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PDB: 1 results

9EP8
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BU of 9ep8 by Molmil
Crystal structure of ROCK2 in complex with a 8-(azaindolyl)-benzoazepinone inhibitor
Descriptor: 1,2-ETHANEDIOL, 8-(azaindolyl)-benzoazepinone, Rho-associated protein kinase 2
Authors:Pala, D, Clark, D, Pioselli, B, Accetta, A, Rancati, F.
Deposit date:2024-03-18
Release date:2024-09-25
Method:X-RAY DIFFRACTION (2.63 Å)
Cite:Design and synthesis of novel 8-(azaindolyl)-benzoazepinones as potent and selective ROCK inhibitors
Rsc Med Chem, 2024

225399

數據於2024-09-25公開中

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