6-[[(1~{S},2~{R})-2-phenylcyclopropyl]methyl]-7,8-dihydro-5~{H}-1,6-naphthyridin-3-yl]-2-[(2-methylpropan-2-yl)oxy]ethanoic acid, 1,2-ETHANEDIOL, Integrase, ... | 著者 | Nolte, R.T. | 登録日 | 2018-12-11 | 公開日 | 2019-01-16 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | 5,6,7,8-Tetrahydro-1,6-naphthyridine Derivatives as Potent HIV-1-Integrase-Allosteric-Site Inhibitors. J. Med. Chem., 62, 2019
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6P2H
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6CIH
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![BU of 6cih by Molmil](/molmil-images/mine/6cih) | Crystal structure of a group II intron lariat in the post-catalytic state | 分子名称: | IRIDIUM HEXAMMINE ION, MAGNESIUM ION, RNA (5'-R(P*UP*GP*UP*UP*UP*AP*UP*UP*AP*AP*AP*AP*AP*C*-3'), ... | 著者 | Chan, R.T, Peters, J.K, Robart, A.R, Wiryaman, T, Rajashankar, K.R, Toor, N. | 登録日 | 2018-02-23 | 公開日 | 2018-11-21 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (3.676 Å) | 主引用文献 | Structural basis for the second step of group II intron splicing. Nat Commun, 9, 2018
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6DN2
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![BU of 6dn2 by Molmil](/molmil-images/mine/6dn2) | CRYSTAL STRUCTURE OF THE FMN RIBOSWITCH BOUND TO BRX1354 SPLIT RNA | 分子名称: | 4-{benzyl[2-(7,8-dimethyl-2,4-dioxo-3,4-dihydrobenzo[g]pteridin-10(2H)-yl)ethyl]amino}butanoic acid, MAGNESIUM ION, POTASSIUM ION, ... | 著者 | Vicens, Q, Mondragon, E, Reyes, F.E, Berman, J, Kaur, H, Kells, K, Wickens, P, Wilson, J, Gadwood, R, Schostarez, H, Suto, R.K, Coish, P, Blount, K.F, Batey, R.T. | 登録日 | 2018-06-05 | 公開日 | 2018-09-05 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (2.88 Å) | 主引用文献 | Structure-Activity Relationship of Flavin Analogues That Target the Flavin Mononucleotide Riboswitch. ACS Chem. Biol., 13, 2018
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6DN3
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![BU of 6dn3 by Molmil](/molmil-images/mine/6dn3) | CRYSTAL STRUCTURE OF THE FMN RIBOSWITCH BOUND TO BRX1555 SPLIT RNA | 分子名称: | 7,8-dimethyl-2,4-dioxo-10-(3-phenylpropyl)-1,2,3,4-tetrahydrobenzo[g]pteridin-10-ium, CHLORIDE ION, MAGNESIUM ION, ... | 著者 | Vicens, Q, Mondragon, E, Reyes, F.E, Berman, J, Kaur, H, Kells, K, Wickens, P, Wilson, J, Gadwood, R, Schostarez, H, Suto, R.K, Coish, P, Blount, K.F, Batey, R.T. | 登録日 | 2018-06-05 | 公開日 | 2018-09-05 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Structure-Activity Relationship of Flavin Analogues That Target the Flavin Mononucleotide Riboswitch. ACS Chem. Biol., 13, 2018
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6DKQ
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![BU of 6dkq by Molmil](/molmil-images/mine/6dkq) | Crystal structure of the Shr Hemoglobin Interacting Domain 2 | 分子名称: | Heme-binding protein Shr, SULFATE ION | 著者 | Macdonald, R, Cascio, D, Collazo, M.J, Clubb, R.T. | 登録日 | 2018-05-30 | 公開日 | 2018-10-24 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | The Streptococcus pyogenes Shr protein captures human hemoglobin using two structurally unique binding domains. J.Biol.Chem., 293, 2018
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6DN1
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![BU of 6dn1 by Molmil](/molmil-images/mine/6dn1) | CRYSTAL STRUCTURE OF THE FMN RIBOSWITCH BOUND TO BRX1151 SPLIT RNA | 分子名称: | 10-(6-carboxyhexyl)-8-(cyclopentylamino)-2,4-dihydroxy-7-methylbenzo[g]pteridin-10-ium, MAGNESIUM ION, POTASSIUM ION, ... | 著者 | Vicens, Q, Mondragon, E, Reyes, F.E, Berman, J, Kaur, H, Kells, K, Wickens, P, Wilson, J, Gadwood, R, Schostarez, H, Suto, R.K, Coish, P, Blount, K.F, Batey, R.T. | 登録日 | 2018-06-05 | 公開日 | 2018-09-05 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (3.03 Å) | 主引用文献 | Structure-Activity Relationship of Flavin Analogues That Target the Flavin Mononucleotide Riboswitch. ACS Chem. Biol., 13, 2018
