9EP8
| Crystal structure of ROCK2 in complex with a 8-(azaindolyl)-benzoazepinone inhibitor | Descriptor: | 1,2-ETHANEDIOL, 8-(azaindolyl)-benzoazepinone, Rho-associated protein kinase 2 | Authors: | Pala, D, Clark, D, Pioselli, B, Accetta, A, Rancati, F. | Deposit date: | 2024-03-18 | Release date: | 2024-09-25 | Method: | X-RAY DIFFRACTION (2.63 Å) | Cite: | Design and synthesis of novel 8-(azaindolyl)-benzoazepinones as potent and selective ROCK inhibitors Rsc Med Chem, 2024
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