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PDB: 3 件

8ESX
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BU of 8esx by Molmil
HIV protease in complex with benzoxaborolone analog of darunavir
分子名称: ACETATE ION, CHLORIDE ION, GLYCEROL, ...
著者Windsor, I.W, Graham, B.J, Raines, R.T.
登録日2022-10-15
公開日2023-02-08
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.35 Å)
主引用文献Inhibition of HIV-1 Protease by a Boronic Acid with High Oxidative Stability.
Acs Med.Chem.Lett., 14, 2023
8ESY
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BU of 8esy by Molmil
D30N mutant HIV protease in complex with benzoxaborolone analog of darunavir
分子名称: CHLORIDE ION, GLYCEROL, Protease, ...
著者Windsor, I.W, Graham, B.J, Raines, R.T.
登録日2022-10-15
公開日2023-02-08
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.35 Å)
主引用文献Inhibition of HIV-1 Protease by a Boronic Acid with High Oxidative Stability.
Acs Med.Chem.Lett., 14, 2023
6U0Q
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BU of 6u0q by Molmil
Transthyretin in complex with (E)-5,5'-(ethene-1,2-diyl)bis(1,1-dihydroxy-3-oxo-1,3-dihydrobenzo[c][1,2]oxaborol-1-uide)
分子名称: 3-[(~{E})-2-[7,7-bis(oxidanyl)-9-oxidanylidene-8-oxa-7-boranuidabicyclo[4.3.0]nona-1,3,5-trien-3-yl]ethenyl]-7,7-bis(oxidanyl)-8-oxa-7-boranuidabicyclo[4.3.0]nona-1(6),2,4-trien-9-one, Transthyretin
著者Windsor, I.W, Graham, B.J, Raines, R.T.
登録日2019-08-14
公開日2021-01-27
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Boronic acid with high oxidative stability and utility in biological contexts.
Proc.Natl.Acad.Sci.USA, 118, 2021

224004

件を2024-08-21に公開中

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