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4AEL
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BU of 4ael by Molmil
PDE10A in complex with the inhibitor AZ5
分子名称: 2-(2'-ETHOXYBIPHENYL-4-YL)-4-HYDROXY-1,6-NAPHTHYRIDINE-3-CARBONITRILE, CAMP AND CAMP-INHIBITED CGMP 3', 5'-CYCLIC PHOSPHODIESTERASE 10A, ...
著者Bauer, U, Giordanetto, F, Bauer, M, OMahony, G, Johansson, K.E, Knecht, W, Hartleib-Geschwindner, J, Toppner Carlsson, E, Enroth, C, Sjogren, T.
登録日2012-01-11
公開日2012-01-25
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Discovery of 4-Hydroxy-1,6-Naphthyridine-3-Carbonitrile Derivatives as Novel Pde10A Inhibitors.
Bioorg.Med.Chem.Lett., 22, 2012
1W9C
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BU of 1w9c by Molmil
Proteolytic fragment of CRM1 spanning six C-terminal HEAT repeats
分子名称: CRM1 PROTEIN
著者Petosa, C, Schoehn, G, Askjaer, P, Bauer, U, Moulin, M, Steuerwald, U, Soler-Lopez, M, Baudin, F, Mattaj, I.W, Muller, C.W.
登録日2004-10-08
公開日2004-12-03
最終更新日2019-11-13
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Architecture of Crm1-Exportin 1 Suggests How Cooperativity is Achieved During Formation of a Nuclear Export Complex
Mol.Cell, 16, 2004
6BVU
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BU of 6bvu by Molmil
SFTI-HFRW-1
分子名称: Trypsin inhibitor 1 HFRW-1
著者Schroeder, C.I.
登録日2017-12-13
公開日2018-12-19
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献Development of Novel Melanocortin Receptor Agonists Based on the Cyclic Peptide Framework of Sunflower Trypsin Inhibitor-1.
J.Med.Chem., 61, 2018
6BVW
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BU of 6bvw by Molmil
SFTI-HFRW-3
分子名称: Trypsin inhibitor 1 HFRW-3
著者Schroeder, C.I.
登録日2017-12-14
公開日2018-12-19
最終更新日2023-11-15
実験手法SOLUTION NMR
主引用文献Development of Novel Melanocortin Receptor Agonists Based on the Cyclic Peptide Framework of Sunflower Trypsin Inhibitor-1.
J.Med.Chem., 61, 2018
6BVX
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BU of 6bvx by Molmil
SFTI-HFRW-2
分子名称: Trypsin inhibitor 1 HFRW-2
著者Schroeder, C.I.
登録日2017-12-14
公開日2018-12-19
最終更新日2023-11-15
実験手法SOLUTION NMR
主引用文献Development of Novel Melanocortin Receptor Agonists Based on the Cyclic Peptide Framework of Sunflower Trypsin Inhibitor-1.
J.Med.Chem., 61, 2018
6BVY
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BU of 6bvy by Molmil
SFTI-HFRW-4
分子名称: Trypsin inhibitor 1 HFRW-4
著者Schroeder, C.I, White, A.
登録日2017-12-14
公開日2018-04-18
最終更新日2023-11-15
実験手法SOLUTION NMR
主引用文献Development of Novel Melanocortin Receptor Agonists Based on the Cyclic Peptide Framework of Sunflower Trypsin Inhibitor-1.
J. Med. Chem., 61, 2018

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件を2024-04-24に公開中

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