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PDB: 8 件

8G2N
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Crystal structure of Tetrahymena thermophila G-rich DNA with novel ligand PyDH2
分子名称: 4,4'-{pyridine-2,6-diylbis[carbonyl-(1E)-hydrazin-2-yl-1-ylidene-(E)-methanylylidene]}bis(1-methylquinolin-1-ium), G-rich DNA, MAGNESIUM ION, ...
著者Martin, K.N, Yatsunyk, L.A.
登録日2023-02-06
公開日2024-02-14
実験手法X-RAY DIFFRACTION (1.33 Å)
主引用文献Crystal structure of Tetrahymena thermophila G-rich DNA with novel ligand PyDH2
To be published
7OQH
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CryoEM structure of the transcription termination factor Rho from Mycobacterium tuberculosis
分子名称: ADENOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, Transcription termination factor Rho
著者Saridakis, E, Vishwakarma, R, Lai Kee Him, J, Martin, K, Simon, I, Cohen-Gonsaud, M, Coste, F, Bron, P, Margeat, E, Boudvillain, M.
登録日2021-06-03
公開日2022-02-09
最終更新日2024-07-17
実験手法ELECTRON MICROSCOPY (3.32 Å)
主引用文献Cryo-EM structure of transcription termination factor Rho from Mycobacterium tuberculosis reveals bicyclomycin resistance mechanism.
Commun Biol, 5, 2022
2ZFC
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X-ray crystal structure of an engineered N-terminal HIV-1 GP41 trimer with enhanced stability and potency
分子名称: HIV-1 GP41
著者Dwyer, J.J, Wilson, K.L, Martin, K, Seedorff, J.E, Hasan, A, Kim, H.
登録日2007-12-29
公開日2008-04-22
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Design of an engineered N-terminal HIV-1 gp41 trimer with enhanced stability and potency
Protein Sci., 17, 2008
1VYW
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Structure of CDK2/Cyclin A with PNU-292137
分子名称: CELL DIVISION PROTEIN KINASE 2, CYCLIN A2, N-(3-CYCLOPROPYL-1H-PYRAZOL-5-YL)-2-(2-NAPHTHYL)ACETAMIDE, ...
著者Pevarello, P, Brasca, M.G, Amici, R, Orsini, P, Traquandi, G, Corti, L, Piutti, C, Sansonna, P, Villa, M, Pierce, B.S, Pulici, M, Giordano, P, Martina, K, Fritzen, E.L, Nugent, R.A, Casale, E, Cameron, A, Ciomei, M, Roletto, F, Isacchi, A, Fogliatto, G, Pesenti, E, Pastori, W, Marsiglio, A, Leach, K.L, Clare, P.M, Fiorentini, F, Varasi, M, Vulpetti, A, Warpehoski, M.A.
登録日2004-05-07
公開日2004-06-10
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献3-Aminopyrazole Inhibitors of Cdk2/Cyclin a as Antitumor Agents. Part 1. Lead Finding
J.Med.Chem., 47, 2004
1VYZ
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Structure of CDK2 complexed with PNU-181227
分子名称: CELL DIVISION PROTEIN KINASE 2, N-(5-CYCLOPROPYL-1H-PYRAZOL-3-YL)BENZAMIDE
著者Pevarello, P, Brasca, M.G, Amici, R, Orsini, P, Traquandi, G, Corti, L, Piutti, C, Sansonna, P, Villa, M, Pierce, B.S, Pulici, M, Giordano, G, Martina, K, Lfritzen, E, Nugent, R.A, Casale, E, Cameron, A, Ciomei, M, Roletto, F, Isacchi, A, Fogliatto, G, Pesenti, E, Pastori, W, Marsiglio, W, Leach, K.L, Clare, P.M, Fiorentini, F, Varasi, M, Vulpetti, A, Warpehoski, M.A.
登録日2004-05-07
公開日2004-06-17
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.21 Å)
主引用文献3-Aminopyrazole Inhibitors of Cdk2/Cyclin a as Antitumor Agents. 1. Lead Finding
J.Med.Chem., 47, 2004
4EW1
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High resolution structure of human glycinamide ribonucleotide transformylase in apo form.
分子名称: PHOSPHATE ION, SULFATE ION, Trifunctional purine biosynthetic protein adenosine-3
著者Connelly, S, DeMartino, K, Boger, D.L, Wilson, I.A.
登録日2012-04-26
公開日2013-07-31
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.522 Å)
主引用文献Biological and Structural Evaluation of 10R- and 10S-Methylthio-DDACTHF Reveals a New Role for Sulfur in Inhibition of Glycinamide Ribonucleotide Transformylase.
Biochemistry, 52, 2013
4EW2
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The structure of human glycinamide ribonucleotide transformylase in complex with 10S-methylthio-DDATHF.
分子名称: N-({4-[(1S)-4-(2,4-diamino-6-oxo-1,6-dihydropyrimidin-5-yl)-1-(methylsulfanyl)butyl]phenyl}carbonyl)-L-glutamic acid, PHOSPHATE ION, SULFATE ION, ...
著者Connelly, S, DeMartino, K, Boger, D.L, Wilson, I.A.
登録日2012-04-26
公開日2013-07-31
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.602 Å)
主引用文献Biological and Structural Evaluation of 10R- and 10S-Methylthio-DDACTHF Reveals a New Role for Sulfur in Inhibition of Glycinamide Ribonucleotide Transformylase.
Biochemistry, 52, 2013
4EW3
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The structure of human glycinamide ribonucleotide transformylase in complex with 10R-methylthio-DDATHF.
分子名称: N-({4-[(1R)-4-(2,4-diamino-6-oxo-1,6-dihydropyrimidin-5-yl)-1-(methylsulfanyl)butyl]phenyl}carbonyl)-L-glutamic acid, PHOSPHATE ION, SULFATE ION, ...
著者Connelly, S, DeMartino, K, Boger, D.L, Wilson, I.A.
登録日2012-04-26
公開日2013-07-31
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.702 Å)
主引用文献Biological and Structural Evaluation of 10R- and 10S-Methylthio-DDACTHF Reveals a New Role for Sulfur in Inhibition of Glycinamide Ribonucleotide Transformylase.
Biochemistry, 52, 2013

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件を2024-07-24に公開中

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