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6WR2
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6WRF
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![BU of 6wrf by Molmil](/molmil-images/mine/6wrf) | ClpX-ClpP complex bound to GFP-ssrA, recognition complex | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, ATP-dependent Clp protease ATP-binding subunit ClpX, ATP-dependent Clp protease proteolytic subunit, ... | 著者 | Fei, X, Sauer, R.T. | 登録日 | 2020-04-29 | 公開日 | 2020-11-04 | 最終更新日 | 2024-03-06 | 実験手法 | ELECTRON MICROSCOPY (3.14 Å) | 主引用文献 | Structural basis of ClpXP recognition and unfolding of ssrA-tagged substrates. Elife, 9, 2020
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6WSG
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5WB4
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![BU of 5wb4 by Molmil](/molmil-images/mine/5wb4) | Crystal structure of the TarA wall teichoic acid glycosyltransferase | 分子名称: | N-acetylglucosaminyldiphosphoundecaprenol N-acetyl-beta-D-mannosaminyltransferase, SULFATE ION | 著者 | Kattke, M.D, Cascio, D, Sawaya, M.R, Clubb, R.T. | 登録日 | 2017-06-27 | 公開日 | 2019-01-16 | 最終更新日 | 2019-07-31 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Structure and mechanism of TagA, a novel membrane-associated glycosyltransferase that produces wall teichoic acids in pathogenic bacteria. Plos Pathog., 15, 2019
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5WFG
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![BU of 5wfg by Molmil](/molmil-images/mine/5wfg) | Crystal structure of the TarA wall teichoic acid glycosyltransferase bound to UDP | 分子名称: | N-acetylglucosaminyldiphosphoundecaprenol N-acetyl-beta-D-mannosaminyltransferase, URIDINE-5'-DIPHOSPHATE | 著者 | Kattke, M.D, Cascio, D, Sawaya, M.R, Clubb, R.T. | 登録日 | 2017-07-11 | 公開日 | 2019-01-16 | 最終更新日 | 2019-07-31 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | Structure and mechanism of TagA, a novel membrane-associated glycosyltransferase that produces wall teichoic acids in pathogenic bacteria. Plos Pathog., 15, 2019
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8P1I
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![BU of 8p1i by Molmil](/molmil-images/mine/8p1i) | Single particle cryo-EM co-structure of Klebsiella pneumoniae AcrB with the BDM91288 efflux pump inhibitor at 2.97 Angstrom resolution | 分子名称: | 1,2-DIOCTANOYL-SN-GLYCERO-3-[PHOSPHO-RAC-(1-GLYCEROL), 3-chloranyl-2,6-di(piperazin-4-ium-1-yl)quinoline, Efflux pump membrane transporter, ... | 著者 | Boernsen, C, Mueller, R.T, Pos, K.M, Frangakis, A.S. | 登録日 | 2023-05-12 | 公開日 | 2024-01-17 | 最終更新日 | 2024-01-31 | 実験手法 | ELECTRON MICROSCOPY (2.97 Å) | 主引用文献 | Pyridylpiperazine efflux pump inhibitor boosts in vivo antibiotic efficacy against K. pneumoniae. Embo Mol Med, 16, 2024
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6PP7
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![BU of 6pp7 by Molmil](/molmil-images/mine/6pp7) | ClpX in ClpX-ClpP complex bound to substrate and ATP-gamma-S, class 2 | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, ATP-dependent Clp protease ATP-binding subunit ClpX, PHOSPHOTHIOPHOSPHORIC ACID-ADENYLATE ESTER, ... | 著者 | Fei, X, Jenni, S, Harrison, S.C, Sauer, R.T. | 登録日 | 2019-07-05 | 公開日 | 2020-03-11 | 最終更新日 | 2024-03-20 | 実験手法 | ELECTRON MICROSCOPY (4.05 Å) | 主引用文献 | Structures of the ATP-fueled ClpXP proteolytic machine bound to protein substrate. Elife, 9, 2020
