3WD1
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![BU of 3wd1 by Molmil](/molmil-images/mine/3wd1) | Serratia marcescens Chitinase B complexed with syn-triazole inhibitor | Descriptor: | Chitinase B, GLYCEROL, N,N-dibenzyl-N~5~-[N-(methylcarbamoyl)carbamimidoyl]-N~2~-{[5-({[(E)-(quinolin-4-ylmethylidene)amino]oxy}methyl)-1H-1,2,3-triazol-1-yl]acetyl}-L-ornithinamide, ... | Authors: | Hirose, T, Maita, N, Gouda, H, Koseki, J, Yamamoto, T, Sugawara, A, Nakano, H, Hirono, S, Shiomi, K, Watanabe, T, Taniguchi, H, Sharpless, K.B, Omura, S, Sunazuka, T. | Deposit date: | 2013-06-06 | Release date: | 2013-09-18 | Last modified: | 2023-11-08 | Method: | X-RAY DIFFRACTION (2.3 Å) | Cite: | Observation of the controlled assembly of preclick components in the in situ click chemistry generation of a chitinase inhibitor Proc.Natl.Acad.Sci.USA, 110, 2013
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3WD3
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![BU of 3wd3 by Molmil](/molmil-images/mine/3wd3) | Serratia marcescens Chitinase B complexed with azide inhibitor | Descriptor: | Chitinase B, GLYCEROL, SULFATE ION, ... | Authors: | Hirose, T, Maita, N, Gouda, H, Koseki, J, Yamamoto, T, Sugawara, A, Nakano, H, Hirono, S, Shiomi, K, Watanabe, T, Taniguchi, H, Sharpless, K.B, Omura, S, Sunazuka, T. | Deposit date: | 2013-06-06 | Release date: | 2013-09-18 | Last modified: | 2023-11-08 | Method: | X-RAY DIFFRACTION (2.2 Å) | Cite: | Observation of the controlled assembly of preclick components in the in situ click chemistry generation of a chitinase inhibitor Proc.Natl.Acad.Sci.USA, 110, 2013
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3WD0
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![BU of 3wd0 by Molmil](/molmil-images/mine/3wd0) | Serratia marcescens Chitinase B, tetragonal form | Descriptor: | Chitinase B, DITHIANE DIOL, GLYCEROL, ... | Authors: | Hirose, T, Maita, N, Gouda, H, Koseki, J, Yamamoto, T, Sugawara, A, Nakano, H, Hirono, S, Shiomi, K, Watanabe, T, Taniguchi, H, Sharpless, K.B, Omura, S, Sunazuka, T. | Deposit date: | 2013-06-06 | Release date: | 2013-09-18 | Last modified: | 2023-11-08 | Method: | X-RAY DIFFRACTION (1.7 Å) | Cite: | Observation of the controlled assembly of preclick components in the in situ click chemistry generation of a chitinase inhibitor Proc.Natl.Acad.Sci.USA, 110, 2013
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2ZZO
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![BU of 2zzo by Molmil](/molmil-images/mine/2zzo) | Crystal structure of the complex between GP41 fragment N36 and fusion inhibitor C34/S138A | Descriptor: | Transmembrane protein | Authors: | Watabe, T, Nakano, H, Nakatsu, T, Kato, H, Fujii, N. | Deposit date: | 2009-02-20 | Release date: | 2009-08-04 | Last modified: | 2023-11-01 | Method: | X-RAY DIFFRACTION (2.2 Å) | Cite: | X-ray crystallographic study of an HIV-1 fusion inhibitor with the gp41 S138A substitution J.Mol.Biol., 392, 2009
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3TK5
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![BU of 3tk5 by Molmil](/molmil-images/mine/3tk5) | Factor Xa in complex with D102-4380 | Descriptor: | 4-{3-[(4-chlorophenyl)amino]-3-oxopropyl}-3-({[5-(propan-2-yl)-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl]carbonyl}amino)benzoic acid, CALCIUM ION, Factor X heavy chain, ... | Authors: | Suzuki, M, Mochizuki, A, Nagata, T, Takano, H, Kanno, H, Kishida, M, Ohta, T. | Deposit date: | 2011-08-25 | Release date: | 2012-08-29 | Last modified: | 2017-11-08 | Method: | X-RAY DIFFRACTION (2.2 Å) | Cite: | Zwitter ionic potent durable orally active Factor Xa inhibitor. To be Published
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3TK6
