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PDB: 1 results

8RDK
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Crystal structure of human Haspin (GSG2) kinase bound to MD420
Descriptor: (4S)-2-METHYL-2,4-PENTANEDIOL, 3-pyridin-4-yl-1~{H}-pyrrolo[3,2-g]isoquinoline, Serine/threonine-protein kinase haspin, ...
Authors:Kraemer, A, Defois, M, Giraud, F, Moreau, P, Anizon, F, Knapp, S, Structural Genomics Consortium (SGC)
Deposit date:2023-12-08
Release date:2024-03-06
Last modified:2024-08-07
Method:X-RAY DIFFRACTION (2 Å)
Cite:Synthesis and evaluation of chemical linchpins for highly selective CK2 alpha targeting.
Eur.J.Med.Chem., 276, 2024

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PDB entries from 2024-09-11

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