7L3M
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![BU of 7l3m by Molmil](/molmil-images/mine/7l3m) | PEPCK MMQX structure 40ms post-mixing with oxaloacetic acid | Descriptor: | CARBON DIOXIDE, GUANOSINE-5'-DIPHOSPHATE, MANGANESE (II) ION, ... | Authors: | Clinger, J.A, Moreau, D.W, McLeod, M.J, Holyoak, T, Thorne, R.E. | Deposit date: | 2020-12-18 | Release date: | 2021-10-13 | Last modified: | 2023-10-18 | Method: | X-RAY DIFFRACTION (2.07 Å) | Cite: | Millisecond mix-and-quench crystallography (MMQX) enables time-resolved studies of PEPCK with remote data collection. Iucrj, 8, 2021
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7L3V
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![BU of 7l3v by Molmil](/molmil-images/mine/7l3v) | PEPCK MMQX structure 120ms post-mixing with oxaloacetic acid | Descriptor: | CARBON DIOXIDE, GUANOSINE-5'-DIPHOSPHATE, MANGANESE (II) ION, ... | Authors: | Clinger, J.A, Moreau, D.W, McLeod, M.J, Holyoak, T, Thorne, R.E. | Deposit date: | 2020-12-18 | Release date: | 2021-10-13 | Last modified: | 2023-10-18 | Method: | X-RAY DIFFRACTION (1.98 Å) | Cite: | Millisecond mix-and-quench crystallography (MMQX) enables time-resolved studies of PEPCK with remote data collection. Iucrj, 8, 2021
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4YWD
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![BU of 4ywd by Molmil](/molmil-images/mine/4ywd) | Structure of rat cytosolic pepck in complex with 2,3-Pyridine dicarboxylic acid | Descriptor: | MANGANESE (II) ION, Phosphoenolpyruvate carboxykinase, cytosolic [GTP], ... | Authors: | Balan, M.D, Johnson, T.A, Mcleod, M.J, Lotosky, W.R, Holyoak, T. | Deposit date: | 2015-03-20 | Release date: | 2015-09-23 | Last modified: | 2023-09-27 | Method: | X-RAY DIFFRACTION (2.1 Å) | Cite: | Inhibition and Allosteric Regulation of Monomeric Phosphoenolpyruvate Carboxykinase by 3-Mercaptopicolinic Acid. Biochemistry, 54, 2015
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3DT4
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![BU of 3dt4 by Molmil](/molmil-images/mine/3dt4) | |
3DTB
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![BU of 3dtb by Molmil](/molmil-images/mine/3dtb) | |
3DT2
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![BU of 3dt2 by Molmil](/molmil-images/mine/3dt2) | |
3DT7
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![BU of 3dt7 by Molmil](/molmil-images/mine/3dt7) | |
8E1U
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![BU of 8e1u by Molmil](/molmil-images/mine/8e1u) | |
8DD6
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![BU of 8dd6 by Molmil](/molmil-images/mine/8dd6) | SARS-CoV-2 Main Protease (Mpro) H163A Mutant in Complex with GC376 | Descriptor: | (1S,2S)-2-({N-[(benzyloxy)carbonyl]-L-leucyl}amino)-1-hydroxy-3-[(3S)-2-oxopyrrolidin-3-yl]propane-1-sulfonic acid, DIMETHYL SULFOXIDE, ORF1a polyprotein | Authors: | Tran, N, McLeod, M.J, Kalyaanamoorthy, S, Ganesan, A, Holyoak, T. | Deposit date: | 2022-06-17 | Release date: | 2023-09-27 | Method: | X-RAY DIFFRACTION (2.3 Å) | Cite: | The H163A mutation unravels an oxidized conformation of the SARS-CoV-2 main protease. Nat Commun, 14, 2023
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2ID4
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![BU of 2id4 by Molmil](/molmil-images/mine/2id4) | |
4GMM
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![BU of 4gmm by Molmil](/molmil-images/mine/4gmm) | |
4GMW
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![BU of 4gmw by Molmil](/molmil-images/mine/4gmw) | |
4GMU
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![BU of 4gmu by Molmil](/molmil-images/mine/4gmu) | |
4GNQ
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![BU of 4gnq by Molmil](/molmil-images/mine/4gnq) | |
4GNP
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![BU of 4gnp by Molmil](/molmil-images/mine/4gnp) | |
4GNO
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![BU of 4gno by Molmil](/molmil-images/mine/4gno) | |
4GNM
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![BU of 4gnm by Molmil](/molmil-images/mine/4gnm) | |
4GNL
