3F7U
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![BU of 3f7u by Molmil](/molmil-images/mine/3f7u) | Crystal Structure of soluble domain of CA4 in complex with small molecule. | 分子名称: | Carbonic anhydrase 4, N-(3-methoxypropyl)-2-(phenylsulfanyl)-5-sulfamoylpyridine-3-carboxamide, ZINC ION | 著者 | Pauly, T.A, Ferre, R.A.A, Greasley, S.E, Paz, R. | 登録日 | 2008-11-10 | 公開日 | 2009-09-22 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Thioether benzenesulfonamide inhibitors of carbonic anhydrases II and IV: structure-based drug design, synthesis, and biological evaluation. Bioorg.Med.Chem., 18, 2010
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1D5T
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![BU of 1d5t by Molmil](/molmil-images/mine/1d5t) | GUANINE NUCLEOTIDE DISSOCIATION INHIBITOR, ALPHA-ISOFORM | 分子名称: | GUANINE NUCLEOTIDE DISSOCIATION INHIBITOR, SULFATE ION | 著者 | Peng, L, Zeng, K, Heine, A, Moyer, B, Greasley, S.E, Kuhn, P, Balch, W.E, Wilson, I.A. | 登録日 | 1999-10-11 | 公開日 | 2000-10-25 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (1.04 Å) | 主引用文献 | A new functional domain of guanine nucleotide dissociation inhibitor (alpha-GDI) involved in Rab recycling. Traffic, 1, 2000
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3PS6
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3PRE
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![BU of 3pre by Molmil](/molmil-images/mine/3pre) | Quinazolines with intra-molecular hydrogen bonding scaffold (iMHBS) as PI3K/mTOR dual inhibitors. | 分子名称: | 2-amino-8-(trans-4-methoxycyclohexyl)-4-methyl-6-(1H-pyrazol-3-yl)pyrido[2,3-d]pyrimidin-7(8H)-one, Phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit gamma isoform | 著者 | Knighton, D.R, Greasley, S.E, Rodgers, C.M.-L. | 登録日 | 2010-11-29 | 公開日 | 2011-02-09 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (2.91 Å) | 主引用文献 | Quinazolines with intra-molecular hydrogen bonding scaffold (iMHBS) as PI3K/mTOR dual inhibitors. Bioorg.Med.Chem.Lett., 21, 2011
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3PRZ
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![BU of 3prz by Molmil](/molmil-images/mine/3prz) | |