5N49
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![BU of 5n49 by Molmil](/molmil-images/mine/5n49) | BRPF2 in complex with Compound 7 | 分子名称: | 2-(1,3,6-trimethyl-2-oxidanylidene-benzimidazol-5-yl)benzo[de]isoquinoline-1,3-dione, Bromodomain-containing protein 1 | 著者 | Bouche, L, Christ, C.D, Siegel, S, Fernandez-Montalvan, A.E, Holton, S.J, Fedorov, O, ter Laak, A, Sugawara, T, Stoeckigt, D, Tallant, C, Bennett, J, Monteiro, O, Saez, L.D, Siejka, P, Meier, J, Puetter, V, Weiske, J, Mueller, S, Huber, K.V.M, Hartung, I.V, Haendler, B. | 登録日 | 2017-02-10 | 公開日 | 2017-05-03 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (1.94 Å) | 主引用文献 | Benzoisoquinolinediones as Potent and Selective Inhibitors of BRPF2 and TAF1/TAF1L Bromodomains. J. Med. Chem., 60, 2017
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4TU1
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![BU of 4tu1 by Molmil](/molmil-images/mine/4tu1) | Structure of Toxoplasma gondii fructose 1,6 bisphosphate aldolase | 分子名称: | Fructose-1,6-bisphosphate aldolase, GLYCEROL | 著者 | Boucher, L.E, Bosch, J, Seattle Structural Genomics Center for Infectious Disease (SSGCID) | 登録日 | 2014-06-23 | 公開日 | 2014-09-03 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Structure of Toxoplasma gondii fructose-1,6-bisphosphate aldolase. Acta Crystallogr.,Sect.F, 70, 2014
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4W5V
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![BU of 4w5v by Molmil](/molmil-images/mine/4w5v) | Crystal structure of Human SUMO E2-conjugating enzyme (Ubc9) in complex with E1-activating enzyme (Uba2) ubiquitin fold domain (Ufd) | 分子名称: | FORMIC ACID, GLYCEROL, POTASSIUM ION, ... | 著者 | Boucher, L.E, Reiter, K.H, Matunis, M.J, Bosch, J. | 登録日 | 2014-08-19 | 公開日 | 2015-09-09 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Crystal structure of human SUMO complex To Be Published
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4M1N
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![BU of 4m1n by Molmil](/molmil-images/mine/4m1n) | Crystal structure of Plasmodium falciparum ubiquitin conjugating enzyme UBC9 | 分子名称: | SODIUM ION, Ubiquitin conjugating enzyme UBC9 | 著者 | Boucher, L.E, Reiter, K.H, Bosch, J, Matunis, J.M. | 登録日 | 2013-08-03 | 公開日 | 2013-08-21 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Identification of Biochemically Distinct Properties of the Small Ubiquitin-related Modifier (SUMO) Conjugation Pathway in Plasmodium falciparum. J.Biol.Chem., 288, 2013
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5MG2
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![BU of 5mg2 by Molmil](/molmil-images/mine/5mg2) | Crystal structure of the second bromodomain of human TAF1 in complex with BAY-299 chemical probe | 分子名称: | 1,2-ETHANEDIOL, 6-(3-oxidanylpropyl)-2-(1,3,6-trimethyl-2-oxidanylidene-benzimidazol-5-yl)benzo[de]isoquinoline-1,3-dione, Transcription initiation factor TFIID subunit 1 | 著者 | Tallant, C, Bouche, L, Holton, S.J, Fedorov, O, Siejka, P, Picaud, S, Krojer, T, Srikannathasan, V, von Delft, F, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Hartung, I.V, Haendler, B, Muller, S, Huber, K.V.M, Structural Genomics Consortium (SGC) | 登録日 | 2016-11-20 | 公開日 | 2017-05-03 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | Benzoisoquinolinediones as Potent and Selective Inhibitors of BRPF2 and TAF1/TAF1L Bromodomains. J. Med. Chem., 60, 2017
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4XDI
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![BU of 4xdi by Molmil](/molmil-images/mine/4xdi) | Structure of Chlamydomonas reinhardtii THB1 | 分子名称: | Chlamydomonas reinhardtii THB1, PROTOPORPHYRIN IX CONTAINING FE | 著者 | Rice, S.L, Boucher, L.E, Schlessman, J.L, Bosch, J, Lecomte, J.T.J. | 登録日 | 2014-12-19 | 公開日 | 2015-01-21 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.893 Å) | 主引用文献 | Structure of Chlamydomonas reinhardtii THB1, a group 1 truncated hemoglobin with a rare histidine-lysine heme ligation. Acta Crystallogr.,Sect.F, 71, 2015
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7JGU
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![BU of 7jgu by Molmil](/molmil-images/mine/7jgu) | Structure of FN3tt mut | 分子名称: | Fibronectin type-III domain-containing protein, PENTAETHYLENE GLYCOL | 著者 | Luo, J, Boucher, L.E. | 登録日 | 2020-07-19 | 公開日 | 2021-07-21 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.2 Å) | 主引用文献 | Surface salt bridges contribute to the extreme thermal stability of an FN3-like domain from a thermophilic bacterium. Proteins, 90, 2022
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4JUE
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![BU of 4jue by Molmil](/molmil-images/mine/4jue) | |
8DY5
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![BU of 8dy5 by Molmil](/molmil-images/mine/8dy5) | |
8DY2
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![BU of 8dy2 by Molmil](/molmil-images/mine/8dy2) | Crystal Structure of spFv GLK1 | 分子名称: | SULFATE ION, spFv GLK1 LH | 著者 | Luo, J, Boucher, L.E. | 登録日 | 2022-08-03 | 公開日 | 2023-05-03 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.65 Å) | 主引用文献 | "Stapling" scFv for multispecific biotherapeutics of superior properties. Mabs, 15, 2023
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8DY4
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![BU of 8dy4 by Molmil](/molmil-images/mine/8dy4) | |
8DY0
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![BU of 8dy0 by Molmil](/molmil-images/mine/8dy0) | |
8DY3
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![BU of 8dy3 by Molmil](/molmil-images/mine/8dy3) | |