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PDB: 1 件

8C12
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Identification of an intermediate activation state of PAK5 reveals a novel mechanism of kinase inhibition.
分子名称: PAK5-Af17, Serine/threonine-protein kinase PAK 5
著者Martin, H.L, Turner, A.L, Trinh, C.H, Bayliss, R.W, Tomlinson, D.C.
登録日2022-12-19
公開日2023-10-25
実験手法X-RAY DIFFRACTION (1.549 Å)
主引用文献Affimer-mediated locking of p21-activated kinase 5 in an intermediate activation state results in kinase inhibition.
Cell Rep, 42, 2023

222926

件を2024-07-24に公開中

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