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6POD
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![BU of 6pod by Molmil](/molmil-images/mine/6pod) | ClpX-ClpP complex bound to substrate and ATP-gamma-S, class 2 | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, ATP-dependent Clp protease ATP-binding subunit ClpX, ATP-dependent Clp protease proteolytic subunit, ... | 著者 | Fei, X, Jenni, S, Harrison, S.C, Sauer, R.T. | 登録日 | 2019-07-03 | 公開日 | 2020-03-11 | 最終更新日 | 2024-03-20 | 実験手法 | ELECTRON MICROSCOPY (4.05 Å) | 主引用文献 | Structures of the ATP-fueled ClpXP proteolytic machine bound to protein substrate. Elife, 9, 2020
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6PP5
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![BU of 6pp5 by Molmil](/molmil-images/mine/6pp5) | ClpX in ClpX-ClpP complex bound to substrate and ATP-gamma-S, class 4 | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, ATP-dependent Clp protease ATP-binding subunit ClpX, PHOSPHOTHIOPHOSPHORIC ACID-ADENYLATE ESTER, ... | 著者 | Fei, X, Jenni, S, Harrison, S.C, Sauer, R.T. | 登録日 | 2019-07-05 | 公開日 | 2020-03-11 | 最終更新日 | 2024-03-20 | 実験手法 | ELECTRON MICROSCOPY (3.98 Å) | 主引用文献 | Structures of the ATP-fueled ClpXP proteolytic machine bound to protein substrate. Elife, 9, 2020
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6PO3
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![BU of 6po3 by Molmil](/molmil-images/mine/6po3) | ClpX-ClpP complex bound to substrate and ATP-gamma-S, class 3 | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, ATP-dependent Clp protease ATP-binding subunit ClpX, ATP-dependent Clp protease proteolytic subunit, ... | 著者 | Fei, X, Jenni, S, Harrison, S.C, Sauer, R.T. | 登録日 | 2019-07-03 | 公開日 | 2020-03-11 | 最終更新日 | 2024-03-20 | 実験手法 | ELECTRON MICROSCOPY (4.28 Å) | 主引用文献 | Structures of the ATP-fueled ClpXP proteolytic machine bound to protein substrate. Elife, 9, 2020
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6PPE
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![BU of 6ppe by Molmil](/molmil-images/mine/6ppe) | ClpP and ClpX IGF loop in ClpX-ClpP complex with D7 symmetry | 分子名称: | ATP-dependent Clp protease ATP-binding subunit ClpX, ATP-dependent Clp protease proteolytic subunit | 著者 | Fei, X, Jenni, S, Harrison, S.C, Sauer, R.T. | 登録日 | 2019-07-06 | 公開日 | 2020-03-11 | 最終更新日 | 2024-03-20 | 実験手法 | ELECTRON MICROSCOPY (3.19 Å) | 主引用文献 | Structures of the ATP-fueled ClpXP proteolytic machine bound to protein substrate. Elife, 9, 2020
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6POS
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![BU of 6pos by Molmil](/molmil-images/mine/6pos) | ClpX-ClpP complex bound to substrate and ATP-gamma-S, class 1 | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, ATP-dependent Clp protease ATP-binding subunit ClpX, ATP-dependent Clp protease proteolytic subunit, ... | 著者 | Fei, X, Jenni, S, Harrison, S.C, Sauer, R.T. | 登録日 | 2019-07-05 | 公開日 | 2020-03-11 | 実験手法 | ELECTRON MICROSCOPY (4.12 Å) | 主引用文献 | Structures of the ATP-fueled ClpXP proteolytic machine bound to protein substrate. Elife, 9, 2020
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6PO1
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![BU of 6po1 by Molmil](/molmil-images/mine/6po1) | ClpX-ClpP complex bound to substrate and ATP-gamma-S, class 4 | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, ATP-dependent Clp protease ATP-binding subunit ClpX, ATP-dependent Clp protease proteolytic subunit, ... | 著者 | Fei, X, Jenni, S, Harrison, S.C, Sauer, R.T. | 登録日 | 2019-07-03 | 公開日 | 2020-03-11 | 最終更新日 | 2024-03-20 | 実験手法 | ELECTRON MICROSCOPY (4.2 Å) | 主引用文献 | Structures of the ATP-fueled ClpXP proteolytic machine bound to protein substrate. Elife, 9, 2020
