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PDB: 1 件

8GD7
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Loop Deleted DNA Polymerase Theta Polymerase Domain in Complex with Double Strand DNA Overhang and Inhibitor
分子名称: 2'-3'-DIDEOXYGUANOSINE-5'-TRIPHOSPHATE, 2-(3-methyl-2-oxoimidazolidin-1-yl)-4,6-bis(trifluoromethyl)phenyl (4-fluorophenyl)methylcarbamate, DNA Primer, ...
著者Fried, W.A, Chen, X.S, Li, S.X.
登録日2023-03-03
公開日2024-06-19
実験手法X-RAY DIFFRACTION (3.24 Å)
主引用文献Discovery of a small-molecule inhibitor that traps Pol theta on DNA and synergizes with PARP inhibitors.
Nat Commun, 15, 2024

222624

件を2024-07-17に公開中

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