2E8Z
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 2e8z by Molmil](/molmil-images/mine/2e8z) | Crystal structure of pullulanase type I from Bacillus subtilis str. 168 complexed with alpha-cyclodextrin | Descriptor: | ACETATE ION, AmyX protein, CALCIUM ION, ... | Authors: | Mikami, B, Malle, D, Utsumi, S, Iwamoto, H, Katsuya, Y. | Deposit date: | 2007-01-24 | Release date: | 2008-02-19 | Last modified: | 2023-10-25 | Method: | X-RAY DIFFRACTION (2.2 Å) | Cite: | Crystal structure of pullulanase type I from Bacillus subtilis str. 168 in complex with maltose and alpha-cyclodextrin To be Published
|
|
2E8Y
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 2e8y by Molmil](/molmil-images/mine/2e8y) | Crystal structure of pullulanase type I from Bacillus subtilis str. 168 | Descriptor: | ACETATE ION, AmyX protein, CALCIUM ION, ... | Authors: | Mikami, B, Malle, D, Utsumi, S, Iwamoto, H, Katsuya, Y. | Deposit date: | 2007-01-24 | Release date: | 2008-02-19 | Last modified: | 2023-10-25 | Method: | X-RAY DIFFRACTION (2.11 Å) | Cite: | Crystal structure of pullulanase type I from Bacillus subtilis str. 168
in complex with maltose and alpha-cyclodextrin To be Published
|
|
2E9B
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 2e9b by Molmil](/molmil-images/mine/2e9b) | Crystal structure of pullulanase type I from Bacillus subtilis str. 168 complexed with maltose | Descriptor: | ACETATE ION, AmyX protein, CALCIUM ION, ... | Authors: | Mikami, B, Malle, D, Utsumi, S, Iwamoto, H, Katsuya, Y. | Deposit date: | 2007-01-24 | Release date: | 2008-02-19 | Last modified: | 2023-10-25 | Method: | X-RAY DIFFRACTION (2.3 Å) | Cite: | Crystal structure of pullulanase type I from Bacillus subtilis str. 168 in complex with maltose and alpha-cyclodextrin To be Published
|
|
2FH8
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 2fh8 by Molmil](/molmil-images/mine/2fh8) | Crystal Structure Analysis of Klebsiella pneumoniae pullulanase complexed with isomaltose | Descriptor: | Alpha-dextrin endo-1,6-alpha-glucosidase, CALCIUM ION, alpha-D-glucopyranose-(1-6)-beta-D-glucopyranose | Authors: | Mikami, B, Iwamoto, H, Katsuya, Y, Yoon, H.-J, Demirkan-Sarikaya, E, Malle, D. | Deposit date: | 2005-12-23 | Release date: | 2006-06-13 | Last modified: | 2022-03-09 | Method: | X-RAY DIFFRACTION (1.9 Å) | Cite: | Crystal structure of pullulanase: evidence for parallel binding of oligosaccharides in the active site J.Mol.Biol., 359, 2006
|
|
2FHC
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 2fhc by Molmil](/molmil-images/mine/2fhc) | Crystal Structure Analysis of Klebsiella pneumoniae pullulanase complexed with maltotriose | Descriptor: | Alpha-dextrin endo-1,6-alpha-glucosidase, CALCIUM ION, alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose, ... | Authors: | Mikami, B, Iwamoto, H, Katsuya, Y, Yoon, H.-J, Demirkan-Sarikaya, E, Malle, D. | Deposit date: | 2005-12-23 | Release date: | 2006-06-13 | Last modified: | 2022-03-09 | Method: | X-RAY DIFFRACTION (1.85 Å) | Cite: | Crystal structure of pullulanase: evidence for parallel binding of oligosaccharides in the active site J.Mol.Biol., 359, 2006
|
|
2FH6
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 2fh6 by Molmil](/molmil-images/mine/2fh6) | Crystal Structure Analysis of Klebsiella pneumoniae pullulanase complexed with glucose | Descriptor: | Alpha-dextrin endo-1,6-alpha-glucosidase, CALCIUM ION, alpha-D-glucopyranose | Authors: | Mikami, B, Iwamoto, H, Katsuya, Y, Yoon, H.-J, Demirkan-Sarikaya, E, Malle, D. | Deposit date: | 2005-12-23 | Release date: | 2006-06-13 | Last modified: | 2022-03-09 | Method: | X-RAY DIFFRACTION (1.8 Å) | Cite: | Crystal structure of pullulanase: evidence for parallel binding of oligosaccharides in the active site J.Mol.Biol., 359, 2006
