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PDB: 1 results

7CBX
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BU of 7cbx by Molmil
Crystal structure of MAP2K7 complexed with a covalent inhibitor 12
Descriptor: 3-(1H-indazol-3-yl)-5-(prop-2-enoylamino)-N-prop-2-ynyl-benzamide, Dual specificity mitogen-activated protein kinase kinase 7, GLYCEROL
Authors:Kinoshita, T, Murakawa, Y.
Deposit date:2020-06-15
Release date:2020-09-30
Last modified:2023-11-29
Method:X-RAY DIFFRACTION (2.061 Å)
Cite:Structural basis for producing selective MAP2K7 inhibitors.
Bioorg.Med.Chem.Lett., 30, 2020

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