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![BU of 3tk6 by Molmil](/molmil-images/mine/3tk6) | factor Xa in complex with D46-5241 | Descriptor: | CALCIUM ION, Factor X heavy chain, Factor X light chain, ... | Authors: | Suzuki, M, Mochizuki, A, Nagata, T, Takano, H, Kanno, H, Kishida, M, Ohta, T. | Deposit date: | 2011-08-25 | Release date: | 2012-08-29 | Last modified: | 2017-11-08 | Method: | X-RAY DIFFRACTION (1.8 Å) | Cite: | Zwitter ionic potent durable orally active Factor Xa inhibitor. To be Published
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1GE9
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![BU of 1ge9 by Molmil](/molmil-images/mine/1ge9) | SOLUTION STRUCTURE OF THE RIBOSOME RECYCLING FACTOR | Descriptor: | RIBOSOME RECYCLING FACTOR | Authors: | Yoshida, T, Uchiyama, S, Nakano, H, Kashimori, H, Kijima, H, Ohshima, T, Saihara, Y, Ishino, T, Shimahara, T, Yoshida, T, Yokose, K, Ohkubo, T, Kaji, A, Kobayashi, Y. | Deposit date: | 2000-10-19 | Release date: | 2001-05-16 | Last modified: | 2023-12-27 | Method: | SOLUTION NMR | Cite: | Solution structure of the ribosome recycling factor from Aquifex aeolicus. Biochemistry, 40, 2001
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2ZWS
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![BU of 2zws by Molmil](/molmil-images/mine/2zws) | Crystal Structure Analysis of neutral ceramidase from Pseudomonas aeruginosa | Descriptor: | FORMIC ACID, GLYCEROL, MAGNESIUM ION, ... | Authors: | Kakuta, Y, Okino, N, Inoue, T, Okano, H, Ito, M. | Deposit date: | 2008-12-17 | Release date: | 2009-03-03 | Last modified: | 2011-07-13 | Method: | X-RAY DIFFRACTION (1.4 Å) | Cite: | Mechanistic insights into the hydrolysis and synthesis of ceramide by neutral ceramidase. J.Biol.Chem., 284, 2009
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2DT4
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![BU of 2dt4 by Molmil](/molmil-images/mine/2dt4) | Crystal structure of Pyrococcus horikoshii a plant- and prokaryote-conserved (PPC) protein at 1.60 resolution | Descriptor: | GLYCEROL, Hypothetical protein PH0802 | Authors: | Lin, L, Nakano, H, Uchiyama, S, Fujimoto, S, Matsunaga, S, Nakamura, S. | Deposit date: | 2006-07-10 | Release date: | 2007-05-22 | Last modified: | 2024-03-13 | Method: | X-RAY DIFFRACTION (1.6 Å) | Cite: | Crystal structure of Pyrococcus horikoshii PPC protein at 1.60 A resolution Proteins, 67, 2007
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3WHP
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![BU of 3whp by Molmil](/molmil-images/mine/3whp) | Crystal structure of the C-terminal domain of Themus thermophilus LitR in complex with cobalamin | Descriptor: | COBALAMIN, Probable transcriptional regulator | Authors: | Agari, Y, Takano, H, Beppu, T, Ueda, K, Shinkai, A. | Deposit date: | 2013-08-30 | Release date: | 2014-09-03 | Last modified: | 2024-03-20 | Method: | X-RAY DIFFRACTION (2.52 Å) | Cite: | Crystal structure of the C-terminal domain of Themus thermophilus LitR in complex with cobalamin To be Published
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3AHA
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![BU of 3aha by Molmil](/molmil-images/mine/3aha) | Crystal structure of the complex between gp41 fragments N36 and C34 mutant N126K/E137Q | Descriptor: | (4S)-2-METHYL-2,4-PENTANEDIOL, CHLORIDE ION, Transmembrane protein gp41 | Authors: | Izumi, K, Nakamura, S, Nakano, H, Shimura, K, Sakagami, Y, Oishi, S, Uchiyama, S, Ohkubo, T, Kobayashi, Y, Fujii, N, Matsuoka, M, Kodama, E.N. | Deposit date: | 2010-04-22 | Release date: | 2010-05-19 | Last modified: | 2023-11-01 | Method: | X-RAY DIFFRACTION (1.7 Å) | Cite: | Characterization of HIV-1 resistance to a fusion inhibitor, N36, derived from the gp41 amino terminal heptad repeat. Antiviral Res., 2010
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