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4P8P
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BU of 4p8p by Molmil
Crystal structure of M. tuberculosis DprE1 in complex with the non-covalent inhibitor QN127
Descriptor: (2R)-2-{[(2R)-2-{[(2R)-2-hydroxypropyl]oxy}propyl]oxy}propan-1-ol, 3-[(4-chlorobenzyl)amino]-6-(trifluoromethyl)quinoxaline-2-carboxylic acid, FLAVIN-ADENINE DINUCLEOTIDE, ...
Authors:Neres, J, Pojer, F, Cole, S.T.
Deposit date:2014-03-31
Release date:2014-12-10
Last modified:2023-12-27
Method:X-RAY DIFFRACTION (2.2 Å)
Cite:2-Carboxyquinoxalines Kill Mycobacterium tuberculosis through Noncovalent Inhibition of DprE1.
Acs Chem.Biol., 10, 2015
4P8Y
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BU of 4p8y by Molmil
Crystal structure of M. tuberculosis DprE1 in complex with the non-covalent inhibitor Ty21c
Descriptor: 3-[(4-methoxybenzyl)amino]-6-(trifluoromethyl)quinoxaline-2-carboxylic acid, FLAVIN-ADENINE DINUCLEOTIDE, IMIDAZOLE, ...
Authors:Neres, J, Pojer, F, Cole, S.T.
Deposit date:2014-04-01
Release date:2014-12-10
Last modified:2023-12-27
Method:X-RAY DIFFRACTION (2.01 Å)
Cite:2-Carboxyquinoxalines Kill Mycobacterium tuberculosis through Noncovalent Inhibition of DprE1.
Acs Chem.Biol., 10, 2015
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