1OP8
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![BU of 1op8 by Molmil](/molmil-images/mine/1op8) | Crystal Structure of Human Granzyme A | Descriptor: | Granzyme A, SULFATE ION | Authors: | Hink-Schauer, C, Estebanez-Perpina, E, Bode, W, Jenne, D. | Deposit date: | 2003-03-05 | Release date: | 2003-07-01 | Last modified: | 2011-07-13 | Method: | X-RAY DIFFRACTION (2.5 Å) | Cite: | Crystal structure of the apoptosis-inducing human granzyme A dimer NAT.STRUCT.BIOL., 10, 2003
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6IC6
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![BU of 6ic6 by Molmil](/molmil-images/mine/6ic6) | Human cathepsin-C in complex with cyclopropyl peptidyl nitrile inhibitor 1 | Descriptor: | (2~{S})-~{N}-[(1~{R},2~{R})-1-(aminomethyl)-2-[4-[4-(trifluoromethyl)phenyl]phenyl]cyclopropyl]-2-azanyl-butanamide, 2-acetamido-2-deoxy-beta-D-glucopyranose, CHLORIDE ION, ... | Authors: | Hakansson, M, Logan, D.T, Korkmaz, B, Lesner, A, Wysocka, M, Gieldon, A, Gauthier, F, Jenne, D, Lauritzen, C, Pedersen, J. | Deposit date: | 2018-12-02 | Release date: | 2019-04-24 | Last modified: | 2024-05-01 | Method: | X-RAY DIFFRACTION (1.898 Å) | Cite: | Structure-based design and in vivo anti-arthritic activity evaluation of a potent dipeptidyl cyclopropyl nitrile inhibitor of cathepsin C. Biochem. Pharmacol., 164, 2019
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6IC7
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![BU of 6ic7 by Molmil](/molmil-images/mine/6ic7) | Human cathepsin-C in complex with dipeptidyl cyclopropyl nitrile inhibitor 3 | Descriptor: | 1-azanyl-~{N}-[(1~{R},2~{R})-1-cyano-2-[4-[4-(4-methylpiperazin-1-yl)sulfonylphenyl]phenyl]cyclopropyl]cyclohexane-1-carboxamide, 2-acetamido-2-deoxy-beta-D-glucopyranose, CHLORIDE ION, ... | Authors: | Hakansson, M, Logan, D.T, Korkmaz, B, Lesner, A, Wysocka, M, Gieldon, A, Gauthier, F, Jenne, D, Lauritzen, C, Pedersen, J. | Deposit date: | 2018-12-02 | Release date: | 2019-04-24 | Last modified: | 2020-07-29 | Method: | X-RAY DIFFRACTION (2 Å) | Cite: | Structure-based design and in vivo anti-arthritic activity evaluation of a potent dipeptidyl cyclopropyl nitrile inhibitor of cathepsin C. Biochem. Pharmacol., 164, 2019
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6IC5
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![BU of 6ic5 by Molmil](/molmil-images/mine/6ic5) | Human cathepsin-C in complex with dipeptidyl cyclopropyl nitrile inhibitor 2 | Descriptor: | (2~{S})-2-azanyl-~{N}-[(1~{R},2~{R})-1-(iminomethyl)-2-[4-[4-(4-methylpiperazin-1-yl)sulfonylphenyl]phenyl]cyclopropyl]-3-thiophen-2-yl-propanamide, 2-acetamido-2-deoxy-beta-D-glucopyranose, CHLORIDE ION, ... | Authors: | Hakansson, M, Logan, D.T, Korkmaz, B, Lesner, A, Wysocka, M, Gieldon, A, Gauthier, F, Jenne, D, Lauritzen, C, Pedersen, J. | Deposit date: | 2018-12-02 | Release date: | 2019-04-24 | Last modified: | 2020-07-29 | Method: | X-RAY DIFFRACTION (2 Å) | Cite: | Structure-based design and in vivo anti-arthritic activity evaluation of a potent dipeptidyl cyclopropyl nitrile inhibitor of cathepsin C. Biochem. Pharmacol., 164, 2019
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4DZ3
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![BU of 4dz3 by Molmil](/molmil-images/mine/4dz3) | |
4DZ2
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![BU of 4dz2 by Molmil](/molmil-images/mine/4dz2) | |
4FN2
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![BU of 4fn2 by Molmil](/molmil-images/mine/4fn2) | |
4GGQ
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![BU of 4ggq by Molmil](/molmil-images/mine/4ggq) | |
4GIV
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![BU of 4giv by Molmil](/molmil-images/mine/4giv) | |
4G50
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![BU of 4g50 by Molmil](/molmil-images/mine/4g50) | |
3UF8
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![BU of 3uf8 by Molmil](/molmil-images/mine/3uf8) | |
3VAW
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![BU of 3vaw by Molmil](/molmil-images/mine/3vaw) | |
3UQB
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![BU of 3uqb by Molmil](/molmil-images/mine/3uqb) | |
3UQA
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![BU of 3uqa by Molmil](/molmil-images/mine/3uqa) | |