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PDB: 2 results

8AV1
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BU of 8av1 by Molmil
Crystal structure of GSK3 beta (GSK3b) in complex with CD7.
Descriptor: 1,2-ETHANEDIOL, 2-pyridin-3-yl-8-thiomorpholin-4-yl-[1,3]oxazolo[5,4-f]quinoxaline, Glycogen synthase kinase-3 beta, ...
Authors:Chaikuad, A, Mongin, F, Knapp, S, Structural Genomics Consortium (SGC)
Deposit date:2022-08-26
Release date:2023-04-19
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (2.15 Å)
Cite:Oxazolo[5,4-f]quinoxaline-type selective inhibitors of glycogen synthase kinase-3 alpha (GSK-3 alpha ): Development and impact on temozolomide treatment of glioblastoma cells.
Bioorg.Chem., 134, 2023
8AUZ
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BU of 8auz by Molmil
Crystal structure of GSK3 beta (GSK3b) in complex with FL291.
Descriptor: 8-morpholin-4-yl-2-pyridin-3-yl-[1,3]oxazolo[5,4-f]quinoxaline, Glycogen synthase kinase-3 beta, SULFATE ION
Authors:Chaikuad, A, Mongin, F, Knapp, S, Structural Genomics Consortium (SGC)
Deposit date:2022-08-26
Release date:2023-04-19
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (2.66 Å)
Cite:Oxazolo[5,4-f]quinoxaline-type selective inhibitors of glycogen synthase kinase-3 alpha (GSK-3 alpha ): Development and impact on temozolomide treatment of glioblastoma cells.
Bioorg.Chem., 134, 2023

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PDB entries from 2024-07-10

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