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PDB: 249 件

5GWN
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Crystal structure of human RCC2
分子名称: Protein RCC2, SULFATE ION
著者Liang, L, Yun, C.H, Yin, Y.X.
登録日2016-09-12
公開日2017-09-13
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.309 Å)
主引用文献RCC2 is a novel p53 target in suppressing metastasis.
Oncogene, 37, 2018
1S5Y
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BU of 1s5y by Molmil
The crystal structure of Trematomus bernacchii hemoglobin oxidized by ferricyanide
分子名称: Hemoglobin alpha chain, Hemoglobin beta chain, PROTOPORPHYRIN IX CONTAINING FE
著者Vitagliano, L, Bonomi, G, Riccio, A, di Prisco, G, Smulevich, G, Mazzarella, L.
登録日2004-01-22
公開日2004-05-04
最終更新日2017-10-11
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献The oxidation process of Antarctic fish hemoglobins
Eur.J.Biochem., 271, 2004
1S5X
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The crystal structure of Trematomus bernacchii hemoglobin oxidized by air
分子名称: Hemoglobin alpha chain, Hemoglobin beta chain, PROTOPORPHYRIN IX CONTAINING FE
著者Vitagliano, L, Bonomi, G, Riccio, A, di Prisco, G, Smulevich, G, Mazzarella, L.
登録日2004-01-22
公開日2004-05-04
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献The oxidation process of Antarctic fish hemoglobins
Eur.J.Biochem., 271, 2004
5XDP
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BU of 5xdp by Molmil
K11/48-branched teraubiquitin
分子名称: D-ubiquitin, ubiquitin-B
著者Liang, L, Gao, S, Tang, S.
登録日2017-03-28
公開日2017-04-19
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.376 Å)
主引用文献K11/48-branched teraubiquitin
To Be Published
3RDC
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BU of 3rdc by Molmil
Human Cyclophilin D Complexed with an Inhibitor
分子名称: Peptidyl-prolyl cis-trans isomerase F, mitochondrial, ethyl N-[(4-aminobenzyl)carbamoyl]glycinate
著者Colliandre, L, Ahmed-Belkacem, H, Bessin, Y, Pawlotsky, J.M, Guichou, J.F.
登録日2011-04-01
公開日2012-03-21
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.94 Å)
主引用文献Combining 'dry' co-crystallization and in situ diffraction to facilitate ligand screening by X-ray crystallography.
Acta Crystallogr.,Sect.D, 71, 2015
1SKQ
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BU of 1skq by Molmil
The crystal structure of Sulfolobus solfataricus elongation factor 1-alpha in complex with magnesium and GDP
分子名称: Elongation factor 1-alpha, GUANOSINE-5'-DIPHOSPHATE, MAGNESIUM ION
著者Vitagliano, L, Ruggiero, A, Masullo, M, Cantiello, P, Arcari, P, Zagari, A.
登録日2004-03-05
公開日2004-07-20
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献The crystal structure of Sulfolobus solfataricus elongation factor 1alpha in complex with magnesium and GDP.
Biochemistry, 43, 2004
3QYU
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Crystal structure of human cyclophilin D at 1.54 A resolution at room temperature
分子名称: Peptidyl-prolyl cis-trans isomerase F
著者Colliandre, L, Gelin, M, Labesse, G, Guichou, J.-F.
登録日2011-03-04
公開日2011-08-24
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.54 Å)
主引用文献In-plate protein crystallization, in situ ligand soaking and X-ray diffraction.
Acta Crystallogr.,Sect.D, 67, 2011
7WM2
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Cryo-EM structure of AKT1
分子名称: (2S)-3-(hexadecanoyloxy)-2-[(9Z)-octadec-9-enoyloxy]propyl 2-(trimethylammonio)ethyl phosphate, POTASSIUM ION, Potassium channel AKT1
著者Dongliang, L, Zijie, Z, Yannan, Q, Yuyue, T, Huaizong, S.
登録日2022-01-14
公開日2023-01-25
最終更新日2024-06-26
実験手法ELECTRON MICROSCOPY (2.69 Å)
主引用文献Structural basis for the regulation mechanism of a hyperpolarization-activated K+ channel AKT1 by AtKC1
To Be Published
7WM1
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Cryo-EM structure of AKT1-AtKC1
分子名称: (2S)-3-(hexadecanoyloxy)-2-[(9Z)-octadec-9-enoyloxy]propyl 2-(trimethylammonio)ethyl phosphate, POTASSIUM ION, Potassium channel AKT1, ...
著者Dongliang, L, Zijie, Z, Yannan, Q, Yuyue, T, Huaizong, S.
