4CP3
| The structure of BCL6 BTB (POZ) domain in complex with the ansamycin antibiotic rifabutin. | 分子名称: | B-CELL LYMPHOMA 6 PROTEIN, RIFABUTIN | 著者 | Evans, S.E, Fairall, L, Goult, B.T, Jamieson, A.G, Ferrigno, P.K, Ford, R, Wagner, S.D, Schwabe, J.W.R. | 登録日 | 2014-01-31 | 公開日 | 2014-03-19 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | The Ansamycin Antibiotic, Rifamycin Sv, Inhibits Bcl6 Transcriptional Repression and Forms a Complex with the Bcl6-Btb/Poz Domain. Plos One, 9, 2014
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7BDE
| HUMAN BCL6 BTB-DOMAIN IN COMPLEX WITH GSK137 | 分子名称: | 5-[(5S,7R)-3-fluoranyl-7-(2-methylpyridin-3-yl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-5-yl]quinolin-2-amine, DIMETHYL SULFOXIDE, GLYCEROL, ... | 著者 | Somers, D.O. | 登録日 | 2020-12-21 | 公開日 | 2021-07-28 | 最終更新日 | 2021-08-18 | 実験手法 | X-RAY DIFFRACTION (2.044 Å) | 主引用文献 | GSK137, a potent small-molecule BCL6 inhibitor with in vivo activity, suppresses antibody responses in mice. J.Biol.Chem., 297, 2021
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