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6VND
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BU of 6vnd by Molmil
Quaternary Complex of human dihydroorotate dehydrogenase (DHODH) with flavin mononucleotide (FMN), orotic acid and AG-636
分子名称: 1-methyl-5-(2'-methyl[1,1'-biphenyl]-4-yl)-1H-benzotriazole-7-carboxylic acid, ACETATE ION, CHLORIDE ION, ...
著者Padyana, A, Jin, L.
登録日2020-01-29
公開日2020-11-04
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (1.97 Å)
主引用文献Selective Vulnerability to Pyrimidine Starvation in Hematologic Malignancies Revealed by AG-636, a Novel Clinical-Stage Inhibitor of Dihydroorotate Dehydrogenase.
Mol.Cancer Ther., 19, 2020
3UNW
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BU of 3unw by Molmil
Crystal Structure of Human GAC in Complex with Glutamate
分子名称: GLUTAMIC ACID, Glutaminase kidney isoform, mitochondrial
著者DeLaBarre, B, Gross, S, Cheng, F, Gao, Y, Jha, A, Jiang, F, Song, J.J, Wie, W, Hurov, J.
登録日2011-11-16
公開日2011-12-07
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.56 Å)
主引用文献Full-length human glutaminase in complex with an allosteric inhibitor.
Biochemistry, 50, 2011

218853

件を2024-04-24に公開中

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