登録日2022-01-14
公開日2023-01-25
最終更新日2024-06-26
実験手法ELECTRON MICROSCOPY (2.8 Å)
主引用文献Structural basis for the regulation mechanism of a hyper polarization-activated K+ channel AKT1 by AtKC1
To Be Published
3R4G
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BU of 3r4g by Molmil
Human Cyclophilin D Complexed with a Fragment
分子名称: 4-sulfamoylbenzoic acid, GLYCEROL, Peptidyl-prolyl cis-trans isomerase F, ...
著者Colliandre, L, Ahmed-Belkacem, H, Bessin, Y, Pawlotsky, J.M, Guichou, J.F.
登録日2011-03-17
公開日2012-03-21
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.05 Å)
主引用文献Fragment-based discovery of a new family of non-peptidic small-molecule cyclophilin inhibitors with potent antiviral activities.
Nat Commun, 7, 2016
3R57
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Human Cyclophilin D Complexed with a Fragment
分子名称: GLYCEROL, N-(3-aminophenyl)acetamide, Peptidyl-prolyl cis-trans isomerase F, ...
著者Colliandre, L, Ahmed-Belkacem, H, Bessin, Y, Pawlotsky, J.M, Guichou, J.F.
登録日2011-03-18
公開日2012-03-21
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.71 Å)
主引用文献Fragment-based discovery of a new family of non-peptidic small-molecule cyclophilin inhibitors with potent antiviral activities.
Nat Commun, 7, 2016
3RCF
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Human cyclophilin D complexed with N-[(4-aminophenyl)sulfonyl]benzamide
分子名称: N-[(4-aminophenyl)sulfonyl]benzamide, Peptidyl-prolyl cis-trans isomerase F, mitochondrial
著者Colliandre, L, Ahmed-Belkacem, H, Bessin, Y, Pawlotsky, J.M, Guichou, J.F.
登録日2011-03-31
公開日2012-03-21
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.15 Å)
主引用文献Fragment-based discovery of a new family of non-peptidic small-molecule cyclophilin inhibitors with potent antiviral activities.
Nat Commun, 7, 2016
3RCL
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Human Cyclophilin D Complexed with a Fragment
分子名称: 3-(1,3-oxazol-5-yl)aniline, O-ACETALDEHYDYL-HEXAETHYLENE GLYCOL, Peptidyl-prolyl cis-trans isomerase F, ...
著者Colliandre, L, Ahmed-Belkacem, H, Bessin, Y, Pawlotsky, J.M, Guichou, J.F.
登録日2011-03-31
公開日2012-03-21
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Fragment-based discovery of a new family of non-peptidic small-molecule cyclophilin inhibitors with potent antiviral activities.
Nat Commun, 7, 2016
3R49
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Human cyclophilin D complexed with quinolin-8-amine
分子名称: Peptidyl-prolyl cis-trans isomerase F, mitochondrial, quinolin-8-amine
著者Colliandre, L, Ahmed-Belkacem, H, Bessin, Y, Pawlotsky, J.M, Guichou, J.F.
登録日2011-03-17
公開日2012-03-21
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.77 Å)
主引用文献Fragment-based discovery of a new family of non-peptidic small-molecule cyclophilin inhibitors with potent antiviral activities.
Nat Commun, 7, 2016
3RD9
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Human Cyclophilin D Complexed with a Fragment
分子名称: 3-(3-methyl-5-oxo-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide, DI(HYDROXYETHYL)ETHER, Peptidyl-prolyl cis-trans isomerase F, ...
著者Colliandre, L, Ahmed-Belkacem, H, Bessin, Y, Pawlotsky, J.M, Guichou, J.F.
登録日2011-04-01
公開日2012-03-21
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献Fragment-based discovery of a new family of non-peptidic small-molecule cyclophilin inhibitors with potent antiviral activities.
Nat Commun, 7, 2016
3R59
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Human Cyclophilin D Complexed with a Fragment
分子名称: 1-(3-aminophenyl)ethanone, Peptidyl-prolyl cis-trans isomerase F, mitochondrial
著者Colliandre, L, Ahmed-Belkacem, H, Bessin, Y, Pawlotsky, J.M, Guichou, J.F.
登録日2011-03-18
公開日2012-03-21
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.1 Å)
主引用文献Fragment-based discovery of a new family of non-peptidic small-molecule cyclophilin inhibitors with potent antiviral activities.
Nat Commun, 7, 2016
3RDB
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BU of 3rdb by Molmil
Human Cyclophilin D Complexed with a Fragment
分子名称: 3-[5-(chloromethyl)-1,2,4-oxadiazol-3-yl]aniline, O-ACETALDEHYDYL-HEXAETHYLENE GLYCOL, Peptidyl-prolyl cis-trans isomerase F, ...
著者Colliandre, L, Ahmed-Belkacem, H, Bessin, Y, Pawlotsky, J.M, Guichou, J.F.
