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PDB: 13 件

5N49
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BRPF2 in complex with Compound 7
分子名称: 2-(1,3,6-trimethyl-2-oxidanylidene-benzimidazol-5-yl)benzo[de]isoquinoline-1,3-dione, Bromodomain-containing protein 1
著者Bouche, L, Christ, C.D, Siegel, S, Fernandez-Montalvan, A.E, Holton, S.J, Fedorov, O, ter Laak, A, Sugawara, T, Stoeckigt, D, Tallant, C, Bennett, J, Monteiro, O, Saez, L.D, Siejka, P, Meier, J, Puetter, V, Weiske, J, Mueller, S, Huber, K.V.M, Hartung, I.V, Haendler, B.
登録日2017-02-10
公開日2017-05-03
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (1.94 Å)
主引用文献Benzoisoquinolinediones as Potent and Selective Inhibitors of BRPF2 and TAF1/TAF1L Bromodomains.
J. Med. Chem., 60, 2017
4TU1
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Structure of Toxoplasma gondii fructose 1,6 bisphosphate aldolase
分子名称: Fructose-1,6-bisphosphate aldolase, GLYCEROL
著者Boucher, L.E, Bosch, J, Seattle Structural Genomics Center for Infectious Disease (SSGCID)
登録日2014-06-23
公開日2014-09-03
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structure of Toxoplasma gondii fructose-1,6-bisphosphate aldolase.
Acta Crystallogr.,Sect.F, 70, 2014
4W5V
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Crystal structure of Human SUMO E2-conjugating enzyme (Ubc9) in complex with E1-activating enzyme (Uba2) ubiquitin fold domain (Ufd)
分子名称: FORMIC ACID, GLYCEROL, POTASSIUM ION, ...
著者Boucher, L.E, Reiter, K.H, Matunis, M.J, Bosch, J.
登録日2014-08-19
公開日2015-09-09
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Crystal structure of human SUMO complex
To Be Published
4M1N
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Crystal structure of Plasmodium falciparum ubiquitin conjugating enzyme UBC9
分子名称: SODIUM ION, Ubiquitin conjugating enzyme UBC9
著者Boucher, L.E, Reiter, K.H, Bosch, J, Matunis, J.M.
登録日2013-08-03
公開日2013-08-21
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Identification of Biochemically Distinct Properties of the Small Ubiquitin-related Modifier (SUMO) Conjugation Pathway in Plasmodium falciparum.
J.Biol.Chem., 288, 2013
5MG2
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Crystal structure of the second bromodomain of human TAF1 in complex with BAY-299 chemical probe
分子名称: 1,2-ETHANEDIOL, 6-(3-oxidanylpropyl)-2-(1,3,6-trimethyl-2-oxidanylidene-benzimidazol-5-yl)benzo[de]isoquinoline-1,3-dione, Transcription initiation factor TFIID subunit 1
著者Tallant, C, Bouche, L, Holton, S.J, Fedorov, O, Siejka, P, Picaud, S, Krojer, T, Srikannathasan, V, von Delft, F, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Hartung, I.V, Haendler, B, Muller, S, Huber, K.V.M, Structural Genomics Consortium (SGC)
登録日2016-11-20
公開日2017-05-03
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Benzoisoquinolinediones as Potent and Selective Inhibitors of BRPF2 and TAF1/TAF1L Bromodomains.
J. Med. Chem., 60, 2017
4XDI
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Structure of Chlamydomonas reinhardtii THB1
分子名称: Chlamydomonas reinhardtii THB1, PROTOPORPHYRIN IX CONTAINING FE
著者Rice, S.L, Boucher, L.E, Schlessman, J.L, Bosch, J, Lecomte, J.T.J.
登録日2014-12-19
公開日2015-01-21
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.893 Å)
主引用文献Structure of Chlamydomonas reinhardtii THB1, a group 1 truncated hemoglobin with a rare histidine-lysine heme ligation.
Acta Crystallogr.,Sect.F, 71, 2015
7JGU
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Structure of FN3tt mut
分子名称: Fibronectin type-III domain-containing protein, PENTAETHYLENE GLYCOL
著者Luo, J, Boucher, L.E.
登録日2020-07-19
公開日2021-07-21
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (1.2 Å)
主引用文献Surface salt bridges contribute to the extreme thermal stability of an FN3-like domain from a thermophilic bacterium.
Proteins, 90, 2022
4JUE
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Crystal structure of Plasmodium falciparum ubiquitin conjugating enzyme UBC9
分子名称: Ubiquitin conjugating enzyme UBC9
著者Reiter, K.H, Boucher, L.E, Bosch, J, Matunis, J.M.
登録日2013-03-24
公開日2013-08-21
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (1.851 Å)
主引用文献Identification of Biochemically Distinct Properties of the Small Ubiquitin-related Modifier (SUMO) Conjugation Pathway in Plasmodium falciparum.
J.Biol.Chem., 288, 2013
8DY5
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Crystal Structure of spFv CAT2200 LH in complex with IL-17A
分子名称: CALCIUM ION, CHLORIDE ION, Interleukin-17A, ...
著者Luo, J, Boucher, L.E.
登録日2022-08-03
公開日2023-05-03
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献"Stapling" scFv for multispecific biotherapeutics of superior properties.
Mabs, 15, 2023
8DY2
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Crystal Structure of spFv GLK1
分子名称: SULFATE ION, spFv GLK1 LH
著者Luo, J, Boucher, L.E.
登録日2022-08-03
公開日2023-05-03
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.65 Å)
主引用文献"Stapling" scFv for multispecific biotherapeutics of superior properties.
Mabs, 15, 2023
8DY4
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Crystal Structure of spFv CAT2200 HL
分子名称: spFv CAT2200 HL
著者Luo, J, Boucher, L.E.
登録日2022-08-03
公開日2023-05-03
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献"Stapling" scFv for multispecific biotherapeutics of superior properties.
Mabs, 15, 2023
8DY0
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BU of 8dy0 by Molmil
Crystal Structure of spFv GLK1 HL
分子名称: spFv GLK1 HL
著者Luo, J, Boucher, L.E.
登録日2022-08-03
公開日2023-05-03
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献"Stapling" scFv for multispecific biotherapeutics of superior properties.
Mabs, 15, 2023
8DY3
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BU of 8dy3 by Molmil
Crystal Structure of spFv GLK2 HL
分子名称: SULFATE ION, spFv GLK2 HL
著者Luo, J, Boucher, L.E.
登録日2022-08-03
公開日2023-05-03
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.509 Å)
主引用文献"Stapling" scFv for multispecific biotherapeutics of superior properties.
Mabs, 15, 2023

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件を2024-07-24に公開中

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