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3SVV
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BU of 3svv by Molmil
Crystal Structure of T338C c-Src covalently bound to vinylsulfonamide-pyrazolopyrimidine 9
Descriptor: N-(3-{[4-amino-1-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-3-yl]methyl}phenyl)ethanesulfonamide, Proto-oncogene tyrosine-protein kinase Src
Authors:Garske, A.L, Peters, U, Cortesi, A, Perez, J, Shokat, K.M.
Deposit date:2011-07-12
Release date:2011-08-17
Last modified:2024-03-13
Method:X-RAY DIFFRACTION (2.204 Å)
Cite:Chemical genetic strategy for targeting protein kinases based on covalent complementarity.
Proc.Natl.Acad.Sci.USA, 108, 2011

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