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![BU of 4gnl by Molmil](/molmil-images/mine/4gnl) | |
4GMZ
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![BU of 4gmz by Molmil](/molmil-images/mine/4gmz) | |
2QF2
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![BU of 2qf2 by Molmil](/molmil-images/mine/2qf2) | Rat cytosolic PEPCK in complex with oxaloacetic acid and GDP. | Descriptor: | GUANOSINE-5'-DIPHOSPHATE, MANGANESE (II) ION, OXALOACETATE ION, ... | Authors: | Sullivan, S.M, Holyoak, T. | Deposit date: | 2007-06-26 | Release date: | 2007-08-28 | Last modified: | 2023-11-15 | Method: | X-RAY DIFFRACTION (1.65 Å) | Cite: | Structures of rat cytosolic PEPCK: insight into the mechanism of phosphorylation and decarboxylation of oxaloacetic acid. Biochemistry, 46, 2007
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2QF1
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![BU of 2qf1 by Molmil](/molmil-images/mine/2qf1) | Rat cytosolic PEPCK in complex with oxaloacetic acid. | Descriptor: | MANGANESE (II) ION, OXALOACETATE ION, Phosphoenolpyruvate carboxykinase, ... | Authors: | Sullivan, S.M, Holyoak, T. | Deposit date: | 2007-06-26 | Release date: | 2007-08-21 | Last modified: | 2023-08-30 | Method: | X-RAY DIFFRACTION (1.8 Å) | Cite: | Structures of rat cytosolic PEPCK: insight into the mechanism of phosphorylation and decarboxylation of oxaloacetic acid. Biochemistry, 46, 2007
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2RKA
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![BU of 2rka by Molmil](/molmil-images/mine/2rka) | The Structure of rat cytosolic PEPCK in complex with phosphoglycolate | Descriptor: | 2-PHOSPHOGLYCOLIC ACID, MANGANESE (II) ION, Phosphoenolpyruvate carboxykinase, ... | Authors: | Sullivan, S.M, Stiffin, R.M, Carlson, G.M, Holyoak, T. | Deposit date: | 2007-10-16 | Release date: | 2008-01-29 | Last modified: | 2024-02-21 | Method: | X-RAY DIFFRACTION (1.95 Å) | Cite: | Differential Inhibition of Cytosolic PEPCK by Substrate Analogues. Kinetic and Structural Characterization of Inhibitor Recognition. Biochemistry, 47, 2008
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2RKE
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![BU of 2rke by Molmil](/molmil-images/mine/2rke) | The Structure of rat cytosolic PEPCK in complex with sulfoacetate. | Descriptor: | MANGANESE (II) ION, Phosphoenolpyruvate carboxykinase, cytosolic [GTP], ... | Authors: | Sullivan, S.M, Stiffin, R.M, Carlson, G.M, Holyoak, T. | Deposit date: | 2007-10-16 | Release date: | 2008-01-29 | Last modified: | 2024-02-21 | Method: | X-RAY DIFFRACTION (1.8 Å) | Cite: | Differential Inhibition of Cytosolic PEPCK by Substrate Analogues. Kinetic and Structural Characterization of Inhibitor Recognition. Biochemistry, 47, 2008
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2RK7
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![BU of 2rk7 by Molmil](/molmil-images/mine/2rk7) | The Structure of rat cytosolic PEPCK in complex with oxalate | Descriptor: | MANGANESE (II) ION, OXALATE ION, Phosphoenolpyruvate carboxykinase, ... | Authors: | Sullivan, S.M, Stiffin, R.M, Carlson, G.M, Holyoak, T. | Deposit date: | 2007-10-16 | Release date: | 2008-01-29 | Last modified: | 2024-02-21 | Method: | X-RAY DIFFRACTION (1.9 Å) | Cite: | Differential Inhibition of Cytosolic PEPCK by Substrate Analogues. Kinetic and Structural Characterization of Inhibitor Recognition. Biochemistry, 47, 2008
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2QEW
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![BU of 2qew by Molmil](/molmil-images/mine/2qew) | Rat cytosolic PEPCK, in complex with manganese ion. | Descriptor: | MANGANESE (II) ION, Phosphoenolpyruvate carboxykinase, cytosolic [GTP], ... | Authors: | Sullivan, S.M, Holyoak, T. | Deposit date: | 2007-06-26 | Release date: | 2007-08-21 | Last modified: | 2023-08-30 | Method: | X-RAY DIFFRACTION (1.8 Å) | Cite: | Structures of rat cytosolic PEPCK: insight into the mechanism of phosphorylation and decarboxylation of oxaloacetic acid. Biochemistry, 46, 2007
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