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PDB: 1 results

8OY2
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Human cyclin-dependent kinase 2 in complex with inhibitor HB-29260
Descriptor: (1S,2S,11aS)-1-methoxy-1,4,7,10-tetramethyl-2,9-bis(oxidanyl)-2,11a-dihydrobenzo[b][1,4]benzodioxepine-3,6-dione, Cyclin-dependent kinase 2, GLYCEROL
Authors:Kordes, S, Harvey, C.J.B.
Deposit date:2023-05-03
Release date:2023-11-29
Last modified:2023-12-06
Method:X-RAY DIFFRACTION (2.618 Å)
Cite:Resistance gene-guided genome mining reveals the roseopurpurins as inhibitors of cyclin-dependent kinases.
Proc.Natl.Acad.Sci.USA, 120, 2023

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