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6PXR
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BU of 6pxr by Molmil
Anti-TAU BIIB092 FAB with TAU peptide
分子名称: Microtubule-associated protein tau, gosuranemab Fab, heavy chain, ...
著者Arndt, J.W, Quan, C.
登録日2019-07-26
公開日2020-07-29
最終更新日2021-02-10
実験手法X-RAY DIFFRACTION (1.556 Å)
主引用文献Characterization of tau binding by gosuranemab.
Neurobiol.Dis., 146, 2020
6CR1
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BU of 6cr1 by Molmil
adalimumab EFab
分子名称: DI(HYDROXYETHYL)ETHER, Heavy chain of adalimumab EFab (VH-IgE CH2), Light chain of adalimumab EFab (VL-IgE CH2), ...
著者Arndt, J.W.
登録日2018-03-16
公開日2018-09-26
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (1.521 Å)
主引用文献EFab domain substitution as a solution to the light-chain pairing problem of bispecific antibodies.
MAbs, 10, 2018
1VKH
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BU of 1vkh by Molmil
CRYSTAL STRUCTURE OF A PUTATIVE SERINE HYDROLASE (YDR428C) FROM SACCHAROMYCES CEREVISIAE AT 1.85 A RESOLUTION
分子名称: CHLORIDE ION, GLYCEROL, putative serine hydrolase
著者Joint Center for Structural Genomics (JCSG)
登録日2004-05-20
公開日2004-06-08
最終更新日2023-01-25
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Crystal structure of an alpha/beta serine hydrolase (YDR428C) from Saccharomyces cerevisiae at 1.85 A resolution
Proteins, 58, 2005
3QDD
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BU of 3qdd by Molmil
HSP90A N-terminal domain in complex with BIIB021
分子名称: 6-chloro-9-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-9H-purin-2-amine, Heat shock protein HSP 90-alpha
著者Arndt, J.W, Biamonte, M.A.
登録日2011-01-18
公開日2012-07-18
最終更新日2022-10-05
実験手法X-RAY DIFFRACTION (1.79 Å)
主引用文献EC144 Is a Potent Inhibitor of the Heat Shock Protein 90.
J.Med.Chem., 55, 2012
3PWY
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BU of 3pwy by Molmil
Crystal structure of an extender (SPD28345)-modified human PDK1 complex 2
分子名称: 3-phosphoinositide-dependent protein kinase 1, N-[2-({6-[(2-sulfanylethyl)amino]pyrimidin-4-yl}amino)ethyl]propanamide
著者Elling, R.A, Penny, D.M, Simmons, R.L, Erlanson, D.A, Romanowski, M.J.
登録日2010-12-09
公開日2011-04-20
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (3.5 Å)
主引用文献Discovery of a potent and highly selective PDK1 inhibitor via fragment-based drug discovery.
Bioorg.Med.Chem.Lett., 21, 2011
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