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1E37
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BU of 1e37 by Molmil
PORCINE PANCREATIC ELASTASE COMPLEXED WITH (3S, 4S)N-PARA-NITROBENZENESULPHONYL -3-ETHYL-4-(CARBOXYLIC ACID)PYRROLIDIN-2-ONE SOAKED IN PH 9 BUFFER FOR 1 MINUTE
分子名称: (2S,3S)-3-FORMYL-2-({[(4-NITROPHENYL)SULFONYL]AMINO}METHYL)PENTANOIC ACID, CALCIUM ION, ELASTASE, ...
著者Wright, P.A, Wilmouth, R.C, Clifton, I.J, Schofield, C.J.
登録日2000-06-06
公開日2000-10-18
最終更新日2023-12-06
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献'Ph-Jump' Crystallographic Analyses of Gamma-Lactam-Porcine Pancreatic Elastase Complexes
Biochem.J., 351, 2000
1E38
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BU of 1e38 by Molmil
PORCINE PANCREATIC ELASTASE COMPLEXED WITH (3S, 4S)N-PARA-NITROBENZENESULPHONYL -3-ETHYL-4-(CARBOXYLIC ACID)PYRROLIDIN-2-ONE SOAKED IN PH 9 BUFFER FOR 2 MINUTES
分子名称: (2S,3S)-3-FORMYL-2-({[(4-NITROPHENYL)SULFONYL]AMINO}METHYL)PENTANOIC ACID, CALCIUM ION, ELASTASE, ...
著者Wright, P.A, Wilmouth, R.C, Clifton, I.J, Schofield, C.J.
登録日2000-06-06
公開日2000-10-18
最終更新日2023-12-06
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献'Ph-Jump' Crystallographic Analyses of Gamma-Lactam-Porcine Pancreatic Elastase Complexes
Biochem.J., 351, 2000
1E36
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BU of 1e36 by Molmil
PORCINE PANCREATIC ELASTASE COMPLEXED WITH (3S, 4S)N-PARA-NITROBENZENESULPHONYL -3-ETHYL-4-(CARBOXYLIC ACID)PYRROLIDIN-2-ONE
分子名称: (2S,3S)-3-FORMYL-2-({[(4-NITROPHENYL)SULFONYL]AMINO}METHYL)PENTANOIC ACID, CALCIUM ION, ELASTASE, ...
著者Wright, P.A, Wilmouth, R.C, Clifton, I.J, Schofield, C.J.
登録日2000-06-06
公開日2000-10-18
最終更新日2023-12-06
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献'Ph-Jump' Crystallographic Analyses of Gamma-Lactam-Porcine Pancreatic Elastase Complexes
Biochem.J., 351, 2000
1E35
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BU of 1e35 by Molmil
PORCINE PANCREATIC ELASTASE COMPLEXED WITH (3S, 4S)N-PARA-TOLUENESULPHONYL -3-ETHYL-4-(CARBOXYLIC ACID)PYRROLIDIN-2-ONE SOAKED IN PH 9 BUFFER FOR TWO MINUTES
分子名称: (2S,3S)-3-FORMYL-2-({[(4-METHYLPHENYL)SULFONYL]AMINO}METHYL)PENTANOIC ACID, CALCIUM ION, ELASTASE, ...
著者Wright, P.A, Wilmouth, R.C, Clifton, I.J, Schofield, C.J.
登録日2000-06-06
公開日2000-10-18
最終更新日2023-12-06
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献'Ph-Jump' Crystallographic Analyses of Gamma-Lactam-Porcine Pancreatic Elastase Complexes
Biochem.J., 351, 2000
1E34
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BU of 1e34 by Molmil
PORCINE PANCREATIC ELASTASE COMPLEXED WITH (3S, 4S)N-PARA- TOLUENESULPHONYL-3-ETHYL-4-(CARBOXYLIC ACID) PYRROLIDIN-2-ONE SOAKED IN PH 9 BUFFER FOR ONE MINUTE
分子名称: (2S,3S)-3-FORMYL-2-({[(4-METHYLPHENYL)SULFONYL]AMINO}METHYL)PENTANOIC ACID, CALCIUM ION, ELASTASE, ...
著者Wright, P.A, Wilmouth, R.C, Clifton, I.J, Schofield, C.J.
登録日2000-06-06
公開日2000-10-18
最終更新日2023-12-06
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献`Ph-Jump' Crystallographic Analyses of Gamma-Lactam-Porcine Pancreatic Elastase Complexes
Biochem.J., 351, 2000
1H9L
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BU of 1h9l by Molmil
PORCINE PANCREATIC ELASTASE COMPLEXED WITH ACETYL-VAL-GLU-PRO-ILE-COOH
分子名称: CALCIUM ION, ELASTASE, PEPTIDE INHIBITOR, ...
著者Wright, P.A, Wilmouth, R.C, Clifton, I.J, Schofield, C.J.
