4D08
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 4d08 by Molmil](/molmil-images/mine/4d08) | PDE2a catalytic domain in complex with a brain penetrant inhibitor | 分子名称: | 1-(5-butoxypyridin-3-yl)-4-methyl-8-(morpholin-4-ylmethyl)[1,2,4]triazolo[4,3-a]quinoxaline, CGMP-DEPENDENT 3', 5'-CYCLIC PHOSPHODIESTERASE, ... | 著者 | Buijnsters, P, Andres, J.I, DeAngelis, M, Langlois, X, Rombouts, F, Sanderson, W, Tresadern, G, Trabanco, A, VanHoof, G, VanRoosbroeck, Y. | 登録日 | 2014-04-24 | 公開日 | 2014-08-06 | 最終更新日 | 2024-05-01 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Structure-Based Design of a Potent, Selective, and Brain Penetrating Pde2 Inhibitor with Demonstrated Target Engagement. Acs Med.Chem.Lett., 5, 2014
|
|
6L4O
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 6l4o by Molmil](/molmil-images/mine/6l4o) | Crystal structure of API5-FGF2 complex | 分子名称: | Apoptosis inhibitor 5, Fibroblast growth factor 2 | 著者 | Lee, B.I, Bong, S.M. | 登録日 | 2019-10-18 | 公開日 | 2020-04-29 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Regulation of mRNA export through API5 and nuclear FGF2 interaction. Nucleic Acids Res., 48, 2020
|
|
4C61
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 4c61 by Molmil](/molmil-images/mine/4c61) | Inhibitors of Jak2 Kinase domain | 分子名称: | ACETATE ION, N2-[(1S)-1-(5-fluoropyrimidin-2-yl)ethyl]-7-methyl-N4-(1-methylimidazol-4-yl)thieno[3,2-d]pyrimidine-2,4-diamine, TYROSINE-PROTEIN KINASE JAK2 | 著者 | Read, J.A, Green, I, Pollard, H, Howard, T. | 登録日 | 2013-09-17 | 公開日 | 2014-01-08 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.45 Å) | 主引用文献 | Discovery of 1-Methyl-1H-Imidazole Derivatives as Potent Jak2 Inhibitors. J.Med.Chem., 57, 2014
|
|
6S3G
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 6s3g by Molmil](/molmil-images/mine/6s3g) | Crystal Structure of lipase from Geobacillus stearothermophilus T6 variant A187C/F291C | 分子名称: | CALCIUM ION, Lipase, ZINC ION | 著者 | Gihaz, S, Bash, Y, Rush, I, Shahar, A, Pazy, Y, Fishman, A. | 登録日 | 2019-06-25 | 公開日 | 2019-10-09 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Bridges to Stability: Engineering Disulfide Bonds Towards Enhanced Lipase Biodiesel Synthesis Chemcatchem, 2019
|
|
6RJW
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 6rjw by Molmil](/molmil-images/mine/6rjw) | |
4XPE
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 4xpe by Molmil](/molmil-images/mine/4xpe) | |
4XPK
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 4xpk by Molmil](/molmil-images/mine/4xpk) | The crystal structure of Campylobacter jejuni N-acetyltransferase PseH | 分子名称: | N-Acetyltransferase, PseH | 著者 | Song, W.S, Nam, M.S, Namgung, B, Yoon, S.I. | 登録日 | 2015-01-17 | 公開日 | 2015-03-18 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.95 Å) | 主引用文献 | Structural analysis of PseH, the Campylobacter jejuni N-acetyltransferase involved in bacterial O-linked glycosylation. Biochem.Biophys.Res.Commun., 458, 2015
|
|
6KZ7
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 6kz7 by Molmil](/molmil-images/mine/6kz7) | The crystal structure of BAF155 SWIRM domain and N-terminal elongated hSNF5 RPT1 domain complex: Chromatin remodeling complex | 分子名称: | SWI/SNF complex subunit SMARCC1, SWI/SNF-related matrix-associated actin-dependent regulator of chromatin subfamily B member 1 | 著者 | Lee, W, Han, J, Kim, I, Park, J.H, Joo, K, Lee, J, Suh, J.Y. | 登録日 | 2019-09-23 | 公開日 | 2020-07-08 | 最終更新日 | 2024-03-27 | 実験手法 | X-RAY DIFFRACTION (2.28 Å) | 主引用文献 | A Coil-to-Helix Transition Serves as a Binding Motif for hSNF5 and BAF155 Interaction. Int J Mol Sci, 21, 2020
|
|
4XQ1