|
|
2FHB
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 2fhb by Molmil](/molmil-images/mine/2fhb) | Crystal Structure Analysis of Klebsiella pneumoniae pullulanase complexed with maltose | Descriptor: | Alpha-dextrin endo-1,6-alpha-glucosidase, CALCIUM ION, alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose | Authors: | Mikami, B, Iwamoto, H, Katsuya, Y, Yoon, H.-J, Demirkan-Sarikaya, E, Malle, D. | Deposit date: | 2005-12-23 | Release date: | 2006-06-13 | Last modified: | 2022-03-09 | Method: | X-RAY DIFFRACTION (1.8 Å) | Cite: | Crystal structure of pullulanase: evidence for parallel binding of oligosaccharides in the active site J.Mol.Biol., 359, 2006
|
|
2FGZ
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 2fgz by Molmil](/molmil-images/mine/2fgz) | Crystal Structure Analysis of apo pullulanase from Klebsiella pneumoniae | Descriptor: | Alpha-dextrin endo-1,6-alpha-glucosidase, CALCIUM ION | Authors: | Mikami, B, Iwamoto, H, Katsuya, Y, Yoon, H.-J, Demirkan-Sarikaya, E, Malle, D. | Deposit date: | 2005-12-23 | Release date: | 2006-06-13 | Last modified: | 2022-03-09 | Method: | X-RAY DIFFRACTION (1.75 Å) | Cite: | Crystal structure of pullulanase: evidence for parallel binding of oligosaccharides in the active site J.Mol.Biol., 359, 2006
|
|
2FHF
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 2fhf by Molmil](/molmil-images/mine/2fhf) | Crystal Structure Analysis of Klebsiella pneumoniae pullulanase complexed with maltotetraose | Descriptor: | Alpha-dextrin endo-1,6-alpha-glucosidase, CALCIUM ION, alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose, ... | Authors: | Mikami, B, Iwamoto, H, Katsuya, Y, Yoon, H.-J, Demirkan-Sarikaya, E, Malle, D. | Deposit date: | 2005-12-23 | Release date: | 2006-06-13 | Last modified: | 2022-03-09 | Method: | X-RAY DIFFRACTION (1.65 Å) | Cite: | Crystal structure of pullulanase: evidence for parallel binding of oligosaccharides in the active site J.Mol.Biol., 359, 2006
|
|
5YNA
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5yna by Molmil](/molmil-images/mine/5yna) | Crystal structure of Pullulanase from Klebsiella pneumoniae complex at 1 mM alpha-cyclodextrin | Descriptor: | ACETATE ION, CALCIUM ION, Cyclohexakis-(1-4)-(alpha-D-glucopyranose), ... | Authors: | Saka, N, Iwamoto, H, Takahashi, N, Mizutani, K, Mikami, B. | Deposit date: | 2017-10-24 | Release date: | 2018-10-24 | Last modified: | 2023-11-22 | Method: | X-RAY DIFFRACTION (1.96 Å) | Cite: | Elucidation of the mechanism of interaction between Klebsiella pneumoniae pullulanase and cyclodextrin Acta Crystallogr D Struct Biol, 74, 2018
|
|
5YNC
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5ync by Molmil](/molmil-images/mine/5ync) | Crystal structure of Pullulanase from Klebsiella pneumoniae complex at 1 mM beta-cyclodextrin | Descriptor: | ACETATE ION, CALCIUM ION, Cycloheptakis-(1-4)-(alpha-D-glucopyranose), ... | Authors: | Saka, N, Iwamoto, H, Takahashi, N, Mizutani, K, Mikami, B. | Deposit date: | 2017-10-24 | Release date: | 2018-10-24 | Last modified: | 2023-11-22 | Method: | X-RAY DIFFRACTION (2.32 Å) | Cite: | Elucidation of the mechanism of interaction between Klebsiella pneumoniae pullulanase and cyclodextrin Acta Crystallogr D Struct Biol, 74, 2018
|
|
5YNE
