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5JVD
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BU of 5jvd by Molmil
Tubulin-TUB092 complex
分子名称: (2E)-3-(3-hydroxy-4-methoxyphenyl)-1-(7-methoxy-2H-1,3-benzodioxol-5-yl)-2-methylprop-2-en-1-one, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CALCIUM ION, ...
著者Canela, M.-D, Noppen, S, Bueno, O, Prota, A.E, Bargsten, K, Saez-Calvo, G, Jimeno, M.-L, Benkheil, M, Ribatti, D, Velazquez, S, Camarasa, M.-J, Diaz, J.F, Steinmetz, M.O, Priego, E.-M, Perez-Perez, M.-J, Liekens, S.
登録日2016-05-11
公開日2016-06-08
最終更新日2017-09-06
実験手法X-RAY DIFFRACTION (2.393 Å)
主引用文献Antivascular and antitumor properties of the tubulin-binding chalcone TUB091.
Oncotarget, 8, 2017
6UH7
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BU of 6uh7 by Molmil
EV-A71 strain 11316 complexed with MADAL compound 30
分子名称: SPHINGOSINE, VP1, VP2, ...
著者Lee, H, Hafenstein, S.
登録日2019-09-26
公開日2019-12-18
最終更新日2024-03-20
実験手法ELECTRON MICROSCOPY (2.87 Å)
主引用文献Scaffold Simplification Strategy Leads to a Novel Generation of Dual Human Immunodeficiency Virus and Enterovirus-A71 Entry Inhibitors.
J.Med.Chem., 63, 2020
6UH6
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BU of 6uh6 by Molmil
EV-A71 strain 11316 complexed with MADAL compound 22
分子名称: SPHINGOSINE, VP1, VP2, ...
著者Lee, H, Hafenstein, S.
登録日2019-09-26
公開日2019-12-18
最終更新日2024-03-20
実験手法ELECTRON MICROSCOPY (2.98 Å)
主引用文献Scaffold Simplification Strategy Leads to a Novel Generation of Dual Human Immunodeficiency Virus and Enterovirus-A71 Entry Inhibitors.
J.Med.Chem., 63, 2020
6UH1
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BU of 6uh1 by Molmil
Structure of the EVA71 strain 11316 capsid
分子名称: SPHINGOSINE, VP1, VP2, ...
著者Lee, H, Hafenstein, S.
登録日2019-09-26
公開日2019-12-18
最終更新日2024-03-20
実験手法ELECTRON MICROSCOPY (3.04 Å)
主引用文献Scaffold Simplification Strategy Leads to a Novel Generation of Dual Human Immunodeficiency Virus and Enterovirus-A71 Entry Inhibitors.
J.Med.Chem., 63, 2020
5OUG
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BU of 5oug by Molmil
Humanized alpha-AChBP (acetylcholine binding protein) in complex with lobeline and allosteric binder fragment 4.
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 4,5-dibromo-N-(3-hydroxypropyl)-1H-pyrrole-2-carboxamide, Alpha-Lobeline, ...
著者Delbart, F, Gruss, F, Ulens, C.
登録日2017-08-23
公開日2017-12-20
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2.57 Å)
主引用文献An allosteric binding site of the alpha 7 nicotinic acetylcholine receptor revealed in a humanized acetylcholine-binding protein.
J. Biol. Chem., 293, 2018
5OUH
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BU of 5ouh by Molmil
Humanized alpha-AChBP (acetylcholine binding protein) in complex with lobeline.
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Acetylcholine binding protein, Alpha-Lobeline, ...
著者Delbart, F, Gruss, F, Ulens, C.
登録日2017-08-23
公開日2017-11-29
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献An allosteric binding site of the alpha 7 nicotinic acetylcholine receptor revealed in a humanized acetylcholine-binding protein.
J. Biol. Chem., 293, 2018
5OUI
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BU of 5oui by Molmil
Humanized alpha-AChBP (acetylcholine binding protein) in complex with allosteric binder fragment CU2017
分子名称: (3~{R})-~{N}-(5-bromanylpyridin-2-yl)piperidine-3-carboxamide, 1,2-ETHANEDIOL, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Delbart, F, Gruss, F, Ulens, C.
登録日2017-08-23
公開日2017-11-29
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献An allosteric binding site of the alpha 7 nicotinic acetylcholine receptor revealed in a humanized acetylcholine-binding protein.
J. Biol. Chem., 293, 2018

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件を2024-04-24に公開中

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