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 4xq1 by Molmil](/molmil-images/mine/4xq1) | Crystal structure of hemerythrin: L114A mutant | 分子名称: | Bacteriohemerythrin, FE (III) ION, NITRATE ION, ... | 著者 | Chuankhayan, P, Chen, K.H.C, Wu, H.H, Chen, C.J, Fukuda, M, Yu, S.S.F, Chan, S.I. | 登録日 | 2015-01-18 | 公開日 | 2015-04-29 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (1.4 Å) | 主引用文献 | The bacteriohemerythrin from Methylococcus capsulatus (Bath): Crystal structures reveal that Leu114 regulates a water tunnel. J.Inorg.Biochem., 150, 2015
|
|
5TOH
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5toh by Molmil](/molmil-images/mine/5toh) | Crystal Structure of the Marburg Virus VP35 Oligomerization Domain I2 | 分子名称: | Polymerase cofactor VP35 | 著者 | Bruhn, J.F, Kirchdoerfer, R.N, Tickle, I.J, Bricogne, G, Saphire, E.O. | 登録日 | 2016-10-17 | 公開日 | 2016-11-09 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (2.01 Å) | 主引用文献 | Crystal Structure of the Marburg Virus VP35 Oligomerization Domain. J. Virol., 91, 2017
|
|
5TR3
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5tr3 by Molmil](/molmil-images/mine/5tr3) | 2.5 Angstrom Resolution Crystal Structure of Dihydrolipoyl Dehydrogenase from Pseudomonas putida in Complex with FAD. | 分子名称: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Dihydrolipoyl dehydrogenase, FLAVIN-ADENINE DINUCLEOTIDE, ... | 著者 | Minasov, G, Wawrzak, Z, Shuvalova, L, Kiryukhina, O, Dubrovska, I, Grimshaw, S, Kwon, K, Anderson, W.F, Center for Structural Genomics of Infectious Diseases (CSGID) | 登録日 | 2016-10-25 | 公開日 | 2016-11-09 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | 2.5 Angstrom Resolution Crystal Structure of Dihydrolipoyl Dehydrogenase from Pseudomonas putida in Complex with FAD. To Be Published
|
|
4Y03
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 4y03 by Molmil](/molmil-images/mine/4y03) | Crystal Structure of the fifth bromodomain of human PB1 in complex with salicylic acid | 分子名称: | 2-HYDROXYBENZOIC ACID, CITRIC ACID, Protein polybromo-1 | 著者 | Filippakopoulos, P, Picaud, S, Felletar, I, Fedorov, O, von Delft, F, Edwards, A.M, Arrowsmith, C.H, Bountra, C, Knapp, S, Structural Genomics Consortium (SGC) | 登録日 | 2015-02-05 | 公開日 | 2015-05-20 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (1.94 Å) | 主引用文献 | Crystal Structure of the fifth bromodomain of human PB1 in complex with salicylic acid To Be Published
|
|
6RWP
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 6rwp by Molmil](/molmil-images/mine/6rwp) | |
6RWQ
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 6rwq by Molmil](/molmil-images/mine/6rwq) | Engineered beta-lactoglobulin: variant F105L in complex with myristic acid | 分子名称: | 1,2-ETHANEDIOL, Beta-lactoglobulin, MYRISTIC ACID | 著者 | Loch, J.I, Gotkowski, M, Lewinski, K. | 登録日 | 2019-06-05 | 公開日 | 2019-06-19 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (2.05 Å) | 主引用文献 | Structure-based design approach to rational site-directed mutagenesis of beta-lactoglobulin. J.Struct.Biol., 210, 2020
|
|
5IEM
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5iem by Molmil](/molmil-images/mine/5iem) | NMR structure of the 5'-terminal hairpin of the 7SK snRNA | 分子名称: | 7SK snRNA | 著者 | Bourbigot, S, Dock-Bregeon, A.C, Coutant, J, Kieffer, B, Lebars, I. | 登録日 | 2016-02-25 | 公開日 | 2016-11-02 | 最終更新日 | 2024-06-19 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution structure of the 5'-terminal hairpin of the 7SK small nuclear RNA. RNA, 22, 2016
|
|
4Y0R
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 4y0r by Molmil](/molmil-images/mine/4y0r) | Bovine beta-lactoglobulin complex with pramocaine crystallized from ammonium sulphate (BLG-PRM2) | 分子名称: | Beta-lactoglobulin, Pramocaine | 著者 | Loch, J.I, Bonarek, P, Polit, A, Jablonski, M, Czub, M, Ye, X, Lewinski, K. | 登録日 | 2015-02-06 | 公開日 | 2015-07-01 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | beta-Lactoglobulin interactions with local anaesthetic drugs - Crystallographic and calorimetric studies. Int.J.Biol.Macromol., 80, 2015
