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PDB: 251 件

8CV1
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BU of 8cv1 by Molmil
ACP1-KS-AT domains of mycobacterial Pks13
分子名称: Polyketide synthase PKS13, UNKNOWN LIGAND
著者Kim, S.K, Dickinson, M.S, Finer-Moore, J.S, Rosenberg, O.S, Stroud, R.M.
登録日2022-05-17
公開日2023-02-15
最終更新日2023-03-29
実験手法ELECTRON MICROSCOPY (2.6 Å)
主引用文献Structure and dynamics of the essential endogenous mycobacterial polyketide synthase Pks13.
Nat.Struct.Mol.Biol., 30, 2023
3GAY
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BU of 3gay by Molmil
Structure of Giardia fructose-1,6-biphosphate aldolase in complex with tagatose-1,6-biphosphate
分子名称: 1,6-di-O-phosphono-D-tagatose, Fructose-bisphosphate aldolase, ZINC ION
著者Galkin, A, Herzberg, O.
登録日2009-02-18
公開日2009-03-31
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Structural insights into the substrate binding and stereoselectivity of giardia fructose-1,6-bisphosphate aldolase.
Biochemistry, 48, 2009
1KTW
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IOTA-CARRAGEENASE COMPLEXED TO IOTA-CARRAGEENAN FRAGMENTS
分子名称: 3,6-anhydro-2-O-sulfo-alpha-D-galactopyranose-(1-3)-4-O-sulfo-beta-D-galactopyranose, 3,6-anhydro-2-O-sulfo-alpha-D-galactopyranose-(1-3)-4-O-sulfo-beta-D-galactopyranose-(1-4)-3,6-anhydro-2-O-sulfo-alpha-D-galactopyranose-(1-3)-4-O-sulfo-beta-D-galactopyranose, CALCIUM ION, ...
著者Michel, G, Kahn, R, Dideberg, O.
登録日2002-01-18
公開日2003-06-10
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献The Structural Bases of the Processive Degradation of iota-Carrageenan, a Main Cell Wall Polysaccharide of Red Algae.
J.Mol.Biol., 334, 2003
7UK4
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BU of 7uk4 by Molmil
KS-AT di-domain of mycobacterial Pks13 with endogenous KS ligand bound
分子名称: Polyketide synthase PKS13, UNKNOWN LIGAND
著者Kim, S.K, Dickinson, M.S, Finer-Moore, J.S, Rosenberg, O.S, Stroud, R.M.
登録日2022-03-31
公開日2023-02-15
最終更新日2023-03-29
実験手法ELECTRON MICROSCOPY (1.94 Å)
主引用文献Structure and dynamics of the essential endogenous mycobacterial polyketide synthase Pks13.
Nat.Struct.Mol.Biol., 30, 2023
8SOT
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BU of 8sot by Molmil
Structure of the PPIase domain of borrelial BB0108
分子名称: Basic membrane protein, GLYCEROL
著者Shakya, A.K, Herzberg, O.
登録日2023-04-30
公開日2023-10-11
最終更新日2024-04-24
実験手法X-RAY DIFFRACTION (1.99 Å)
主引用文献A unique borrelial protein facilitates microbial immune evasion.
Mbio, 14, 2023
1MOV
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BU of 1mov by Molmil
Crystal structure of Coral protein mutant
分子名称: GFP-like non-fluorescent chromoprotein, IODIDE ION
著者Prescott, M, Ling, M, Beddoe, T, Oakley, A.J, Dove, S, Hoegh-Guldberg, O, Devenish, R.J, Rossjohn, J.
登録日2002-09-10
公開日2003-04-08
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献The 2.2 a crystal structure of a pocilloporin pigment reveals a nonplanar chromophore conformation.
Structure, 11, 2003
6UMM
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BU of 6umm by Molmil
A complete structure of the ESX-3 translocon complex
分子名称: ESX-3 secretion system ATPase EccB3, ESX-3 secretion system protein EccC3, ESX-3 secretion system protein EccD3, ...
著者Poweleit, N, Rosenberg, O.S.
登録日2019-10-09
公開日2019-10-23
最終更新日2024-03-20
実験手法ELECTRON MICROSCOPY (3.7 Å)
主引用文献A large inner membrane pore defines the ESX translocon
To Be Published
8P33
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BB0238 from Borrelia burgdorferi
分子名称: BB0238
著者Brangulis, K, Foor, S.D, Shakya, A.K, Rana, V.S, Bista, S, Kitsou, C, Ronzetti, M, Linden, S.B, Altieri, A.S, Akopjana, I, Baljinnyam, B, Nelson, D.C, Simeonov, A, Herzberg, O, Caimano, M.J, Pal, U.
登録日2023-05-16
公開日2023-10-11
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献A unique borrelial protein facilitates microbial immune evasion.
Mbio, 14, 2023
8P32
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BB0238 from Borrelia burgdorferi, Se-Met data for Leu240Met mutant
分子名称: BB0238
著者Brangulis, K, Foor, S.D, Shakya, A.K, Rana, V.S, Bista, S, Kitsou, C, Ronzetti, M, Linden, S.B, Altieri, A.S, Akopjana, I, Baljinnyam, B, Nelson, D.C, Simeonov, A, Herzberg, O, Caimano, M.J, Pal, U.
