Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help
PDB: 2 results

8YKI
DownloadVisualize
BU of 8yki by Molmil
FGFR-1 in complex with ligand tasurgratinib
Descriptor: CHLORIDE ION, Fibroblast growth factor receptor 1, Tasurgratinib
Authors:Ikemori-Kawada, M, Watanabe Miyano, S.
Deposit date:2024-03-05
Release date:2024-06-12
Method:X-RAY DIFFRACTION (2.79 Å)
Cite:Antitumor Activity of Tasurgratinib as an Orally Available FGFR1-3 Inhibitor in Cholangiocarcinoma Models With FGFR2-fusion.
Anticancer Res., 44, 2024
5ZV2
DownloadVisualize
BU of 5zv2 by Molmil
FGFR-1 in complex with ligand lenvatinib
Descriptor: 4-{3-chloro-4-[(cyclopropylcarbamoyl)amino]phenoxy}-7-methoxyquinoline-6-carboxamide, Fibroblast growth factor receptor 1
Authors:Matsuki, M, Hoshi, T, Yamamoto, Y, Ikemori-Kawada, M, Minoshima, Y, Funahashi, Y, Matsui, J.
Deposit date:2018-05-09
Release date:2018-07-11
Last modified:2023-11-22
Method:X-RAY DIFFRACTION (2.86 Å)
Cite:Lenvatinib inhibits angiogenesis and tumor fibroblast growth factor signaling pathways in human hepatocellular carcinoma models.
Cancer Med, 7, 2018

222624

數據於2024-07-17公開中

PDB statisticsPDBj update infoContact PDBjnumon