|
|
6RWR
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 6rwr by Molmil](/molmil-images/mine/6rwr) | |
6RY3
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 6ry3 by Molmil](/molmil-images/mine/6ry3) | Structure of the WUS homeodomain | 分子名称: | ACETYL GROUP, Protein WUSCHEL, SULFATE ION | 著者 | Sloan, J.J, Wild, K, Sinning, I. | 登録日 | 2019-06-10 | 公開日 | 2020-04-29 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.374 Å) | 主引用文献 | Structural basis for the complex DNA binding behavior of the plant stem cell regulator WUSCHEL. Nat Commun, 11, 2020
|
|
4C62
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 4c62 by Molmil](/molmil-images/mine/4c62) | Inhibitors of Jak2 Kinase domain | 分子名称: | ACETATE ION, N2-[(1S)-1-(5-fluoropyrimidin-2-yl)ethyl]-n4-(1-methylimidazol-4-yl)-6-morpholino-1,3,5-triazine-2,4-diamine, TYROSINE-PROTEIN KINASE JAK2 | 著者 | Read, J, Green, I, Pollard, H, Howard, T. | 登録日 | 2013-09-17 | 公開日 | 2014-01-08 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.75 Å) | 主引用文献 | Discovery of 1-Methyl-1H-Imidazole Derivatives as Potent Jak2 Inhibitors. J.Med.Chem., 57, 2014
|
|
6RK3
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 6rk3 by Molmil](/molmil-images/mine/6rk3) | Solution structure of the ribosome Elongation Factor P (EF-P) from Staphylococcus aureus | 分子名称: | Elongation factor P | 著者 | Usachev, K, Fatkhullin, B, Gabdulkhakov, A, Khusainov, I, Golubev, A, Validov, S, Yusupova, G, Yusupov, M. | 登録日 | 2019-04-30 | 公開日 | 2020-03-11 | 最終更新日 | 2024-05-15 | 実験手法 | SOLUTION NMR | 主引用文献 | NMR and crystallographic structural studies of the Elongation factor P from Staphylococcus aureus. Eur.Biophys.J., 49, 2020
|
|
4XNG
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 4xng by Molmil](/molmil-images/mine/4xng) | |
5IWR
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5iwr by Molmil](/molmil-images/mine/5iwr) | Structure of Transient Receptor Potential (TRP) channel TRPV6 in the presence of barium | 分子名称: | 6-(5-METHYL-2-OXO-IMIDAZOLIDIN-4-YL)-HEXANOIC ACID, BARIUM ION, Transient receptor potential cation channel subfamily V member 6 | 著者 | Saotome, K, Singh, A.K, Yelshanskaya, M.V, Sobolevsky, A.I. | 登録日 | 2016-03-22 | 公開日 | 2016-06-15 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (3.85 Å) | 主引用文献 | Crystal structure of the epithelial calcium channel TRPV6. Nature, 534, 2016
|
|
4XPW
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 4xpw by Molmil](/molmil-images/mine/4xpw) | Crystal structures of Leu114F mutant | 分子名称: | Bacteriohemerythrin, FE (II) ION, GLYCEROL | 著者 | Chuankhayan, P, Chen, K.H.C, Wu, H.H, Chen, C.J, Fukuda, M, Yu, S.S.F, Chan, S.I. | 登録日 | 2015-01-18 | 公開日 | 2015-04-29 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.17 Å) | 主引用文献 | The bacteriohemerythrin from Methylococcus capsulatus (Bath): Crystal structures reveal that Leu114 regulates a water tunnel. J.Inorg.Biochem., 150, 2015
|
|
4XNO
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 4xno by Molmil](/molmil-images/mine/4xno) | Crystal structure of 5'-CTTATPPPZZZATAAG | 分子名称: | DNA (5'-D(*CP*TP*(BRU)P*AP*TP*(1WA)P*(1WA)P*(1WA)P*(1W5)P*(1W5)P*(1W5)P*AP*TP*AP*AP*G)-3') | 著者 | Georgiadis, M.M, Singh, I. | 登録日 | 2015-01-15 | 公開日 | 2015-05-27 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.985 Å) | 主引用文献 | Structural basis for a six nucleotide genetic alphabet. J. Am. Chem. Soc., 137, 2015
|
|
4XXU
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 4xxu by Molmil](/molmil-images/mine/4xxu) | ModA - chromate bound | 分子名称: | Chromate, Molybdate-binding periplasmic protein | 著者 | He, C, Karpus, J, Ajiboye, I. | 登録日 | 2015-01-30 | 公開日 | 2016-09-14 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.43 Å) | 主引用文献 | Structure of chromate bound ModA from E.coli at 1.43 Angstroms resolution. To Be Published
|
|