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PDB: 94 results

1ID5
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BU of 1id5 by Molmil
CRYSTAL STRUCTURE OF BOVINE THROMBIN COMPLEX WITH PROTEASE INHIBITOR ECOTIN
Descriptor: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, CALCIUM ION, ECOTIN, ...
Authors:Wang, S.X, Fletterick, R.J.
Deposit date:2001-04-03
Release date:2001-09-05
Last modified:2021-10-27
Method:X-RAY DIFFRACTION (2.5 Å)
Cite:Crystal structure of thrombin-ecotin reveals conformational changes and extended interactions.
Biochemistry, 40, 2001
1BSX
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BU of 1bsx by Molmil
STRUCTURE AND SPECIFICITY OF NUCLEAR RECEPTOR-COACTIVATOR INTERACTIONS
Descriptor: 3,5,3'TRIIODOTHYRONINE, PROTEIN (GRIP1), PROTEIN (THYROID HORMONE RECEPTOR BETA)
Authors:Wagner, R.L, Darimont, B.D, Apriletti, J.W, Stallcup, M.R, Kushner, P.J, Baxter, J.D, Fletterick, R.J, Yamamoto, K.R.
Deposit date:1998-08-31
Release date:1999-08-26
Last modified:2024-04-03
Method:X-RAY DIFFRACTION (3.7 Å)
Cite:Structure and specificity of nuclear receptor-coactivator interactions.
Genes Dev., 12, 1998
1AZZ
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BU of 1azz by Molmil
FIDDLER CRAB COLLAGENASE COMPLEXED TO ECOTIN
Descriptor: COLLAGENASE, ECOTIN
Authors:Perona, J.J, Fletterick, R.J.
Deposit date:1997-11-24
Release date:1998-02-25
Last modified:2024-06-05
Method:X-RAY DIFFRACTION (2.3 Å)
Cite:Crystal structure of an ecotin-collagenase complex suggests a model for recognition and cleavage of the collagen triple helix.
Biochemistry, 36, 1997
1BG2
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BU of 1bg2 by Molmil
HUMAN UBIQUITOUS KINESIN MOTOR DOMAIN
Descriptor: ACETATE ION, ADENOSINE-5'-DIPHOSPHATE, KINESIN, ...
Authors:Kull, F.J, Sablin, E.P, Lau, R, Fletterick, R.J, Vale, R.D.
Deposit date:1998-06-04
Release date:1998-10-14
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (1.8 Å)
Cite:Crystal structure of the kinesin motor domain reveals a structural similarity to myosin.
Nature, 380, 1996
1CU4
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CRYSTAL STRUCTURE OF THE ANTI-PRION FAB 3F4 IN COMPLEX WITH ITS PEPTIDE EPITOPE
Descriptor: FAB HEAVY CHAIN, FAB LIGHT CHAIN, RECOGNITION PEPTIDE
Authors:Kanyo, Z.F, Pan, K.M, Williamson, R.A, Burton, D.R, Prusiner, S.B, Fletterick, R.J, Cohen, F.E.
Deposit date:1999-08-20
Release date:2000-04-17
Last modified:2018-04-04
Method:X-RAY DIFFRACTION (2.9 Å)
Cite:Antibody binding defines a structure for an epitope that participates in the PrPC-->PrPSc conformational change.
J.Mol.Biol., 293, 1999
1CR9
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CRYSTAL STRUCTURE OF THE ANTI-PRION FAB 3F4
Descriptor: FAB ANTIBODY HEAVY CHAIN, FAB ANTIBODY LIGHT CHAIN
Authors:Kanyo, Z.F, Pan, K.M, Williamson, R.A, Burton, D.R, Prusiner, S.B, Fletterick, R.J, Cohen, F.E.
Deposit date:1999-08-14
Release date:2000-04-17
Last modified:2018-04-04
Method:X-RAY DIFFRACTION (2 Å)
Cite:Antibody binding defines a structure for an epitope that participates in the PrPC-->PrPSc conformational change.
J.Mol.Biol., 293, 1999
1EZS
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BU of 1ezs by Molmil
CRYSTAL STRUCTURE OF ECOTIN MUTANT M84R, W67A, G68A, Y69A, D70A BOUND TO RAT ANIONIC TRYPSIN II
Descriptor: CALCIUM ION, ECOTIN, TRYPSIN II, ...