登録日2011-04-01
公開日2012-03-21
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.55 Å)
主引用文献Fragment-based discovery of a new family of non-peptidic small-molecule cyclophilin inhibitors with potent antiviral activities.
Nat Commun, 7, 2016
3RDA
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BU of 3rda by Molmil
Human Cyclophilin D Complexed with a Fragment
分子名称: 3-methyl-1,2-oxazol-5-amine, Peptidyl-prolyl cis-trans isomerase F, mitochondrial
著者Colliandre, L, Ahmed-Belkacem, H, Bessin, Y, Pawlotsky, J.M, Guichou, J.F.
登録日2011-04-01
公開日2012-03-21
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.07 Å)
主引用文献Fragment-based discovery of a new family of non-peptidic small-molecule cyclophilin inhibitors with potent antiviral activities.
Nat Commun, 7, 2016
3R54
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Human Cyclophilin D Complexed with a Fragment
分子名称: Peptidyl-prolyl cis-trans isomerase F, mitochondrial, pyrrolidine-1-carbaldehyde
著者Colliandre, L, Ahmed-Belkacem, H, Bessin, Y, Pawlotsky, J.M, Guichou, J.F.
登録日2011-03-18
公開日2012-03-21
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.35 Å)
主引用文献Fragment-based discovery of a new family of non-peptidic small-molecule cyclophilin inhibitors with potent antiviral activities.
Nat Commun, 7, 2016
3RCK
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BU of 3rck by Molmil
Human Cyclophilin D Complexed with a Fragment
分子名称: Peptidyl-prolyl cis-trans isomerase F, mitochondrial, piperazine-1-carbaldehyde
著者Colliandre, L, Ahmed-Belkacem, H, Bessin, Y, Pawlotsky, J.M, Guichou, J.F.
登録日2011-03-31
公開日2012-03-21
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.26 Å)
主引用文献Fragment-based discovery of a new family of non-peptidic small-molecule cyclophilin inhibitors with potent antiviral activities.
Nat Commun, 7, 2016
3R56
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Human Cyclophilin D Complexed with a Fragment
分子名称: 1H-indazol-6-amine, 3,6,9,12,15,18-HEXAOXAICOSANE-1,20-DIOL, Peptidyl-prolyl cis-trans isomerase F, ...
著者Colliandre, L, Ahmed-Belkacem, H, Bessin, Y, Pawlotsky, J.M, Guichou, J.F.
登録日2011-03-18
公開日2012-03-21
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献Fragment-based discovery of a new family of non-peptidic small-molecule cyclophilin inhibitors with potent antiviral activities.
Nat Commun, 7, 2016
3RCI
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BU of 3rci by Molmil
Human cyclophilin D complexed with 5-methyl-1,2-oxazol-3-amine
分子名称: 5-methyl-1,2-oxazol-3-amine, Peptidyl-prolyl cis-trans isomerase F, mitochondrial
著者Colliandre, L, Ahmed-Belkacem, H, Bessin, Y, Pawlotsky, J.M, Guichou, J.F.
登録日2011-03-31
公開日2012-03-21
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.44 Å)
主引用文献Fragment-based discovery of a new family of non-peptidic small-molecule cyclophilin inhibitors with potent antiviral activities.
Nat Commun, 7, 2016
3RDD
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BU of 3rdd by Molmil
Human Cyclophilin A Complexed with an Inhibitor
分子名称: Peptidyl-prolyl cis-trans isomerase A, ethyl N-[(4-aminobenzyl)carbamoyl]glycinate
著者Colliandre, L, Ahmed-Belkacem, H, Bessin, Y, Pawlotsky, J.M, Guichou, J.F.
登録日2011-04-01
公開日2012-03-21
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (2.14 Å)
主引用文献Fragment-based discovery of a new family of non-peptidic small-molecule cyclophilin inhibitors with potent antiviral activities.
Nat Commun, 7, 2016
3RCG
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Human cyclophilin D complexed with dimethylformamide
分子名称: CHLORIDE ION, DIMETHYLFORMAMIDE, Peptidyl-prolyl cis-trans isomerase F, ...
著者Colliandre, L, Ahmed-Belkacem, H, Bessin, Y, Pawlotsky, J.M, Guichou, J.F.
登録日2011-03-31
公開日2012-03-21
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (0.97 Å)
主引用文献Fragment-based discovery of a new family of non-peptidic small-molecule cyclophilin inhibitors with potent antiviral activities.
Nat Commun, 7, 2016
4R94
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Structure of the nickase domain of NS1 from MVM complexed with magnesium
分子名称: MAGNESIUM ION, Non-structural protein NS1
著者Liang, L, Zhao, H, Tang, L.
登録日2014-09-03
公開日2015-01-21
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.668 Å)
主引用文献Structures of minute virus of mice replication initiator protein N-terminal domain: Insights into DNA nicking and origin binding.
Virology, 476C, 2014

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