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PDB: 1559 件

5S8Q
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XChem group deposition -- Crystal Structure of the second bromodomain of pleckstrin homology domain interacting protein (PHIP) in complex with FMO3D000185a (space group P212121)
分子名称: (3R)-3-methyl-1,2,3,4-tetrahydro-5H-1,4-benzodiazepin-5-one, 1,2-ETHANEDIOL, CALCIUM ION, ...
著者Krojer, T, Talon, R, Fairhead, M, Szykowska, A, Burgess-Brown, N.A, Brennan, P.E, Arrowsmith, C.H, Edwards, A.M, Bountra, C, von Delft, F.
登録日2020-12-17
公開日2021-01-13
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献XChem group deposition
To Be Published
5S8C
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XChem group deposition -- Crystal Structure of the second bromodomain of pleckstrin homology domain interacting protein (PHIP) in complex with N00322e (space group C2)
分子名称: (1-methylbenzotriazol-5-yl)methanol, PH-interacting protein
著者Krojer, T, Talon, R, Fairhead, M, Szykowska, A, Burgess-Brown, N.A, Brennan, P.E, Arrowsmith, C.H, Edwards, A.M, Bountra, C, von Delft, F.
登録日2020-12-17
公開日2021-01-13
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (1.25 Å)
主引用文献XChem group deposition
To Be Published
5S8L
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XChem group deposition -- Crystal Structure of the second bromodomain of pleckstrin homology domain interacting protein (PHIP) in complex with E11289c (space group C2)
分子名称: 1-METHYLQUINOLIN-2(1H)-ONE, PH-interacting protein
著者Krojer, T, Talon, R, Fairhead, M, Szykowska, A, Burgess-Brown, N.A, Brennan, P.E, Arrowsmith, C.H, Edwards, A.M, Bountra, C, von Delft, F.
登録日2020-12-17
公開日2021-01-13
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (1.23 Å)
主引用文献XChem group deposition
To Be Published
5S8F
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XChem group deposition -- Crystal Structure of the second bromodomain of pleckstrin homology domain interacting protein (PHIP) in complex with N00572d (space group C2)
分子名称: PH-interacting protein, ~{N}-(5-oxidanylidene-7,8-dihydro-6~{H}-naphthalen-2-yl)ethanamide
著者Krojer, T, Talon, R, Fairhead, M, Szykowska, A, Burgess-Brown, N.A, Brennan, P.E, Arrowsmith, C.H, Edwards, A.M, Bountra, C, von Delft, F.
登録日2020-12-17
公開日2021-01-13
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (1.18 Å)
主引用文献XChem group deposition
To Be Published
5S8P
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XChem group deposition -- Crystal Structure of the second bromodomain of pleckstrin homology domain interacting protein (PHIP) in complex with E07179c (space group P212121)
分子名称: 1,2-ETHANEDIOL, 3-methyl-3,4-dihydroquinazolin-2(1H)-one, CALCIUM ION, ...
著者Krojer, T, Talon, R, Fairhead, M, Szykowska, A, Burgess-Brown, N.A, Brennan, P.E, Arrowsmith, C.H, Edwards, A.M, Bountra, C, von Delft, F.
登録日2020-12-17
公開日2021-01-13
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (1.41 Å)
主引用文献XChem group deposition
To Be Published
5U7G
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BU of 5u7g by Molmil
Crystal Structure of the Catalytic Core of CBP
分子名称: CREB-binding protein, ZINC ION
著者Park, S, Stanfield, R.L, Martinez-Yamout, M.M, Dyson, H.J, Wilson, I.A, Wright, P.E.
登録日2016-12-12
公開日2017-06-21
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.401 Å)
主引用文献Role of the CBP catalytic core in intramolecular SUMOylation and control of histone H3 acetylation.
Proc. Natl. Acad. Sci. U.S.A., 114, 2017
5SBM
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BU of 5sbm by Molmil
CD44 PanDDA analysis group deposition -- The hyaluronan-binding domain of CD44 in complex with Z1267885772
分子名称: (3S)-3-methyl-1-(6-methylpyridin-2-yl)piperazine, 1,2-ETHANEDIOL, CD44 antigen, ...
