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4QP8
Crystal Structure of ERK2 in complex with 2-(1H-pyrazol-4-yl)-7-(pyridin-3-yl)-5H-pyrrolo[2,3-b]pyrazine
Descriptor:
2-(1H-pyrazol-4-yl)-7-(pyridin-3-yl)-5H-pyrrolo[2,3-b]pyrazine, Mitogen-activated protein kinase 1
Authors:
Yin, J
,
Wang, W.
Deposit date:
2014-06-22
Release date:
2015-09-23
Last modified:
2024-02-28
Method:
X-RAY DIFFRACTION (2.446 Å)
Cite:
Fragment-based discovery of potent ERK2 pyrrolopyrazine inhibitors.
Bioorg.Med.Chem.Lett., 25, 2015
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PDB entries from 2024-07-03