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5TQH
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BU of 5tqh by Molmil
IDH1 R132H mutant in complex with IDH889
分子名称: (4S)-3-[2-({(1S)-1-[5-(4-fluoro-3-methylphenyl)pyrimidin-2-yl]ethyl}amino)pyrimidin-4-yl]-4-(propan-2-yl)-1,3-oxazolidin-2-one, CITRATE ANION, Isocitrate dehydrogenase [NADP] cytoplasmic, ...
著者Xie, X, Kulathila, R.
登録日2016-10-24
公開日2017-01-25
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Optimization of 3-Pyrimidin-4-yl-oxazolidin-2-ones as Allosteric and Mutant Specific Inhibitors of IDH1.
ACS Med Chem Lett, 8, 2017
6HNG
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BU of 6hng by Molmil
Peptide-membrane interaction between targeting and lysis
分子名称: LYS-LEU-LEU-LYS-LEU-LEU-LYS-LYS-LEU-LEU-LYS-LEU-LEU-LYS-NHE
著者Schneider, G, Blatter, M, Mueller, A.
登録日2018-09-14
公開日2018-10-24
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献Peptide-membrane interaction between targeting and lysis
To Be Published
6HNE
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BU of 6hne by Molmil
Peptide-membrane interaction between targeting and lysis
分子名称: GLY-LEU-PHE-ASP-ILE-VAL-LYS-LYS-VAL-LEU-LYS-LEU-LEU-LYS-NHE
著者Schneider, G, Blatter, M, Mueller, A.
登録日2018-09-14
公開日2018-10-24
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献Peptide-membrane interaction between targeting and lysis
To Be Published
2TCT
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BU of 2tct by Molmil
THE COMPLEX FORMED BETWEEN TET REPRESSOR AND TETRACYCLINE-MG2+ REVEALS MECHANISM OF ANTIBIOTIC RESISTANCE
分子名称: 7-CHLOROTETRACYCLINE, MAGNESIUM ION, TETRACYCLINE REPRESSOR
著者Hinrichs, W, Kisker, C, Saenger, W.
登録日1995-03-02
公開日1996-04-03
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献The complex formed between Tet repressor and tetracycline-Mg2+ reveals mechanism of antibiotic resistance.
J.Mol.Biol., 247, 1995
2FJ1
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BU of 2fj1 by Molmil
Crystal Structure Analysis of Tet Repressor (class D) in Complex with 7-Chlortetracycline-Nickel(II)
分子名称: 7-CHLOROTETRACYCLINE, CHLORIDE ION, NICKEL (II) ION, ...
著者Orth, P, Saenger, W, Palm, G.J, Hinrichs, W.
登録日2005-12-30
公開日2007-01-09
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Specific binding of divalent metal ions to tetracycline and to the Tet repressor/tetracycline complex.
J.Biol.Inorg.Chem., 13, 2008
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