著者Bradshaw, W.J, Katis, V.L, Bezerra, G.A, Koekemoer, L, von Delft, F, Bountra, C, Brennan, P.E, Gileadi, O.
登録日2021-09-14
公開日2021-09-22
実験手法X-RAY DIFFRACTION (1.14 Å)
主引用文献CD44 PanDDA analysis group deposition
To Be Published
5SBN
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BU of 5sbn by Molmil
CD44 PanDDA analysis group deposition -- The hyaluronan-binding domain of CD44 in complex with Z57040482
分子名称: 1,2-ETHANEDIOL, CD44 antigen, DIMETHYL SULFOXIDE, ...
著者Bradshaw, W.J, Katis, V.L, Bezerra, G.A, Koekemoer, L, von Delft, F, Bountra, C, Brennan, P.E, Gileadi, O.
登録日2021-09-14
公開日2021-09-22
実験手法X-RAY DIFFRACTION (1.181 Å)
主引用文献CD44 PanDDA analysis group deposition
To Be Published
5SBL
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CD44 PanDDA analysis group deposition -- The hyaluronan-binding domain of CD44 in complex with Z126932614
分子名称: 1,2-ETHANEDIOL, 2-[(methylsulfonyl)methyl]-1H-benzimidazole, CD44 antigen, ...
著者Bradshaw, W.J, Katis, V.L, Bezerra, G.A, Koekemoer, L, von Delft, F, Bountra, C, Brennan, P.E, Gileadi, O.
登録日2021-09-14
公開日2021-09-22
実験手法X-RAY DIFFRACTION (1.198 Å)
主引用文献CD44 PanDDA analysis group deposition
To Be Published
5SBK
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BU of 5sbk by Molmil
CD44 PanDDA analysis group deposition -- The hyaluronan-binding domain of CD44 in complex with Z1258992717
分子名称: 1,2-ETHANEDIOL, CD44 antigen, DIMETHYL SULFOXIDE, ...
著者Bradshaw, W.J, Katis, V.L, Bezerra, G.A, Koekemoer, L, von Delft, F, Bountra, C, Brennan, P.E, Gileadi, O.
登録日2021-09-14
公開日2021-09-22
実験手法X-RAY DIFFRACTION (1.23 Å)
主引用文献CD44 PanDDA analysis group deposition
To Be Published
5SBO
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BU of 5sbo by Molmil
CD44 PanDDA analysis group deposition -- The hyaluronan-binding domain of CD44 in complex with Z2856434878
分子名称: 1,2-ETHANEDIOL, 4-[(3,4-dimethoxyphenyl)methyl]morpholine, CD44 antigen, ...
著者Bradshaw, W.J, Katis, V.L, Bezerra, G.A, Koekemoer, L, von Delft, F, Bountra, C, Brennan, P.E, Gileadi, O.
登録日2021-09-14
公開日2021-09-22
実験手法X-RAY DIFFRACTION (1.274 Å)
主引用文献CD44 PanDDA analysis group deposition
To Be Published
5SBP
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CD44 PanDDA analysis group deposition -- The hyaluronan-binding domain of CD44 in complex with Z1229798311
分子名称: 1,2-ETHANEDIOL, 2-acetamido-6-fluorobenzoic acid, CD44 antigen, ...
著者Bradshaw, W.J, Katis, V.L, Bezerra, G.A, Koekemoer, L, von Delft, F, Bountra, C, Brennan, P.E, Gileadi, O.
登録日2021-09-14
公開日2021-09-22
実験手法X-RAY DIFFRACTION (1.275 Å)
主引用文献CD44 PanDDA analysis group deposition
To Be Published
5SBQ
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CD44 PanDDA analysis group deposition -- The hyaluronan-binding domain of CD44 in complex with Z44592329
分子名称: CD44 antigen, DIMETHYL SULFOXIDE, N-phenyl-N'-pyridin-3-ylurea, ...
著者Bradshaw, W.J, Katis, V.L, Bezerra, G.A, Koekemoer, L, von Delft, F, Bountra, C, Brennan, P.E, Gileadi, O.
