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PDB: 1 件

8JF5
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BU of 8jf5 by Molmil
Crystal structure of Lysine Specific Demethylase 1 (LSD1) with TAS1440
分子名称: 4-[5-[(3~{R})-3-azanylpyrrolidin-1-yl]carbonyl-2-[2-fluoranyl-4-(2-methyl-2-oxidanyl-propyl)phenyl]phenyl]-2-fluoranyl-benzenecarbonitrile, FLAVIN-ADENINE DINUCLEOTIDE, GLYCEROL, ...
著者Fukushima, H, Machida, T, Yamashita, S, Suzuki, T.
登録日2023-05-17
公開日2024-05-22
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献TAS1440, a histone H3 competitive LSD1 inhibitor, activates both TGF-beta and notch signaling pathways via INSM1 dissociation in neuroendocrine small cell lung cancer
To Be Published

222415

件を2024-07-10に公開中

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