登録日2023-05-16
公開日2023-10-11
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献A unique borrelial protein facilitates microbial immune evasion.
Mbio, 14, 2023
8CV0
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BU of 8cv0 by Molmil
KS-AT domains of mycobacterial Pks13 with outward AT conformation
分子名称: Polyketide synthase PKS13, UNKNOWN LIGAND
著者Kim, S.K, Dickinson, M.S, Finer-Moore, J.S, Rosenberg, O.S, Stroud, R.M.
登録日2022-05-17
公開日2023-02-15
最終更新日2023-03-29
実験手法ELECTRON MICROSCOPY (3.1 Å)
主引用文献Structure and dynamics of the essential endogenous mycobacterial polyketide synthase Pks13.
Nat.Struct.Mol.Biol., 30, 2023
8CUZ
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BU of 8cuz by Molmil
KS-AT domains of mycobacterial Pks13 with inward AT conformation
分子名称: Polyketide synthase PKS13, UNKNOWN LIGAND
著者Kim, S.K, Dickinson, M.S, Finer-Moore, J.S, Rosenberg, O.S, Stroud, R.M.
登録日2022-05-17
公開日2023-02-15
最終更新日2023-03-29
実験手法ELECTRON MICROSCOPY (3 Å)
主引用文献Structure and dynamics of the essential endogenous mycobacterial polyketide synthase Pks13.
Nat.Struct.Mol.Biol., 30, 2023
5DPX
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BU of 5dpx by Molmil
1,2,4-Triazole-3-thione compounds as inhibitors of L1, di-zinc metallo-beta-lactamases.
分子名称: 5-(2-methylphenyl)-3H-1,2,4-triazole-3-thione, Metallo-beta-lactamase L1 type 3, SULFATE ION, ...
著者Nauton, L, Garau, G, Khan, R, Dideberg, O.
登録日2015-09-14
公開日2017-01-11
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献1,2,4-Triazole-3-thione Compounds as Inhibitors of Dizinc Metallo-beta-lactamases.
ChemMedChem, 12, 2017
4UUQ
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BU of 4uuq by Molmil
Crystal structure of human mono-glyceride lipase in complex with SAR127303
分子名称: 4-({[(4-chlorophenyl)sulfonyl]amino}methyl)piperidine-1-carboxylic acid, MONOGLYCERIDE LIPASE
著者Griebel, G, Pichat, P, Beeske, S, Leroy, T, Redon, N, Francon, D, Bert, L, Even, L, Lopez-Grancha, M, Tolstykh, T, Sun, F, Yu, Q, Brittain, S, Arlt, H, He, T, Zhang, B, Wiederschain, D, Bertrand, T, Houtman, J, Rak, A, Vallee, F, Michot, N, Auge, F, Menet, V, Bergis, O.E, George, P, Avenet, P, Mikol, V, Didier, M, Escoubet, J.
登録日2014-07-30
公開日2015-01-21
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.36 Å)
主引用文献Selective Blockade of the Hydrolysis of the Endocannabinoid 2-Arachidonoylglycerol Impairs Learning and Memory Performance While Producing Antinociceptive Activity in Rodents.
Sci.Rep., 5, 2015
3GAK
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BU of 3gak by Molmil
Structure of Giardia fructose-1,6-biphosphate aldolase
分子名称: Fructose-bisphosphate aldolase, SULFATE ION, ZINC ION
著者Galkin, A, Herzberg, O.
登録日2009-02-17
公開日2009-03-31
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Structural insights into the substrate binding and stereoselectivity of giardia fructose-1,6-bisphosphate aldolase.
Biochemistry, 48, 2009
3ZNB
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BU of 3znb by Molmil
METALLO-BETA-LACTAMASE (ZN, HG-BOUND FORM)
分子名称: MERCURY (II) ION, METALLO-BETA-LACTAMASE, SODIUM ION, ...
著者Concha, N.O, Herzberg, O.
登録日1997-10-15
公開日1998-01-28
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Crystal structures of the cadmium- and mercury-substituted metallo-beta-lactamase from Bacteroides fragilis.
Protein Sci., 6, 1997
1F76
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BU of 1f76 by Molmil
ESCHERICHIA COLI DIHYDROOROTATE DEHYDROGENASE
分子名称: Dihydroorotate dehydrogenase (quinone), FLAVIN MONONUCLEOTIDE, FORMIC ACID, ...
著者Norager, S, Jensen, K.F, Bjornberg, O, Larsen, S.
登録日2000-06-26
公開日2002-10-16
最終更新日2014-03-12
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献E. coli Dihydroorotate Dehydrogenase Reveals Structural and Functional Distinction between different classes of dihydroorotate dehydrogenases
Structure, 10, 2002
2ZNB
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BU of 2znb by Molmil
METALLO-BETA-LACTAMASE (CADMIUM-BOUND FORM)
分子名称: CADMIUM ION, METALLO-BETA-LACTAMASE, SODIUM ION
著者Concha, N.O, Herzberg, O.
