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PDB: 2 results

7PWP
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BU of 7pwp by Molmil
PARP15 catalytic domain in complex with OUL221
Descriptor: 4-[(3-bromophenyl)methoxy]-2-methoxy-benzamide, DIMETHYL SULFOXIDE, Protein mono-ADP-ribosyltransferase PARP15
Authors:Maksimainen, M.M, Murthy, S, Nizi, M.G, Lehtio, L.
Deposit date:2021-10-07
Release date:2022-05-11
Last modified:2024-01-31
Method:X-RAY DIFFRACTION (2.1 Å)
Cite:Potent 2,3-dihydrophthalazine-1,4-dione derivatives as dual inhibitors for mono-ADP-ribosyltransferases PARP10 and PARP15.
Eur.J.Med.Chem., 237, 2022
7PWW
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BU of 7pww by Molmil
PARP15 catalytic domain in complex with OUL224
Descriptor: 6-[(3-bromophenyl)methoxy]phthalazine-1,4-dione, Protein mono-ADP-ribosyltransferase PARP15
Authors:Maksimainen, M.M, Murthy, S, Nizi, M.G, Lehtio, L.
Deposit date:2021-10-07
Release date:2022-05-11
Last modified:2024-01-31
Method:X-RAY DIFFRACTION (2.15 Å)
Cite:Potent 2,3-dihydrophthalazine-1,4-dione derivatives as dual inhibitors for mono-ADP-ribosyltransferases PARP10 and PARP15.
Eur.J.Med.Chem., 237, 2022

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