PDB Search results for query - Protein Data Bank Japan

PDB: 3 results

NR2F6 ligand binding domain in complex with NSD1 peptide
Descriptor:	Histone-lysine N-methyltransferase, H3 lysine-36 specific, Maltose/maltodextrin-binding periplasmic protein,Nuclear receptor subfamily 2 group F member 6, ...
Authors:	Oerlemans, G.J.M, van den Oetelaar, M.C.M, Brunsveld, L.
Deposit date:	2023-01-09
Release date:	2024-01-10
Method:	X-RAY DIFFRACTION (2.6 Å)
Cite:	Structural insights into coregulator recruitment to the autorepressed NR2F6 nuclear receptor To Be Published

ROR(gamma)t ligand binding domain in complex with allosteric ligand FM216
Descriptor:	4-[[3-[2-chloranyl-6-(trifluoromethyl)phenyl]-5-(1~{H}-pyrrol-3-yl)-1,2-oxazol-4-yl]methoxy]-2-fluoranyl-benzoic acid, Nuclear receptor ROR-gamma
Authors:	Oerlemans, G.J.M, Somsen, B.A, de Vries, R.M.J.M, Meijer, F.A, Brunsveld, L.
Deposit date:	2021-02-26
Release date:	2021-06-02
Last modified:	2024-01-31
Method:	X-RAY DIFFRACTION (1.55 Å)
Cite:	Structure-Activity Relationship Studies of Trisubstituted Isoxazoles as Selective Allosteric Ligands for the Retinoic-Acid-Receptor-Related Orphan Receptor gamma t. J.Med.Chem., 64, 2021

ROR(gamma)t ligand binding domain in complex with allosteric ligand FM257
Descriptor:	4-[[3-[2-chloranyl-6-(trifluoromethyl)phenyl]-5-(1~{H}-pyrazol-4-yl)-1,2-oxazol-4-yl]methoxy]benzoic acid, Nuclear receptor ROR-gamma
Authors:	Oerlemans, G.J.M, Somsen, B.A, de Vries, R.M.J.M, Meijer, F.A, Brunsveld, L.
Deposit date:	2021-02-26
Release date:	2021-06-02
Last modified:	2024-01-31
Method:	X-RAY DIFFRACTION (1.84 Å)
Cite:	Structure-Activity Relationship Studies of Trisubstituted Isoxazoles as Selective Allosteric Ligands for the Retinoic-Acid-Receptor-Related Orphan Receptor gamma t. J.Med.Chem., 64, 2021