登録日2001-03-13
公開日2001-11-27
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.67 Å)
主引用文献Kinetic and Crystallographic Analysis of Complexes Formed between Elastase and Peptides from Beta-Casein
Eur.J.Biochem., 268, 2001
1HAY
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BU of 1hay by Molmil
Snapshots of serine protease catalysis: (B) acyl-enzyme intermediate between porcine pancreatic elastase and human beta-casomorphin-7 jumped to pH 10 for 10 seconds
分子名称: CALCIUM ION, ELASTASE 1, SULFATE ION
著者Wilmouth, R.C, Edman, K, Neutze, R, Wright, P.A, Clifton, I.J, Schneider, T.R, Schofield, C.J, Hajdu, J.
登録日2001-04-10
公開日2001-08-02
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献X-Ray Snapshots of Serine Protease Catalysis Reveal a Tetrahedral Intermediate
Nat.Struct.Biol., 8, 2001
1GVK
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BU of 1gvk by Molmil
Porcine pancreatic elastase acyl enzyme at 0.95 A resolution
分子名称: CALCIUM ION, ELASTASE 1, PEPTIDE INHIBITOR, ...
著者Katona, G, Wilmouth, R.C, Wright, P.A, Berglund, G.I, Hajdu, J, Neutze, R, Schofield, C.J.
登録日2002-02-14
公開日2002-07-19
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (0.94 Å)
主引用文献X-Ray Structure of a Serine Protease Acyl-Enzyme Complex at 0.95-A Resolution.
J.Biol.Chem., 277, 2002
1HAX
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BU of 1hax by Molmil
Snapshots of serine protease catalysis: (A) acyl-enzyme intermediate between porcine pancreatic elastase and human beta-casomorphin-7 at pH 5
分子名称: BETA-CASOMORPHIN-7, CALCIUM ION, ELASTASE 1, ...
著者Wilmouth, R.C, Edman, K, Neutze, R, Wright, P.A, Clifton, I.J, Schneider, T.R, Schofield, C.J, Hajdu, J.
登録日2001-04-10
公開日2001-08-02
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献X-Ray Snapshots of Serine Protease Catalysis Reveal a Tetrahedral Intermediate
Nat.Struct.Biol., 8, 2001
1HAZ
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BU of 1haz by Molmil
Snapshots of serine protease catalysis: (C) acyl-enzyme intermediate between porcine pancreatic elastase and human beta-casomorphin-7 jumped to pH 9 for 1 minute
分子名称: BETA-CASOMORPHIN-7, CALCIUM ION, ELASTASE 1, ...
著者Wilmouth, R.C, Edman, K, Neutze, R, Wright, P.A, Clifton, I.J, Schneider, T.R, Schofield, C.J, Hajdu, J.
登録日2001-04-10
公開日2001-08-02
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献X-Ray Snapshots of Serine Protease Catalysis Reveal a Tetrahedral Intermediate
Nat.Struct.Biol., 8, 2001
1HB0
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BU of 1hb0 by Molmil
Snapshots of serine protease catalysis: (D) acyl-enzyme intermediate between porcine pancreatic elastase and human beta-casomorphin-7 jumped to pH 10 for 2 minutes
分子名称: CALCIUM ION, ELASTASE 1, SULFATE ION
著者Wilmouth, R.C, Edman, K, Neutze, R, Wright, P.A, Clifton, I.J, Schneider, T.R, Schofield, C.J, Hajdu, J.
登録日2001-04-10
公開日2001-08-02
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献X-Ray Snapshots of Serine Protease Catalysis Reveal a Tetrahedral Intermediate
Nat.Struct.Biol., 8, 2001
1QGF
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BU of 1qgf by Molmil
PORCINE PANCREATIC ELASTASE COMPLEXED WITH (3R, 4S)N-PARA-TOLUENESULPHONYL-3-ETHYL-4-(CARBOXYLIC ACID)PYRROLIDIN-2-ONE
分子名称: (2S,3S)-3-FORMYL-2-({[(4-METHYLPHENYL)SULFONYL]AMINO}METHYL)PENTANOIC ACID, CALCIUM ION, ELASTASE, ...
著者Wilmouth, R.C, Kassamally, S, Westwood, N.J, Sheppard, R.J, Claridge, T.D.W, Wright, P.A, Pritchard, G.J, Schofield, C.J.
登録日1999-04-27
公開日1999-12-29
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Mechanistic insights into the inhibition of serine proteases by monocyclic lactams.
Biochemistry, 38, 1999
2BDB
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BU of 2bdb by Molmil
Porcine pancreatic elastase complexed with Asn-Pro-Ile and Ala-Ala at pH 5.0
分子名称: ALANINE, CALCIUM ION, Elastase-1, ...
著者Liu, B, Schofield, C.J, Wilmouth, R.C.
登録日2005-10-20
公開日2006-05-30
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Structural analyses on intermediates in serine protease catalysis
J.Biol.Chem., 281, 2006
2BDA
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BU of 2bda by Molmil
Porcine pancreatic elastase complexed with N-acetyl-NPI and Ala-Ala at pH 5.0
分子名称: ALANINE, CALCIUM ION, Elastase-1, ...
