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PDB: 1 results

4BV3
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CRYSTAL STRUCTURE OF SIRT3 IN COMPLEX WITH THE INHIBITOR EX-527 AND NAD
Descriptor: (1S)-6-chloro-2,3,4,9-tetrahydro-1H-carbazole-1- carboxamide, ADENOSINE-5-DIPHOSPHORIBOSE, CHLORIDE ION, ...
Authors:Gertz, M, Nguyen, N.T.T, Weyand, M, Steegborn, C.
Deposit date:2013-06-24
Release date:2013-07-17
Last modified:2023-12-20
Method:X-RAY DIFFRACTION (2 Å)
Cite:Ex-527 Inhibits Sirtuins by Exploiting Their Unique Nad+-Dependent Deacetylation Mechanism
Proc.Natl.Acad.Sci.USA, 110, 2013

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