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4ZY4
Crystal structure of P21 activated kinase 1 in complex with an inhibitor compound 4
Descriptor:
2-(4-aminopiperidin-1-yl)-N-(5-cyclopropyl-1H-pyrazol-3-yl)thieno[3,2-d]pyrimidin-4-amine, DIMETHYL SULFOXIDE, SULFATE ION, ...
Authors:
Rouge, R
,
Wang, W.
Deposit date:
2015-05-21
Release date:
2015-07-01
Last modified:
2015-07-15
Method:
X-RAY DIFFRACTION (2.6 Å)
Cite:
Structure-Guided Design of Group I Selective p21-Activated Kinase Inhibitors.
J.Med.Chem., 58, 2015
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PDB entries from 2024-05-15