Authors:Gillmor, S.A, Takeuchi, T, Yang, S.Q, Craik, C.S, Fletterick, R.J.
Deposit date:2000-05-11
Release date:2000-06-23
Last modified:2021-11-03
Method:X-RAY DIFFRACTION (2.3 Å)
Cite:Compromise and accommodation in ecotin, a dimeric macromolecular inhibitor of serine proteases.
J.Mol.Biol., 299, 2000
1PK5
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Crystal structure of the orphan nuclear receptor LRH-1
Descriptor: Orphan nuclear receptor NR5A2
Authors:Sablin, E.P, Krylova, I.N, Fletterick, R.J, Ingraham, H.A.
Deposit date:2003-06-04
Release date:2003-07-01
Last modified:2023-08-16
Method:X-RAY DIFFRACTION (2.4 Å)
Cite:Structural basis for ligand-independent activation of the orphan nuclear receptor LRH-1
Mol.Cell, 11, 2003
1I6I
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CRYSTAL STRUCTURE OF THE KIF1A MOTOR DOMAIN COMPLEXED WITH MG-AMPPCP
Descriptor: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, KINESIN-LIKE PROTEIN KIF1A, MAGNESIUM ION, ...
Authors:Kikkawa, M, Sablin, E.P, Okada, Y, Yajima, H, Fletterick, R.J, Hirokawa, N.
Deposit date:2001-03-02
Release date:2001-05-30
Last modified:2024-04-03
Method:X-RAY DIFFRACTION (2 Å)
Cite:Switch-based mechanism of kinesin motors
Nature, 411, 2001
1I5S
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CRYSTAL STRUCTURE OF THE KIF1A MOTOR DOMAIN COMPLEXED WITH MG-ADP
Descriptor: ADENOSINE-5'-DIPHOSPHATE, KINESIN-LIKE PROTEIN KIF1A, MAGNESIUM ION
Authors:Kikkawa, M, Sablin, E.P, Okada, Y, Yajima, H, Fletterick, R.J, Hirokawa, N.
Deposit date:2001-02-28
Release date:2001-05-30
Last modified:2024-04-03
Method:X-RAY DIFFRACTION (2.2 Å)
Cite:Switch-based mechanism of kinesin motors
Nature, 411, 2001
1IA0
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BU of 1ia0 by Molmil
KIF1A HEAD-MICROTUBULE COMPLEX STRUCTURE IN ATP-FORM
Descriptor: GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, KINESIN-LIKE PROTEIN KIF1A, ...
Authors:Kikkawa, M, Sablin, E.P, Okada, Y, Yajima, H, Fletterick, R.J, Hirokawa, N.
Deposit date:2001-03-22
Release date:2002-03-22
Last modified:2021-10-27
Method:ELECTRON MICROSCOPY (15 Å)
Cite:Switch-based Mechanism of Kinesin Motors
Nature, 411, 2001
1EZU
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BU of 1ezu by Molmil
ECOTIN Y69F, D70P BOUND TO D102N TRYPSIN
Descriptor: CALCIUM ION, ECOTIN, TRYPSIN II, ...
Authors:Gillmor, S.A, Takeuchi, T, Yang, S.Q, Craik, C.S, Fletterick, R.J.
Deposit date:2000-05-11
Release date:2000-06-23
Last modified:2021-11-03
Method:X-RAY DIFFRACTION (2.4 Å)
Cite:Compromise and accommodation in ecotin, a dimeric macromolecular inhibitor of serine proteases.
J.Mol.Biol., 299, 2000
1IFG
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BU of 1ifg by Molmil
CRYSTAL STRUCTURE OF A MONOMERIC FORM OF GENERAL PROTEASE INHIBITOR, ECOTIN IN ABSENCE OF A PROTEASE
Descriptor: ECOTIN
Authors:Eggers, C.T, Wang, S.X, Fletterick, R.J, Craik, C.S.
Deposit date:2001-04-12
Release date:2001-05-18
Last modified:2023-08-16
Method:X-RAY DIFFRACTION (2 Å)
Cite:The role of ecotin dimerization in protease inhibition.