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6PP8
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![BU of 6pp8 by Molmil](/molmil-images/mine/6pp8) | ClpX in ClpX-ClpP complex bound to substrate and ATP-gamma-S, class 1 | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, ATP-dependent Clp protease ATP-binding subunit ClpX, PHOSPHOTHIOPHOSPHORIC ACID-ADENYLATE ESTER, ... | 著者 | Fei, X, Jenni, S, Harrison, S.C, Sauer, R.T. | 登録日 | 2019-07-05 | 公開日 | 2020-03-11 | 実験手法 | ELECTRON MICROSCOPY (4.12 Å) | 主引用文献 | Structures of the ATP-fueled ClpXP proteolytic machine bound to protein substrate. Elife, 9, 2020
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6PP6
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![BU of 6pp6 by Molmil](/molmil-images/mine/6pp6) | ClpX in ClpX-ClpP complex bound to substrate and ATP-gamma-S, class 3 | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, ATP-dependent Clp protease ATP-binding subunit ClpX, PHOSPHOTHIOPHOSPHORIC ACID-ADENYLATE ESTER, ... | 著者 | Fei, X, Jenni, S, Harrison, S.C, Sauer, R.T. | 登録日 | 2019-07-05 | 公開日 | 2020-03-11 | 最終更新日 | 2024-03-20 | 実験手法 | ELECTRON MICROSCOPY (4.28 Å) | 主引用文献 | Structures of the ATP-fueled ClpXP proteolytic machine bound to protein substrate. Elife, 9, 2020
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6PXI
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![BU of 6pxi by Molmil](/molmil-images/mine/6pxi) | The crystal structure of a singly capped HslUV complex with an axial pore plug and a HslU E257Q mutation | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, ATP-dependent protease ATPase subunit HslU, ATP-dependent protease subunit HslV, ... | 著者 | Baytshtok, V, Grant, R.A, Sauer, R.T. | 登録日 | 2019-07-26 | 公開日 | 2020-07-29 | 最終更新日 | 2024-06-19 | 実験手法 | X-RAY DIFFRACTION (3.447 Å) | 主引用文献 | Heat activates the AAA+ HslUV protease by melting an axial autoinhibitory plug. Cell Rep, 34, 2021
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6PVU
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![BU of 6pvu by Molmil](/molmil-images/mine/6pvu) | RNase A in complex with hexametaphosphate | 分子名称: | 2,4,6,8,10,12-hexahydroxy-2lambda~5~,4lambda~5~,6lambda~5~,8lambda~5~,10lambda~5~,12lambda~5~-cyclohexaphosphoxane-2,4,6,8,10,12-hexone, Ribonuclease pancreatic | 著者 | Windsor, I.W, Sheppard, S.M, Cummins, C.C, Raines, R.T. | 登録日 | 2019-07-21 | 公開日 | 2019-11-06 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (1.49 Å) | 主引用文献 | Nucleoside Tetra- and Pentaphosphates Prepared Using a Tetraphosphorylation Reagent Are Potent Inhibitors of Ribonuclease A. J.Am.Chem.Soc., 141, 2019
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6PVW
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![BU of 6pvw by Molmil](/molmil-images/mine/6pvw) | RNase A in complex with cp4pA | 分子名称: | 2,4,6,8-tetrahydroxy-1,3,5,7,2lambda~5~,4lambda~5~,6lambda~5~,8lambda~5~-tetroxatetraphosphocane-2,4,6,8-tetrone, 5'-O-[(R)-hydroxy{[(4R,8S)-4,6,8-trihydroxy-2,4,6,8-tetraoxo-1,3,5,7,2lambda~5~,4lambda~5~,6lambda~5~,8lambda~5~-tetroxatetraphosphocan-2-yl]oxy}phosphoryl]adenosine, Ribonuclease pancreatic | 著者 | Windsor, I.W, Sheppard, S.M, Cummins, C.C, Raines, R.T. | 登録日 | 2019-07-21 | 公開日 | 2019-11-06 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Nucleoside Tetra- and Pentaphosphates Prepared Using a Tetraphosphorylation Reagent Are Potent Inhibitors of Ribonuclease A. J.Am.Chem.Soc., 141, 2019
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