登録日2021-09-14
公開日2021-09-22
実験手法X-RAY DIFFRACTION (0.988 Å)
主引用文献CD44 PanDDA analysis group deposition
To Be Published
5SBR
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BU of 5sbr by Molmil
CD44 PanDDA analysis group deposition -- The hyaluronan-binding domain of CD44 in complex with Z1259341012
分子名称: (1R)-1-[4-(morpholin-4-yl)phenyl]ethan-1-amine, 1,2-ETHANEDIOL, CD44 antigen, ...
著者Bradshaw, W.J, Katis, V.L, Bezerra, G.A, Koekemoer, L, von Delft, F, Bountra, C, Brennan, P.E, Gileadi, O.
登録日2021-09-14
公開日2021-09-22
実験手法X-RAY DIFFRACTION (1.286 Å)
主引用文献CD44 PanDDA analysis group deposition
To Be Published
5SBT
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BU of 5sbt by Molmil
CD44 PanDDA analysis group deposition -- The hyaluronan-binding domain of CD44 in complex with Z445856640
分子名称: 1,2-ETHANEDIOL, CD44 antigen, DIMETHYL SULFOXIDE, ...
著者Bradshaw, W.J, Katis, V.L, Bezerra, G.A, Koekemoer, L, von Delft, F, Bountra, C, Brennan, P.E, Gileadi, O.
登録日2021-09-14
公開日2021-09-22
実験手法X-RAY DIFFRACTION (1.16 Å)
主引用文献CD44 PanDDA analysis group deposition
To Be Published
5SBU
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BU of 5sbu by Molmil
CD44 PanDDA analysis group deposition -- The hyaluronan-binding domain of CD44 in complex with Z839988838
分子名称: CD44 antigen, DIMETHYL SULFOXIDE, N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]cyclohexanamine, ...
著者Bradshaw, W.J, Katis, V.L, Bezerra, G.A, Koekemoer, L, von Delft, F, Bountra, C, Brennan, P.E, Gileadi, O.
登録日2021-09-14
公開日2021-09-22
実験手法X-RAY DIFFRACTION (1.044 Å)
主引用文献CD44 PanDDA analysis group deposition
To Be Published
5SBS
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BU of 5sbs by Molmil
CD44 PanDDA analysis group deposition -- The hyaluronan-binding domain of CD44 in complex with Z340495298
分子名称: 1,2-ETHANEDIOL, CD44 antigen, DIMETHYL SULFOXIDE, ...
著者Bradshaw, W.J, Katis, V.L, Bezerra, G.A, Koekemoer, L, von Delft, F, Bountra, C, Brennan, P.E, Gileadi, O.
登録日2021-09-14
公開日2021-09-22
実験手法X-RAY DIFFRACTION (1.024 Å)
主引用文献CD44 PanDDA analysis group deposition
To Be Published
5SBX
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BU of 5sbx by Molmil
CD44 PanDDA analysis group deposition -- The hyaluronan-binding domain of CD44 in complex with Z53825479
分子名称: 1,2-ETHANEDIOL, CD44 antigen, DI(HYDROXYETHYL)ETHER, ...
著者Bradshaw, W.J, Katis, V.L, Bezerra, G.A, Koekemoer, L, von Delft, F, Bountra, C, Brennan, P.E, Gileadi, O.
登録日2021-09-14
公開日2021-09-22
実験手法X-RAY DIFFRACTION (1.051 Å)
主引用文献CD44 PanDDA analysis group deposition
To Be Published
5SBW
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CD44 PanDDA analysis group deposition -- The hyaluronan-binding domain of CD44 in complex with Z2856434874
分子名称: 1,2-ETHANEDIOL, 1-{[4-(propan-2-yl)phenyl]methyl}piperidin-4-ol, CD44 antigen, ...
著者Bradshaw, W.J, Katis, V.L, Bezerra, G.A, Koekemoer, L, von Delft, F, Bountra, C, Brennan, P.E, Gileadi, O.