登録日1997-10-14
公開日1998-01-28
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献Crystal structures of the cadmium- and mercury-substituted metallo-beta-lactamase from Bacteroides fragilis.
Protein Sci., 6, 1997
1J85
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Structure of YibK from Haemophilus influenzae (HI0766), a truncated sequence homolog of tRNA (guanosine-2'-O-) methyltransferase (SpoU)
分子名称: YibK
著者Lim, K, Zhang, H, Toedt, J, Tempcyzk, A, Krajewski, W, Howard, A, Eisenstein, E, Herzberg, O, Structure 2 Function Project (S2F)
登録日2001-05-20
公開日2003-02-25
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structure of the YibK methyltransferase from Haemophilus influenzae (HI0766): A cofactor bound at a site formed by a knot
Proteins, 51, 2003
1X8I
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Crystal Structure of the Zinc Carbapenemase CphA in Complex with the Antibiotic Biapenem
分子名称: 5H-PYRAZOLO(1,2-A)(1,2,4)TRIAZOL-4-IUM, 6-((2-CARBOXY-6-(1-HYDROXYETHYL)-4-METHYL-7-OXO-1-AZABICYCLO(3.2.0)HEPT-2-EN-3-YL)THIO)-6,7-DIHYDRO-, HYDROXIDE, ...
著者Garau, G, Dideberg, O.
登録日2004-08-18
公開日2004-12-28
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献A Metallo-beta-lactamase Enzyme in Action: Crystal Structures of the Monozinc Carbapenemase CphA and its Complex with Biapenem
J.Mol.Biol., 345, 2005
1X8G
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Crystal Structure of the Mono-Zinc Carbapenemase CphA from Aeromonas Hydrophyla
分子名称: Beta-lactamase, CARBONATE ION, SULFATE ION, ...
著者Garau, G, Dideberg, O.
登録日2004-08-18
公開日2004-12-28
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献A Metallo-beta-lactamase Enzyme in Action: Crystal Structures of the Monozinc Carbapenemase CphA and its Complex with Biapenem
J.Mol.Biol., 345, 2005
1BLH
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BU of 1blh by Molmil
STRUCTURE OF A PHOSPHONATE-INHIBITED BETA-LACTAMASE. AN ANALOG OF THE TETRAHEDRAL TRANSITION STATE(SLASH)INTERMEDIATE OF BETA-LACTAM HYDROLYSIS
分子名称: BETA-LACTAMASE, [[N-(BENZYLOXYCARBONYL)AMINO]METHYL]PHOSPHATE
著者Chen, C.C.H, Herzberg, O.
登録日1993-09-30
公開日1994-08-31
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Structure of a phosphonate-inhibited beta-lactamase. An analog of the tetrahedral transition state/intermediate of beta-lactam hydrolysis.
J.Mol.Biol., 234, 1993
1JUE
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BU of 1jue by Molmil
1.8 A resolution structure of native lactococcus lactis dihydroorotate dehydrogenase A
分子名称: ACETIC ACID, FLAVIN MONONUCLEOTIDE, GLYCEROL, ...
著者Norager, S, Arent, S, Bjornberg, O, Ottosen, M, Lo Leggio, L, Jensen, K.F, Larsen, S.
登録日2001-08-24
公開日2003-09-09
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Lactococcus lactis dihydroorotate dehydrogenase A mutants reveal important facets of the enzymatic function
J.Biol.Chem., 278, 2003
4OLC
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BU of 4olc by Molmil
Carbamate kinase from Giardia lamblia thiocarbamoylated by disulfiram on Cys242
分子名称: CITRIC ACID, Carbamate kinase, DIETHYLCARBAMODITHIOIC ACID
著者Lim, K, Herzberg, O.
登録日2014-01-23
公開日2014-02-26
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Structural Basis for Inactivation of Giardia lamblia Carbamate Kinase by Disulfiram.
J.Biol.Chem., 289, 2014
2QDS
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BU of 2qds by Molmil
Crystal Structure of the Zinc Carbapenemase CPHA in Complex with the Inhibitor D-Captopril
分子名称: 1-(3-MERCAPTO-2-METHYL-PROPIONYL)-PYRROLIDINE-2-CARBOXYLIC ACID, Beta-lactamase, GLYCEROL, ...
著者Garau, G, Dideberg, O.
登録日2007-06-21
公開日2007-07-17
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.66 Å)
主引用文献Structural basis for the broad-spectrum inhibition of metallo-beta-lactamases by thiols.
Org.Biomol.Chem., 6, 2008
2GFK
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Crystal structure of the zinc-beta-lactamase l1 from stenotrophomonas maltophilia (inhibitor 2)
分子名称: 2,5-DIPHENYLFURAN-3,4-DICARBOXYLIC ACID, DI(HYDROXYETHYL)ETHER, Metallo-beta-lactamase L1, ...
著者Nauton, L, Garau, G, Kahn, R, Dideberg, O.
登録日2006-03-22
公開日2007-03-27
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Structural insights into the design of inhibitors for the L1 metallo-beta-lactamase from Stenotrophomonas maltophilia.
J.Mol.Biol., 375, 2008

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