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5yne by Molmil](/molmil-images/mine/5yne) | Crystal structure of Pullulanase from Klebsiella pneumoniae complex at 10 mM alpha-cyclodextrin | Descriptor: | CALCIUM ION, Cyclohexakis-(1-4)-(alpha-D-glucopyranose), DI(HYDROXYETHYL)ETHER, ... | Authors: | Saka, N, Iwamoto, H, Takahashi, N, Mizutani, K, Mikami, B. | Deposit date: | 2017-10-24 | Release date: | 2018-10-24 | Last modified: | 2023-11-22 | Method: | X-RAY DIFFRACTION (2.199 Å) | Cite: | Elucidation of the mechanism of interaction between Klebsiella pneumoniae pullulanase and cyclodextrin Acta Crystallogr D Struct Biol, 74, 2018
|
|
5YN2
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5yn2 by Molmil](/molmil-images/mine/5yn2) | Crystal structure of apo Pullulanase from Klebsiella pneumoniae in space group P43212 | Descriptor: | CALCIUM ION, MAGNESIUM ION, PulA protein | Authors: | Saka, N, Iwamoto, H, Takahashi, N, Mizutani, K, Mikami, B. | Deposit date: | 2017-10-24 | Release date: | 2018-10-24 | Last modified: | 2023-11-22 | Method: | X-RAY DIFFRACTION (2.301 Å) | Cite: | Elucidation of the mechanism of interaction between Klebsiella pneumoniae pullulanase and cyclodextrin Acta Crystallogr D Struct Biol, 74, 2018
|
|
5YN7
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5yn7 by Molmil](/molmil-images/mine/5yn7) | Crystal structure of Pullulanase from Klebsiella pneumoniae complex at 0.1 mM beta-cyclodextrin | Descriptor: | 1,2-ETHANEDIOL, CALCIUM ION, Cycloheptakis-(1-4)-(alpha-D-glucopyranose), ... | Authors: | Saka, N, Iwamoto, H, Takahashi, N, Mizutani, K, Mikami, B. | Deposit date: | 2017-10-24 | Release date: | 2018-10-24 | Last modified: | 2023-11-22 | Method: | X-RAY DIFFRACTION (2.586 Å) | Cite: | Elucidation of the mechanism of interaction between Klebsiella pneumoniae pullulanase and cyclodextrin Acta Crystallogr D Struct Biol, 74, 2018
|
|
5YND
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5ynd by Molmil](/molmil-images/mine/5ynd) | Crystal structure of Pullulanase from Klebsiella pneumoniae complex at 1 mM gamma-cyclodextrin | Descriptor: | CALCIUM ION, DI(HYDROXYETHYL)ETHER, DUF3372 domain-containing protein, ... | Authors: | Saka, N, Iwamoto, H, Takahashi, N, Mizutani, K, Mikami, B. | Deposit date: | 2017-10-24 | Release date: | 2018-10-24 | Last modified: | 2023-11-22 | Method: | X-RAY DIFFRACTION (2.227 Å) | Cite: | Elucidation of the mechanism of interaction between Klebsiella pneumoniae pullulanase and cyclodextrin Acta Crystallogr D Struct Biol, 74, 2018
|
|
5YNH
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5ynh by Molmil](/molmil-images/mine/5ynh) | Crystal structure of Pullulanase from Klebsiella pneumoniae complex at 10 mM gamma-cyclodextrin | Descriptor: | CALCIUM ION, Cyclooctakis-(1-4)-(alpha-D-glucopyranose), GLYCEROL, ... | Authors: | Saka, N, Iwamoto, H, Takahashi, N, Mizutani, K, Mikami, B. | Deposit date: | 2017-10-24 | Release date: | 2018-10-24 | Last modified: | 2023-11-22 | Method: | X-RAY DIFFRACTION (2.05 Å) | Cite: | Elucidation of the mechanism of interaction between Klebsiella pneumoniae pullulanase and cyclodextrin Acta Crystallogr D Struct Biol, 74, 2018
|
|
6J4H
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 6j4h by Molmil](/molmil-images/mine/6j4h) | Crystal Structure of maltotriose-complex of PulA-G680L mutant from Klebsiella pneumoniae | Descriptor: | CALCIUM ION, GLYCEROL, MAGNESIUM ION, ... | Authors: | Saka, N, Iwamoto, H, Takahashi, N, Mizutani, K, Mikami, B. | Deposit date: | 2019-01-09 | Release date: | 2019-09-18 | Last modified: | 2020-07-29 | Method: | X-RAY DIFFRACTION (1.641 Å) | Cite: | Relationship between the induced-fit loop and the activity of Klebsiella pneumoniae pullulanase. Acta Crystallogr D Struct Biol, 75, 2019
|
|
6J35