J.Mol.Biol., 308, 2001
1BRA
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BU of 1bra by Molmil
RELOCATING A NEGATIVE CHARGE IN THE BINDING POCKET OF TRYPSIN
Descriptor: BENZAMIDINE, CALCIUM ION, TRYPSIN
Authors:Perona, J.J, Mcgrath, M.E, Fletterick, R.J.
Deposit date:1992-12-17
Release date:1994-04-30
Last modified:2017-11-29
Method:X-RAY DIFFRACTION (2.2 Å)
Cite:Relocating a negative charge in the binding pocket of trypsin.
J.Mol.Biol., 230, 1993
1BRB
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BU of 1brb by Molmil
CRYSTAL STRUCTURES OF RAT ANIONIC TRYPSIN COMPLEXED WITH THE PROTEIN INHIBITORS APPI AND BPTI
Descriptor: PANCREATIC TRYPSIN INHIBITOR, TRYPSIN
Authors:Perona, J.J, Fletterick, R.J.
Deposit date:1992-12-17
Release date:1994-07-31
Last modified:2017-11-29
Method:X-RAY DIFFRACTION (2.1 Å)
Cite:Crystal structures of rat anionic trypsin complexed with the protein inhibitors APPI and BPTI.
J.Mol.Biol., 230, 1993
1Q4X
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BU of 1q4x by Molmil
Crystal Structure of Human Thyroid Hormone Receptor beta LBD in complex with specific agonist GC-24
Descriptor: Thyroid hormone receptor beta-1, [4-(3-BENZYL-4-HYDROXYBENZYL)-3,5-DIMETHYLPHENOXY]ACETIC ACID
Authors:Borngraeber, S, Budny, M.J, Chiellini, G, Cunha-Lima, S.T, Togashi, M, Webb, P, Baxter, J.D, Scanlan, T.S, Fletterick, R.J.
Deposit date:2003-08-04
Release date:2004-02-03
Last modified:2024-04-03
Method:X-RAY DIFFRACTION (2.8 Å)
Cite:Ligand selectivity by seeking hydrophobicity in thyroid hormone receptor.
Proc.Natl.Acad.Sci.USA, 100, 2003
1SDM
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BU of 1sdm by Molmil
Crystal structure of kinesin-like calmodulin binding protein
Descriptor: ADENOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, kinesin heavy chain-like protein
Authors:Vinogradova, M.V, Reddy, V.S, Reddy, A.S, Sablin, E.P, Fletterick, R.J.
Deposit date:2004-02-13
Release date:2004-06-22
Last modified:2023-08-23
Method:X-RAY DIFFRACTION (2.3 Å)
Cite:Crystal structure of kinesin regulated by Ca(2+)-calmodulin.
J.Biol.Chem., 279, 2004
1EAP
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BU of 1eap by Molmil
CRYSTAL STRUCTURE OF A CATALYTIC ANTIBODY WITH A SERINE PROTEASE ACTIVE SITE
Descriptor: IGG2B-KAPPA 17E8 FAB (HEAVY CHAIN), IGG2B-KAPPA 17E8 FAB (LIGHT CHAIN), PHENYL[1-(N-SUCCINYLAMINO)PENTYL]PHOSPHONATE
Authors:Zhou, G.W, Guo, J, Huang, W, Scanlan, T.S, Fletterick, R.J.
Deposit date:1994-08-10
Release date:1994-12-20
Last modified:2024-06-05
Method:X-RAY DIFFRACTION (2.4 Å)
Cite:Crystal structure of a catalytic antibody with a serine protease active site.
Science, 265, 1994
1B89
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CLATHRIN HEAVY CHAIN PROXIMAL LEG SEGMENT (BOVINE)
Descriptor: PROTEIN (CLATHRIN HEAVY CHAIN)
Authors:Ybe, J.A, Brodsky, F.M, Hofmann, K, Lin, K, Liu, S.-H, Chen, L, Earnest, T.N, Fletterick, R.J, Hwang, P.K.
Deposit date:1999-05-27
Release date:1999-06-04
Last modified:2023-12-27
Method:X-RAY DIFFRACTION (2.6 Å)
Cite:Clathrin self-assembly is mediated by a tandemly repeated superhelix.
Nature, 399, 1999
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