登録日2021-09-14
公開日2021-09-22
実験手法X-RAY DIFFRACTION (1.148 Å)
主引用文献CD44 PanDDA analysis group deposition
To Be Published
5SBV
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CD44 PanDDA analysis group deposition -- The hyaluronan-binding domain of CD44 in complex with Z31721798
分子名称: 1,2-ETHANEDIOL, 3-cyclohexyl-1-(morpholin-4-yl)propan-1-one, CD44 antigen, ...
著者Bradshaw, W.J, Katis, V.L, Bezerra, G.A, Koekemoer, L, von Delft, F, Bountra, C, Brennan, P.E, Gileadi, O.
登録日2021-09-14
公開日2021-09-22
実験手法X-RAY DIFFRACTION (1.109 Å)
主引用文献CD44 PanDDA analysis group deposition
To Be Published
5SBY
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BU of 5sby by Molmil
CD44 PanDDA analysis group deposition -- The hyaluronan-binding domain of CD44 in complex with Z1878656559
分子名称: (1R,2R)-2,4,4-trimethyl-N-[(1H-pyrazol-3-yl)methyl]cyclopentan-1-amine, 1,2-ETHANEDIOL, CD44 antigen, ...
著者Bradshaw, W.J, Katis, V.L, Bezerra, G.A, Koekemoer, L, von Delft, F, Bountra, C, Brennan, P.E, Gileadi, O.
登録日2021-09-14
公開日2021-09-22
実験手法X-RAY DIFFRACTION (1.217 Å)
主引用文献CD44 PanDDA analysis group deposition
To Be Published
5SBZ
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CD44 PanDDA analysis group deposition -- The hyaluronan-binding domain of CD44 in complex with Z768399682
分子名称: 1,2-ETHANEDIOL, CD44 antigen, DIMETHYL SULFOXIDE, ...
著者Bradshaw, W.J, Katis, V.L, Bezerra, G.A, Koekemoer, L, von Delft, F, Bountra, C, Brennan, P.E, Gileadi, O.
登録日2021-09-14
公開日2021-09-22
実験手法X-RAY DIFFRACTION (1.17 Å)
主引用文献CD44 PanDDA analysis group deposition
To Be Published
5SC0
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BU of 5sc0 by Molmil
CD44 PanDDA analysis group deposition -- The hyaluronan-binding domain of CD44 in complex with Z2856434899
分子名称: 1,2-ETHANEDIOL, 1-[(thiophen-3-yl)methyl]piperidin-4-ol, CD44 antigen, ...
著者Bradshaw, W.J, Katis, V.L, Bezerra, G.A, Koekemoer, L, von Delft, F, Bountra, C, Brennan, P.E, Gileadi, O.
登録日2021-09-14
公開日2021-09-22
実験手法X-RAY DIFFRACTION (1.192 Å)
主引用文献CD44 PanDDA analysis group deposition
To Be Published
5SC1
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BU of 5sc1 by Molmil
CD44 PanDDA analysis group deposition -- The hyaluronan-binding domain of CD44 in complex with Z431807512
分子名称: 1,2-ETHANEDIOL, CD44 antigen, DIMETHYL SULFOXIDE, ...
著者Bradshaw, W.J, Katis, V.L, Bezerra, G.A, Koekemoer, L, von Delft, F, Bountra, C, Brennan, P.E, Gileadi, O.
登録日2021-09-14
公開日2021-09-22
実験手法X-RAY DIFFRACTION (1.165 Å)
主引用文献CD44 PanDDA analysis group deposition
To Be Published
5SC2
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CD44 PanDDA analysis group deposition -- The hyaluronan-binding domain of CD44 in complex with Z190780124
分子名称: (3S)-N-[(1R)-1-cyclopropylethyl]-2-oxo-2,3-dihydropyridine-3-carboxamide, 1,2-ETHANEDIOL, CD44 antigen, ...
著者Bradshaw, W.J, Katis, V.L, Bezerra, G.A, Koekemoer, L, von Delft, F, Bountra, C, Brennan, P.E, Gileadi, O.
登録日2021-09-14
公開日2021-09-22
実験手法X-RAY DIFFRACTION (1.208 Å)
主引用文献CD44 PanDDA analysis group deposition
To Be Published

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件を2024-07-24に公開中

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