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PDB: 6 件

4GW4
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Crystal structure of 3BNC60 Fab with P61A mutation
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 3BNC60 Fab Heavy-chain, 3BNC60 Fab Light-chain
著者Diskin, R, Fu, B.Z, Bjorkman, P.J.
登録日2012-08-31
公開日2013-04-17
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2.65 Å)
主引用文献Somatic Mutations of the Immunoglobulin Framework Are Generally Required for Broad and Potent HIV-1 Neutralization.
Cell(Cambridge,Mass.), 153, 2013
4JNM
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Discovery of Potent and Efficacious Urea-containing Nicotinamide Phosphoribosyltransferase (NAMPT) Inhibitors with Reduced CYP2C9 Inhibition Properties
分子名称: 1,2-ETHANEDIOL, 1-[(6-aminopyridin-3-yl)methyl]-3-[4-(phenylsulfonyl)phenyl]urea, Nicotinamide phosphoribosyltransferase, ...
著者Gunzner-Toste, J, Zhao, G, Bauer, P, Baumeister, T, Buckmelter, A.J, Caligiuri, M, Clodfelter, K.H, Fu, B, Han, B, Ho, Y, Kley, N, Liederer, B, Lin, J, Mukadam, S, O'Brien, T, Reynolds, D.J, Sharma, G, Skelton, N, Smith, C.C, Oh, A, Wang, W, Wang, Z, Xiao, Y, Yuen, P, Zak, M, Zhang, L, Zheng, X, Bair, K.W, Dragovich, P.S.
登録日2013-03-15
公開日2013-05-29
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Discovery of potent and efficacious urea-containing nicotinamide phosphoribosyltransferase (NAMPT) inhibitors with reduced CYP2C9 inhibition properties.
Bioorg.Med.Chem.Lett., 23, 2013
6MWY
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The Prp8 intein of Cryptococcus gattii
分子名称: Pre-mRNA-processing-splicing factor 8
著者Li, Z, Fu, B, Green, C.M, Lang, Y, Zhang, J, Oven, T.S, Li, X, Callahan, B.P, Chaturvedi, S, Belfort, M, Liao, G, Li, H.
登録日2018-10-30
公開日2019-11-06
最終更新日2020-05-20
実験手法X-RAY DIFFRACTION (2.594 Å)
主引用文献Cisplatin protects mice from challenge ofCryptococcus neoformansby targeting the Prp8 intein.
Emerg Microbes Infect, 8, 2019
6BJB
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Crystal structure of Acat2-C91S thiolase from Ascaris suum in complex with propionyl-CoA and nitrate
分子名称: Acetyl-CoA acetyltransferase A, NITRATE ION, propionyl Coenzyme A
著者Blaisse, M.R, Fu, B, Chang, M.C.Y.
登録日2017-11-05
公開日2018-02-07
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (1.50000632 Å)
主引用文献Structural and Biochemical Studies of Substrate Selectivity in Ascaris suum Thiolases.
Biochemistry, 57, 2018
6BJ9
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Crystal structure of Acat2 thiolase from Ascaris suum
分子名称: Acetyl-CoA acetyltransferase A, POTASSIUM ION
著者Blaisse, M.R, Fu, B, Chang, M.C.Y.
登録日2017-11-05
公開日2018-02-07
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (1.53014076 Å)
主引用文献Structural and Biochemical Studies of Substrate Selectivity in Ascaris suum Thiolases.
Biochemistry, 57, 2018
6BJA
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Crystal structure of Acat5 thiolase from Ascaris suum in complex with coenzyme A
分子名称: ACETATE ION, Acetyl-CoA acetyltransferase A, COENZYME A
著者Blaisse, M.R, Fu, B, Chang, M.C.Y.
登録日2017-11-05
公開日2018-02-07
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.60001445 Å)
主引用文献Structural and Biochemical Studies of Substrate Selectivity in Ascaris suum Thiolases.
Biochemistry, 57, 2018

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件を2024-06-26に公開中

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