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PDB: 1 件

5HVU
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Rho-associated protein kinase 1 (ROCK 1) in complex with a pyridine thiazole piperidine inhibitor
分子名称: 2-{3-[3-(piperidin-4-yl)propoxy]phenyl}-N-[4-(pyridin-4-yl)-1,3-thiazol-2-yl]acetamide, Rho-associated protein kinase 1
著者Jacobs, M.J.
登録日2016-01-28
公開日2017-02-08
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献ROCK inhibitors 2. Improving potency, selectivity and solubility through the application of rationally designed solubilizing groups.
Bioorg. Med. Chem. Lett., 2018

219869

件を2024-05-15に公開中

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