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PDB: 2 件

5A14
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BU of 5a14 by Molmil
Human CDK2 with type II inhibitor
分子名称: 1-[4-(2-azanylpyrimidin-4-yl)oxyphenyl]-3-[4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]urea, CYCLIN-DEPENDENT KINASE 2
著者Alexander, L.T, Elkins, J.M, Kopec, J, Fedorov, O, Savitsky, P.A, Moebitz, H, Cowan-Jacob, S.W, Szklarz, M, Pike, A.C.W, Carpenter, E.P, Krojer, T, Bountra, C, Edwards, A.M, Knapp, S.
登録日2015-04-27
公開日2015-07-22
最終更新日2019-10-23
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Type II Inhibitors Targeting Cdk2.
Acs Chem.Biol., 10, 2015
6QXK
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Human PIM1 bound to OX0999
分子名称: 2-[(1-methylpiperidin-4-yl)methylamino]-5-[[2-[4-(trifluoromethyloxy)phenyl]-1,3-thiazol-4-yl]methyl]-1,3-thiazol-4-one, Pimtide, Serine/threonine-protein kinase pim-1
著者Alexander, L.T, Elkins, J.M, Russell, A, Bountra, C, Edwards, A.M, Knapp, S.
登録日2019-03-07
公開日2019-04-24
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献PIM1 bound to OX0999
To Be Published

222624

件を2024-07-17に公開中

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