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8TWY
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Structure of PIK3CA with covalent inhibitor ALO26
Descriptor: 1-(4-{[2-(4-{(4P)-4-[2-amino-4-(difluoromethyl)pyrimidin-5-yl]-6-[(3S)-3-methylmorpholin-4-yl]-1,3,5-triazin-2-yl}piperazin-1-yl)-2-oxoethoxy]methyl}piperidin-1-yl)prop-2-en-1-one, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
Authors:Burke, J.E, Barlow-Busch, I.
Deposit date:2023-08-21
Release date:2024-08-28
Method:X-RAY DIFFRACTION (2.67 Å)
Cite:Structure of PIK3CA with covalent inhibitor ALO26
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PDB entries from 2024-10-09

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