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PDB: 8 件

1LOX
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BU of 1lox by Molmil
RABBIT RETICULOCYTE 15-LIPOXYGENASE
分子名称: (2E)-3-(2-OCT-1-YN-1-YLPHENYL)ACRYLIC ACID, 15-LIPOXYGENASE, FE (II) ION
著者Gillmor, S.A, Villasenor, A, Fletterick, R.J, Sigal, E, Browner, M.F.
登録日1997-10-06
公開日1998-11-04
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献The structure of mammalian 15-lipoxygenase reveals similarity to the lipases and the determinants of substrate specificity.
Nat.Struct.Biol., 4, 1997
2AIM
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BU of 2aim by Molmil
CRUZAIN INHIBITED WITH BENZOYL-ARGININE-ALANINE-FLUOROMETHYLKETONE
分子名称: BENZOYL-ARGININE-ALANINE-FLUORO-METHYL KETONE, CRUZAIN
著者Gillmor, S.A, Fletterick, R.J.
登録日1997-04-21
公開日1997-10-22
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Structural determinants of specificity in the cysteine protease cruzain.
Protein Sci., 6, 1997
1EWP
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BU of 1ewp by Molmil
CRUZAIN BOUND TO MOR-LEU-HPQ
分子名称: CRUZAIN, N-[(3S)-1-fluoro-2-oxo-5-phenylpentan-3-yl]-N~2~-(morpholin-4-ylcarbonyl)-L-leucinamide
著者Gillmor, S.A.
登録日2000-04-26
公開日2000-05-17
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Chapter 3: X-ray Structures of Complexes of Cruzain with Designed Covalent Inhibitors
Enzyme-ligand Interactions, Inhibition and Specificity, 1998
1EZU
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BU of 1ezu by Molmil
ECOTIN Y69F, D70P BOUND TO D102N TRYPSIN
分子名称: CALCIUM ION, ECOTIN, TRYPSIN II, ...
著者Gillmor, S.A, Takeuchi, T, Yang, S.Q, Craik, C.S, Fletterick, R.J.
登録日2000-05-11
公開日2000-06-23
最終更新日2021-11-03
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Compromise and accommodation in ecotin, a dimeric macromolecular inhibitor of serine proteases.
J.Mol.Biol., 299, 2000
1EZS
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BU of 1ezs by Molmil
CRYSTAL STRUCTURE OF ECOTIN MUTANT M84R, W67A, G68A, Y69A, D70A BOUND TO RAT ANIONIC TRYPSIN II
分子名称: CALCIUM ION, ECOTIN, TRYPSIN II, ...
著者Gillmor, S.A, Takeuchi, T, Yang, S.Q, Craik, C.S, Fletterick, R.J.
登録日2000-05-11
公開日2000-06-23
最終更新日2021-11-03
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Compromise and accommodation in ecotin, a dimeric macromolecular inhibitor of serine proteases.
J.Mol.Biol., 299, 2000
1EWL
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BU of 1ewl by Molmil
CRYSTAL STRUCTURE OF CRUZAIN BOUND TO WRR-99
分子名称: CRUZAIN, N-[3-CARBOXY-2-HYDROXY-PROPIONYL]-D-HOMOPHENYLALANYL-AMINO-2-METHYLBUTANE
著者Brinen, L.S, Gillmor, S.A, Fletterick, R.J.
登録日2000-04-26
公開日2003-06-10
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Crystal Structure of Cruzain bound to WRR-99
To be Published
1EWM
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BU of 1ewm by Molmil
THE CYSTEINE PROTEASE CRUZAIN BOUND TO WRR-112
分子名称: CRUZAIN, N-[3-CARBOXY-2-HYDROXY-PROPIONYL]-L-HOMOPHENYLALANYL-AMINO-2-METHYLBUTANE
著者Brinen, L.S, Gillmor, S.A, Fletterick, R.J.
登録日2000-04-26
公開日2003-06-10
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Crystal Structure of Cruzain bound to WRR-112
To be Published
1EWO
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BU of 1ewo by Molmil
THE CYSTEINE PROTEASE CRUZAIN BOUND TO WRR-204
分子名称: CRUZAIN, N-[N'-BENZYLOXYCARBONYL-PHENYLALANINYL]-3-AMINO-5-PHENYL-PENTANE-1-SULFONIC ACID PHENYL ESTER
著者Brinen, L.S, Gillmor, S.A, Fletterick, R.J.
登録日2000-04-26
公開日2003-06-10
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Crystal Structure of Cruzain bound to WRR-204
To be Published

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件を2024-09-11に公開中

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