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 6j35 by Molmil](/molmil-images/mine/6j35) | Crystal structure of ligand-free of PulA-G680L mutant from Klebsiella pneumoniae | Descriptor: | CALCIUM ION, GLYCEROL, MAGNESIUM ION, ... | Authors: | Saka, N, Iwamoto, H, Takahashi, N, Mizutani, K, Mikami, B. | Deposit date: | 2019-01-09 | Release date: | 2019-09-18 | Last modified: | 2023-11-22 | Method: | X-RAY DIFFRACTION (1.839 Å) | Cite: | Relationship between the induced-fit loop and the activity of Klebsiella pneumoniae pullulanase. Acta Crystallogr D Struct Biol, 75, 2019
|
|
6J33
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 6j33 by Molmil](/molmil-images/mine/6j33) | Crystal structure of ligand-free of PulA from Klebsiella pneumoniae | Descriptor: | ACETATE ION, CALCIUM ION, MAGNESIUM ION, ... | Authors: | Saka, N, Iwamoto, H, Takahashi, N, Mizutani, K, Mikami, B. | Deposit date: | 2019-01-09 | Release date: | 2019-09-18 | Last modified: | 2023-11-22 | Method: | X-RAY DIFFRACTION (1.297 Å) | Cite: | Relationship between the induced-fit loop and the activity of Klebsiella pneumoniae pullulanase. Acta Crystallogr D Struct Biol, 75, 2019
|
|
6J34
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 6j34 by Molmil](/molmil-images/mine/6j34) | Crystal Structure of maltotriose-complex of PulA from Klebsiella pneumoniae | Descriptor: | ACETATE ION, GLYCEROL, MAGNESIUM ION, ... | Authors: | Saka, N, Iwamoto, H, Takahashi, N, Mizutani, K, Mikami, B. | Deposit date: | 2019-01-09 | Release date: | 2019-09-18 | Last modified: | 2023-11-22 | Method: | X-RAY DIFFRACTION (1.498 Å) | Cite: | Relationship between the induced-fit loop and the activity of Klebsiella pneumoniae pullulanase. Acta Crystallogr D Struct Biol, 75, 2019
|
|
7KXD
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7kxd by Molmil](/molmil-images/mine/7kxd) | |
7KXE
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7kxe by Molmil](/molmil-images/mine/7kxe) | |
7KXF
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7kxf by Molmil](/molmil-images/mine/7kxf) | |
5S9R
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5s9r by Molmil](/molmil-images/mine/5s9r) | CRYSTAL STRUCTURE OF THE FIRST BROMODOMAIN OF HUMAN BRD4 IN COMPLEX WITH BMS-986158, 2-{3-(1,4-dimethyl-1H-1,2,3-triazol-5-yl)-5-[(S)-(oxan-4-yl)(phenyl)methyl]-5H-pyrido[3,2-b]indol-7-yl}propan-2-ol | Descriptor: | 1,2-ETHANEDIOL, 2-{3-(1,4-dimethyl-1H-1,2,3-triazol-5-yl)-5-[(S)-(oxan-4-yl)(phenyl)methyl]-5H-pyrido[3,2-b]indol-7-yl}propan-2-ol, Bromodomain-containing protein 4, ... | Authors: | Sheriff, S. | Deposit date: | 2021-04-01 | Release date: | 2021-09-29 | Last modified: | 2024-05-22 | Method: | X-RAY DIFFRACTION (1.85 Å) | Cite: | Discovery and Preclinical Pharmacology of an Oral Bromodomain and Extra-Terminal (BET) Inhibitor Using Scaffold-Hopping and Structure-Guided Drug Design. J.Med.Chem., 64, 2021
|
|
5S9O
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5s9o by Molmil](/molmil-images/mine/5s9o) | CRYSTAL STRUCTURE OF THE HUMAN BRD2 BD1 BROMODOMAIN IN COMPLEX WITH 9-(cyclopropylmethyl)-7-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-3-(3,5-dimethyl-1,2-oxazol-4-yl)-9H-carbazole-1-carboxamide | Descriptor: | 1,2-ETHANEDIOL, 9-(cyclopropylmethyl)-7-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-3-(3,5-dimethyl-1,2-oxazol-4-yl)-9H-carbazole-1-carboxamide, Bromodomain-containing protein 2 | Authors: | Sheriff, S. | Deposit date: | 2021-04-01 | Release date: | 2021-09-29 | Last modified: | 2024-05-22 | Method: | X-RAY DIFFRACTION (2.49 Å) | Cite: | Discovery and Preclinical Pharmacology of an Oral Bromodomain and Extra-Terminal (BET) Inhibitor Using Scaffold-Hopping and Structure-Guided Drug Design. J.Med.Chem., 64, 2021
|
|