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PDB: 8 件

3MYE
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BU of 3mye by Molmil
Crystal Structure of HP67 L61GL
分子名称: Villin-1
著者Brown, J.W, Farelli, J.D, McKnight, C.J.
登録日2010-05-10
公開日2011-05-25
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.799 Å)
主引用文献Conserving the Hydrophobic Core at the Expense of Backbone Conformation in Villin Headpiece
To be Published
3MYA
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BU of 3mya by Molmil
Crystal Structure of HP67 H41F - P61
分子名称: Villin-1
著者Brown, J.W, Farelli, J.D, McKnight, C.J.
登録日2010-05-10
公開日2011-06-29
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献On unsatisfied hydrogen bonds in the N-terminal subdomain of villin headpiece.
J.Mol.Biol., 413, 2011
3NKJ
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BU of 3nkj by Molmil
Crystal Structure of HP67 L61G
分子名称: Villin-1
著者Brown, J.W, Farelli, J.D, McKnight, C.J.
登録日2010-06-20
公開日2011-06-01
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Conserving the Hydrophobic Core at the Expense of Backbone Conformation in Villin Headpiece
To be Published
3MYC
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BU of 3myc by Molmil
Crystal Structure of HP67 H41F - P212121
分子名称: Villin-1
著者Brown, J.W, Farelli, J.D, McKnight, C.J.
登録日2010-05-10
公開日2011-05-25
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献On unsatisfied hydrogen bonds in the N-terminal subdomain of villin headpiece.
J.Mol.Biol., 413, 2011
2K6M
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BU of 2k6m by Molmil
Solution Structure of Human Supervillin Headpiece
分子名称: Supervillin
著者Brown, J.W, Didem, V, McKnight, C.
登録日2008-07-11
公開日2009-07-14
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献How to arm a supervillin: designing F-actin binding activity into supervillin headpiece.
J.Mol.Biol., 393, 2009
2K6N
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BU of 2k6n by Molmil
Solution Structure of Human Supervillin Headpiece, Minimized Average
分子名称: Supervillin
著者Brown, J.W, Didem, V, McKnight, C.
登録日2008-07-11
公開日2009-07-14
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献How to arm a supervillin: designing F-actin binding activity into supervillin headpiece.
J.Mol.Biol., 393, 2009
9EZG
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BU of 9ezg by Molmil
Crystal structure of human Casein Kinase II subunit alpha (CK2a1) in complex with 5-((4-((2-aminoethyl)(ethyl)amino)-3-(4H-1,2,4-triazol-4-yl)phenyl)amino)-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidine-3-carbonitrile
分子名称: 1,2-ETHANEDIOL, 5-[[4-[2-azanylethyl(ethyl)amino]-3-(1,2,4-triazol-4-yl)phenyl]amino]-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidine-3-carbonitrile, Casein kinase II subunit alpha, ...
著者Kraemer, A, Ong, H.W, Yang, X, Brown, J.W, Chang, E, Willson, T, Knapp, S, Structural Genomics Consortium (SGC)
登録日2024-04-12
公開日2024-07-31
実験手法X-RAY DIFFRACTION (2.18 Å)
主引用文献More than an Amide Bioisostere: Discovery of 1,2,4-Triazole-containing Pyrazolo[1,5- a ]pyrimidine Host CSNK2 Inhibitors for Combatting beta-Coronavirus Replication.
J.Med.Chem., 2024
8P06
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BU of 8p06 by Molmil
Crystal structure of human Casein Kinase II subunit alpha (CK2a1) in complex with 5-((2-(4H-1,2,4-triazol-4-yl)pyridin-4-yl)amino)-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidine-3-carbonitrile
分子名称: 7-(cyclopropylamino)-5-[[2-(1,2,4-triazol-4-yl)pyridin-4-yl]amino]pyrazolo[1,5-a]pyrimidine-3-carbonitrile, Casein kinase II subunit alpha, SULFATE ION
著者Kraemer, A, Ong, H.W, Yang, X, Brown, J.W, Chang, E, Willson, T, Knapp, S, Structural Genomics Consortium (SGC)
登録日2023-05-09
公開日2023-06-21
最終更新日2024-07-31
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献More than an Amide Bioisostere: Discovery of 1,2,4-Triazole-containing Pyrazolo[1,5- a ]pyrimidine Host CSNK2 Inhibitors for Combatting beta-Coronavirus Replication.
J.Med.Chem., 2024

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件を2024-07-31に公開中

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