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1A0L
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HUMAN BETA-TRYPTASE: A RING-LIKE TETRAMER WITH ACTIVE SITES FACING A CENTRAL PORE
分子名称: (2S)-3-(4-carbamimidoylphenyl)-2-hydroxypropanoic acid, BETA-TRYPTASE
著者Pereira, P.J.B, Bergner, A, Macedo-Ribeiro, S, Huber, R, Matschiner, G, Fritz, H, Sommerhoff, C.P, Bode, W.
登録日1997-12-03
公開日1999-03-23
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Human beta-tryptase is a ring-like tetramer with active sites facing a central pore.
Nature, 392, 1998
1BX7
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HIRUSTASIN FROM HIRUDO MEDICINALIS AT 1.2 ANGSTROMS
分子名称: HIRUSTASIN, SULFATE ION
著者Uson, I, Sheldrick, G.M, De La Fortelle, E, Bricogne, G, Di Marco, S, Priestle, J.P, Gruetter, M.G, Mittl, P.R.E.
登録日1998-10-14
公開日1999-04-27
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (1.2 Å)
主引用文献The 1.2 A crystal structure of hirustasin reveals the intrinsic flexibility of a family of highly disulphide-bridged inhibitors.
Structure Fold.Des., 7, 1999
1LDT
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COMPLEX OF LEECH-DERIVED TRYPTASE INHIBITOR WITH PORCINE TRYPSIN
分子名称: CALCIUM ION, TRYPSIN, TRYPTASE INHIBITOR
著者Stubbs, M.T.
登録日1997-05-15
公開日1998-05-20
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献The three-dimensional structure of recombinant leech-derived tryptase inhibitor in complex with trypsin. Implications for the structure of human mast cell tryptase and its inhibition.
J.Biol.Chem., 272, 1997
1HIA
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KALLIKREIN COMPLEXED WITH HIRUSTASIN
分子名称: HIRUSTASIN, KALLIKREIN
著者Mittl, P, Di Marco, S, Gruetter, M.
登録日1996-12-12
公開日1997-12-24
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献A new structural class of serine protease inhibitors revealed by the structure of the hirustasin-kallikrein complex.
Structure, 5, 1997
1CSE
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THE HIGH-RESOLUTION X-RAY CRYSTAL STRUCTURE OF THE COMPLEX FORMED BETWEEN SUBTILISIN CARLSBERG AND EGLIN C, AN ELASTASE INHIBITOR FROM THE LEECH HIRUDO MEDICINALIS. STRUCTURAL ANALYSIS, SUBTILISIN STRUCTURE AND INTERFACE GEOMETRY
分子名称: CALCIUM ION, EGLIN C, SUBTILISIN CARLSBERG
著者Bode, W.
登録日1988-06-03
公開日1988-07-16
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.2 Å)
主引用文献The high-resolution X-ray crystal structure of the complex formed between subtilisin Carlsberg and eglin c, an elastase inhibitor from the leech Hirudo medicinalis. Structural analysis, subtilisin structure and interface geometry.
Eur.J.Biochem., 166, 1987
1AN1
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LEECH-DERIVED TRYPTASE INHIBITOR/TRYPSIN COMPLEX
分子名称: CALCIUM ION, TRYPSIN, TRYPTASE INHIBITOR
著者Priestle, J.P, Di Marco, S.
登録日1997-06-26
公開日1998-07-01
最終更新日2023-08-02
実験手法X-RAY DIFFRACTION (2.03 Å)
主引用文献Structure of the complex of leech-derived tryptase inhibitor (LDTI) with trypsin and modeling of the LDTI-tryptase system.
Structure, 5, 1997
1BX8
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HIRUSTASIN FROM HIRUDO MEDICINALIS AT 1.4 ANGSTROMS
分子名称: HIRUSTASIN, SULFATE ION
著者Uson, I, Sheldrick, G.M, De La Fortelle, E, Bricogne, G, Di Marco, S, Priestle, J.P, Gruetter, M.G, Mittl, P.R.E.
登録日1998-10-14
公開日1999-04-27
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献The 1.2 A crystal structure of hirustasin reveals the intrinsic flexibility of a family of highly disulphide-bridged inhibitors.
Structure Fold.Des., 7, 1999
1C9P
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COMPLEX OF BDELLASTASIN WITH PORCINE TRYPSIN
分子名称: BDELLASTASIN, CALCIUM ION, TRYPSIN
著者Rester, U.
登録日1999-08-03
公開日2000-08-03
最終更新日2021-11-03
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Structure of the complex of the antistasin-type inhibitor bdellastasin with trypsin and modelling of the bdellastasin-microplasmin system.
J.Mol.Biol., 293, 1999
1TFX
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COMPLEX OF THE SECOND KUNITZ DOMAIN OF TISSUE FACTOR PATHWAY INHIBITOR WITH PORCINE TRYPSIN
分子名称: CALCIUM ION, TISSUE FACTOR PATHWAY INHIBITOR, TRYPSIN
著者Stubbs, M.T, Huber, R.
登録日1997-01-21
公開日1998-01-21
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献The second Kunitz domain of human tissue factor pathway inhibitor: cloning, structure determination and interaction with factor Xa.
J.Mol.Biol., 269, 1997
1SBN
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BU of 1sbn by Molmil
REFINED CRYSTAL STRUCTURES OF SUBTILISIN NOVO IN COMPLEX WITH WILD-TYPE AND TWO MUTANT EGLINS. COMPARISON WITH OTHER SERINE PROTEINASE INHIBITOR COMPLEXES
分子名称: CALCIUM ION, EGLIN C, SUBTILISIN NOVO BPN'
著者Gruetter, M.G, Heinz, D.W, Priestle, J.P.
登録日1991-12-20
公開日1994-01-31
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Refined crystal structures of subtilisin novo in complex with wild-type and two mutant eglins. Comparison with other serine proteinase inhibitor complexes.
J.Mol.Biol., 217, 1991
1SIB
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REFINED CRYSTAL STRUCTURES OF SUBTILISIN NOVO IN COMPLEX WITH WILD-TYPE AND TWO MUTANT EGLINS. COMPARISON WITH OTHER SERINE PROTEINASE INHIBITOR COMPLEXES
分子名称: CALCIUM ION, EGLIN C, SUBTILISIN NOVO BPN'
著者Gruetter, M.G, Heinz, D.W, Priestle, J.P.
登録日1993-08-02
公開日1993-10-31
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Refined crystal structures of subtilisin novo in complex with wild-type and two mutant eglins. Comparison with other serine proteinase inhibitor complexes.
J.Mol.Biol., 217, 1991
1EJA
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STRUCTURE OF PORCINE TRYPSIN COMPLEXED WITH BDELLASTASIN, AN ANTISTASIN-TYPE INHIBITOR
分子名称: BDELLASTASIN, SODIUM ION, TRYPSIN
著者Rester, U, Moser, M, Huber, R, Bode, W.
登録日2000-03-02
公開日2001-03-02
最終更新日2017-10-04
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献L-Isoaspartate 115 of porcine beta-trypsin promotes crystallization of its complex with bdellastasin.
Acta Crystallogr.,Sect.D, 56, 2000

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