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Sjoegren syndrome/scleroderma autoantigen 1 (SSSCA1)
Descriptor:	FORMIC ACID, Sjoegren syndrome/scleroderma autoantigen 1, ZINC ION
Authors:	Morth, J.P, Perdreau-Dahl, H.
Deposit date:	2018-08-17
Release date:	2020-03-18
Last modified:	2024-05-15
Method:	X-RAY DIFFRACTION (2.3 Å)
Cite:	Sjogren syndrome/scleroderma autoantigen 1 is a direct Tankyrase binding partner in cancer cells. Commun Biol, 3, 2020

Structural basis and SAR for OD 270, a lead stage 1,2,4-triazole based specific Tankyrase1/2 inhibitor
Descriptor:	4-{5-[(E)-2-{4-(2-chlorophenyl)-5-[5-(methylsulfonyl)pyridin-2-yl]-4H-1,2,4-triazol-3-yl}ethenyl]-1,3,4-oxadiazol-2-yl}benzonitrile, NICOTINAMIDE, Tankyrase-2, ...
Authors:	Perdreau, H, Ekblad, B, Voronkov, A, Holsworth, D.D, Waaler, J, Drewes, G, Schueler, H, Krauss, S, Morth, J.P.
Deposit date:	2012-11-13
Release date:	2013-03-20
Last modified:	2023-09-20
Method:	X-RAY DIFFRACTION (2.8 Å)
Cite:	Structural Basis and SAR for G007-LK, a Lead Stage 1,2,4-Triazole Based Specific Tankyrase 1/2 Inhibitor. J.Med.Chem., 56, 2013