著者Liu, B, Schofield, C.J, Wilmouth, R.C.
登録日2005-10-20
公開日2006-05-30
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Structural analyses on intermediates in serine protease catalysis
J.Biol.Chem., 281, 2006
2BDC
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BU of 2bdc by Molmil
Porcine pancreatic elastase complexed with Asn-Pro-Ile at pH 5.0
分子名称: CALCIUM ION, Elastase-1, SULFATE ION
著者Liu, B, Schofield, C.J, Wilmouth, R.C.
登録日2005-10-20
公開日2006-05-30
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Structural analyses on intermediates in serine protease catalysis
J.Biol.Chem., 281, 2006
2H1U
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BU of 2h1u by Molmil
Porcine pancreatic elastase complexed with MetPheLeuGlu at pH 5.0
分子名称: CALCIUM ION, Elastase-1, MFLE, ...
著者Liu, B, Schofield, C.J, Wilmouth, R.C.
登録日2006-05-17
公開日2006-05-30
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Structural analyses on intermediates in serine protease catalysis.
J.Biol.Chem., 281, 2006
2BB4
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BU of 2bb4 by Molmil
Porcine pancreatic elastase complexed with beta-casomorphin-7 and Asp-Phe at pH 5.0
分子名称: ASPARTIC ACID, CALCIUM ION, Elastase-1, ...
著者Liu, B, Schofield, C.J, Wilmouth, R.C.
登録日2005-10-17
公開日2006-05-30
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Structural analyses on intermediates in serine protease catalysis
J.Biol.Chem., 281, 2006
2BD2
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BU of 2bd2 by Molmil
Porcine pancreatic elastase complexed with beta-casomorphin-7 and Arg-Phe at pH 5.0
分子名称: ARGININE, CALCIUM ION, Elastase-1, ...
著者Liu, B, Schofield, C.J, Wilmouth, R.C.
登録日2005-10-20
公開日2006-05-30
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Structural analyses on intermediates in serine protease catalysis
J.Biol.Chem., 281, 2006
2BD3
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BU of 2bd3 by Molmil
Porcine pancreatic elastase complexed with beta-casomorphin-7 and Lys-Ala-NH2 at pH 5.0
分子名称: ALANINE, CALCIUM ION, Elastase-1, ...
著者Liu, B, Schofield, C.J, Wilmouth, R.C.
登録日2005-10-20
公開日2006-05-30
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Structural analyses on intermediates in serine protease catalysis
J.Biol.Chem., 281, 2006
2BD4
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BU of 2bd4 by Molmil
Porcine pancreatic elastase complexed with beta-casomorphin-7 and Lys-Ser at pH 5.0
分子名称: CALCIUM ION, Elastase-1, LYSINE, ...
著者Liu, B, Schofield, C.J, Wilmouth, R.C.
登録日2005-10-20
公開日2006-05-30
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Structural analyses on intermediates in serine protease catalysis
J.Biol.Chem., 281, 2006
2BD7
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BU of 2bd7 by Molmil
Porcine pancreatic elastase complexed with beta-casomorphin-7 and Arg-Phe at pH 5.0 (50 min soak)
分子名称: ARGININE, CALCIUM ION, Elastase-1, ...
著者Liu, B, Schofield, C.J, Wilmouth, R.C.
登録日2005-10-20
公開日2006-05-30
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Structural analyses on intermediates in serine protease catalysis
J.Biol.Chem., 281, 2006
2BD9
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BU of 2bd9 by Molmil
Porcine pancreatic elastase complexed with beta-casomorphin-7 and Arg-Phe at pH 5.0 (50 min soak) and immersed in pH 9 buffer for 28 seconds (2nd pH jump)
分子名称: CALCIUM ION, Elastase-1, SULFATE ION
著者Liu, B, Schofield, C.J, Wilmouth, R.C.
登録日2005-10-20
公開日2006-05-30
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Structural analyses on intermediates in serine protease catalysis
J.Biol.Chem., 281, 2006
2BD8
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BU of 2bd8 by Molmil
Porcine pancreatic elastase complexed with beta-casomorphin-7 and Arg-Phe at pH 5.0 (50 min soak) and immersed in pH 9 buffer for 30 seconds
分子名称: ARGININE, CALCIUM ION, Elastase-1, ...
著者Liu, B, Schofield, C.J, Wilmouth, R.C.
登録日2005-10-20
公開日2006-05-30
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Structural analyses on intermediates in serine protease catalysis
J.Biol.Chem., 281, 2006
2BD5
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BU of 2bd5 by Molmil
Porcine pancreatic elastase complexed with beta-casomorphin-7 and Lys-Ser at pH 5 and immersed in pH 9 buffer for 30 seconds
分子名称: CALCIUM ION, Elastase-1, LYSINE, ...
著者Liu, B, Schofield, C.J, Wilmouth, R.C.
登録日2005-10-20
公開日2006-05-30
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Structural analyses on intermediates in serine protease catalysis
J.Biol.Chem., 281, 2006

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