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PDB: 58 件

6RHT
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BU of 6rht by Molmil
Structure of Pediococcus acidilactici putative lactate oxidase WT protein
分子名称: FLAVIN MONONUCLEOTIDE, GLYCEROL, Putative L-lactate oxidase
著者Ashok, Y, Maksimainen, M.M, Kilpelainen, P, Lehtio, L.
登録日2019-04-22
公開日2020-02-12
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献FMN-dependent oligomerization of putative lactate oxidase from Pediococcus acidilactici.
Plos One, 15, 2020
7R3Z
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BU of 7r3z by Molmil
Tankyrase 2 catalytic domain in complex with OUL40
分子名称: 6-methyl-[1,2,4]triazolo[3,4-b][1,3]benzothiazole, GLYCEROL, Poly [ADP-ribose] polymerase tankyrase-2, ...
著者Murthy, S, Venkannagari, H, Maksimainen, M.M, Lehtio, L.
登録日2022-02-08
公開日2023-01-25
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.25 Å)
主引用文献[1,2,4]Triazolo[3,4- b ]benzothiazole Scaffold as Versatile Nicotinamide Mimic Allowing Nanomolar Inhibition of Different PARP Enzymes.
J.Med.Chem., 66, 2023
7R4A
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PARP15 catalytic domain in complex with OUL188
分子名称: 6,8-dimethyl-[1,2,4]triazolo[3,4-b][1,3]benzothiazole, DIMETHYL SULFOXIDE, Protein mono-ADP-ribosyltransferase PARP15
著者Murthy, S, Maksimainen, M.M, Lehtio, L.
登録日2022-02-08
公開日2023-01-25
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献[1,2,4]Triazolo[3,4- b ]benzothiazole Scaffold as Versatile Nicotinamide Mimic Allowing Nanomolar Inhibition of Different PARP Enzymes.
J.Med.Chem., 66, 2023
7Z41
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BU of 7z41 by Molmil
PARP15 catalytic domain in complex with OUL209
分子名称: 5,8-dimethoxy-[1,2,4]triazolo[3,4-b][1,3]benzothiazole, DIMETHYL SULFOXIDE, Protein mono-ADP-ribosyltransferase PARP15
著者Murthy, S, Maksimainen, M.M, Lehtio, L.
登録日2022-03-03
公開日2023-01-25
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献[1,2,4]Triazolo[3,4- b ]benzothiazole Scaffold as Versatile Nicotinamide Mimic Allowing Nanomolar Inhibition of Different PARP Enzymes.
J.Med.Chem., 66, 2023
6RY4
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BU of 6ry4 by Molmil
PARP15 catalytic domain in complex with 4-(3-carbamoylphenoxy)benzamide.
分子名称: 3-(4-aminocarbonylphenoxy)benzamide, DIMETHYL SULFOXIDE, Protein mono-ADP-ribosyltransferase PARP15
著者Murthy, S.N, Maksimainen, M.M, Lehtio, L.
登録日2019-06-10
公開日2020-07-15
最終更新日2024-05-29
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Evaluation of 3- and 4-Phenoxybenzamides as Selective Inhibitors of the Mono-ADP-Ribosyltransferase PARP10.
Chemistryopen, 2021
6RHS
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BU of 6rhs by Molmil
Crystal structure of Pediococcus acidilactici (Putative)lactate oxidase Refolded WT protein
分子名称: FLAVIN MONONUCLEOTIDE, GLYCEROL, Putative L-lactate oxidase
著者Ashok, Y, Maksimainen, M.M, Kilpelainen, P, Lehtio, L.
登録日2019-04-22
公開日2020-02-12
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献FMN-dependent oligomerization of putative lactate oxidase from Pediococcus acidilactici.
Plos One, 15, 2020
7R59
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PARP2 catalytic domain in complex with OUL245
分子名称: GLYCEROL, Poly [ADP-ribose] polymerase 2, [1,2,4]triazolo[3,4-b][1,3]benzothiazol-6-ol
著者Galera-Prat, A, Maksimainen, M.M, Lehtio, L.
登録日2022-02-10
公開日2023-01-25
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献[1,2,4]Triazolo[3,4- b ]benzothiazole Scaffold as Versatile Nicotinamide Mimic Allowing Nanomolar Inhibition of Different PARP Enzymes.
J.Med.Chem., 66, 2023
6R9V
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BU of 6r9v by Molmil
Crystal structure of Pediococcus acidilactici lactate oxidase A94G mutant
分子名称: FLAVIN MONONUCLEOTIDE, GLYCEROL, Putative L-lactate oxidase, ...
著者Ashok, Y, Maksimainen, M.M, Lehtio, L.
登録日2019-04-04
公開日2020-02-12
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献FMN-dependent oligomerization of putative lactate oxidase from Pediococcus acidilactici.
Plos One, 15, 2020
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件を2024-07-24に公開中

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